BR0317525A - Compostos pirazol acìclico, composição terapêutica e farmacêutica, kit, bem como respectivos usos - Google Patents
Compostos pirazol acìclico, composição terapêutica e farmacêutica, kit, bem como respectivos usosInfo
- Publication number
- BR0317525A BR0317525A BR0317525-1A BR0317525A BR0317525A BR 0317525 A BR0317525 A BR 0317525A BR 0317525 A BR0317525 A BR 0317525A BR 0317525 A BR0317525 A BR 0317525A
- Authority
- BR
- Brazil
- Prior art keywords
- well
- compounds
- kit
- therapeutic
- pharmaceutical composition
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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Abstract
"COMPOSTOS PIRAZOL ACìCLICO, COMPOSIçãO TERAPêUTICA E FARMACêUTICA, KIT, BEM COMO RESPECTIVOS USOS". A presente invenção refere-se à compostos que inibem proteína quinase e proteína quinase-2 (MK-2) ativadas por mitógeno. Métodos de produção de tais compostos estão descritos, bem como um método de uso dos mesmos para inibição de MK-2 e para prevenção ou tratamento de uma doença ou distúrbio mediado por TNF<244>, onde o método envolve a administração ao indivíduo de um composto inibidor de MK-2 da presente invenção. Também estão descritos composições farmacêuticas e kits contendo os atuais compostos inibidores de MK-2.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US43496202P | 2002-12-20 | 2002-12-20 | |
PCT/US2003/040932 WO2004058176A2 (en) | 2002-12-20 | 2003-12-19 | Acyclic pyrazole compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0317525A true BR0317525A (pt) | 2005-11-16 |
Family
ID=32682131
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0317525-1A BR0317525A (pt) | 2002-12-20 | 2003-12-19 | Compostos pirazol acìclico, composição terapêutica e farmacêutica, kit, bem como respectivos usos |
BR0317430-1A BR0317430A (pt) | 2002-12-20 | 2003-12-19 | Compostos inibidores de quinase-2 de proteìna ativada por quinase de proteìna ativada por mitógeno |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0317430-1A BR0317430A (pt) | 2002-12-20 | 2003-12-19 | Compostos inibidores de quinase-2 de proteìna ativada por quinase de proteìna ativada por mitógeno |
Country Status (15)
Country | Link |
---|---|
US (3) | US20040152739A1 (pt) |
EP (2) | EP1572693A1 (pt) |
JP (2) | JP2006514043A (pt) |
KR (1) | KR20050104339A (pt) |
CN (1) | CN1747949A (pt) |
AU (2) | AU2003301226A1 (pt) |
BR (2) | BR0317525A (pt) |
CA (2) | CA2510298A1 (pt) |
IL (1) | IL169177A0 (pt) |
MX (2) | MXPA05006569A (pt) |
NO (1) | NO20053396L (pt) |
PL (1) | PL377461A1 (pt) |
RU (1) | RU2005119173A (pt) |
WO (2) | WO2004058762A1 (pt) |
ZA (1) | ZA200504898B (pt) |
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- 2003-12-19 ZA ZA200504898A patent/ZA200504898B/en unknown
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- 2003-12-19 PL PL377461A patent/PL377461A1/pl unknown
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- 2003-12-19 EP EP03814309A patent/EP1572682A4/en not_active Withdrawn
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US20040152739A1 (en) | 2004-08-05 |
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US20080113971A1 (en) | 2008-05-15 |
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WO2004058176A3 (en) | 2004-09-16 |
KR20050104339A (ko) | 2005-11-02 |
EP1572693A1 (en) | 2005-09-14 |
AU2003297431A1 (en) | 2004-07-22 |
EP1572682A4 (en) | 2008-01-23 |
CA2510298A1 (en) | 2004-07-15 |
BR0317430A (pt) | 2005-10-25 |
CN1747949A (zh) | 2006-03-15 |
AU2003301226A2 (en) | 2004-07-22 |
NO20053396D0 (no) | 2005-07-13 |
MXPA05006569A (es) | 2005-09-22 |
IL169177A0 (en) | 2007-07-04 |
JP2006511583A (ja) | 2006-04-06 |
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