US3914250A
(en)
|
1974-08-01 |
1975-10-21 |
American Home Prod |
1,4-Diazepino{8 6,5,4-jk{9 carbazoles
|
JPS608117B2
(ja)
|
1977-02-08 |
1985-02-28 |
財団法人微生物化学研究会 |
新生理活性物質エステラスチンおよびその製造法
|
DE2928485A1
(de)
|
1979-07-14 |
1981-01-29 |
Bayer Ag |
Verwendung von harnstoffderivaten als arzneimittel bei der behandlung von fettstoffwechselstoerungen
|
ZA821577B
(en)
|
1981-04-06 |
1983-03-30 |
Boots Co Plc |
Therapeutic agents
|
US4452813A
(en)
|
1981-05-22 |
1984-06-05 |
Taiho Pharmaceutical Company Limited |
Sulfonate derivatives, process for preparing same and antilipemic compositions containing the derivative
|
CA1247547A
(en)
|
1983-06-22 |
1988-12-28 |
Paul Hadvary |
Leucine derivatives
|
EP0136976A3
(de)
|
1983-08-23 |
1985-05-15 |
Ciba-Geigy Ag |
Verwendung von Phenylpyrimidinen als Pflanzenregulatoren
|
IE61928B1
(en)
|
1988-11-29 |
1994-11-30 |
Boots Co Plc |
Treatment of obesity
|
US5391571A
(en)
|
1989-11-15 |
1995-02-21 |
American Home Products Corporation |
Cholesterol ester hydrolase inhibitors
|
US5081122A
(en)
|
1990-03-05 |
1992-01-14 |
Sterling Drug Inc. |
Antiglaucoma compositions containing 4-arylcarbonyl-1-(4-morpholinyl)-lower-alkyl)-1H-indoles and method of use thereof
|
US5112820A
(en)
|
1990-03-05 |
1992-05-12 |
Sterling Drug Inc. |
Anti-glaucoma compositions containing 2- and 3-aminomethyl-6-arylcarbonyl- or 6-phenylthio-2,3-dihydropyrrolo-(1,2,3-de)-1,4-benzoxazines and method of use thereof
|
US5013837A
(en)
|
1990-03-08 |
1991-05-07 |
Sterling Drug Inc. |
3-Arylcarbonyl-1H-indole-containing compounds
|
US4973587A
(en)
|
1990-03-08 |
1990-11-27 |
Sterling Drug Inc. |
3-arylcarbonyl-1-aminoalkyl-1H-indole-containing antiglaucoma method
|
FR2692575B1
(fr)
|
1992-06-23 |
1995-06-30 |
Sanofi Elf |
Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
|
US6472178B1
(en)
|
1998-02-27 |
2002-10-29 |
Regeneron Pharmaceuticals, Inc. |
Nucleic acids encoding a modified ciliary neurotrophic factor and method of making thereof
|
US5349056A
(en)
|
1992-10-09 |
1994-09-20 |
Regeneron Pharmaceuticals |
Modified ciliary neurotrophic factors
|
US5451677A
(en)
|
1993-02-09 |
1995-09-19 |
Merck & Co., Inc. |
Substituted phenyl sulfonamides as selective β 3 agonists for the treatment of diabetes and obesity
|
US5292736A
(en)
|
1993-02-26 |
1994-03-08 |
Sterling Winthrop Inc. |
Morpholinoalkylindenes as antiglaucoma agents
|
FR2714057B1
(fr)
|
1993-12-17 |
1996-03-08 |
Sanofi Elf |
Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant.
|
US5705515A
(en)
|
1994-04-26 |
1998-01-06 |
Merck & Co., Inc. |
Substituted sulfonamides as selective β-3 agonists for the treatment of diabetes and obesity
|
JP3386814B2
(ja)
|
1994-11-07 |
2003-03-17 |
ファイザー・インコーポレーテッド |
ある種の置換ベンジルアミン誘導体:新種の神経ペプチドy1特異的リガンド
|
US5602024A
(en)
|
1994-12-02 |
1997-02-11 |
Synaptic Pharmaceutical Corporation |
DNA encoding a hypothalamic atypical neuropeptide Y/peptide YY receptor (Y5) and uses thereof
|
US5552523A
(en)
|
1995-01-31 |
1996-09-03 |
Eli Lilly And Company |
Anti-obesity proteins
|
WO1996023515A1
(en)
|
1995-01-31 |
1996-08-08 |
Eli Lilly And Company |
Anti-obesity proteins
|
US5552522A
(en)
|
1995-01-31 |
1996-09-03 |
Eli Lilly And Company |
Anti-obesity proteins
|
US5554727A
(en)
|
1995-01-31 |
1996-09-10 |
Eli Lilly And Company |
Anti-obesity proteins
|
US5559208A
(en)
|
1995-01-31 |
1996-09-24 |
Eli Lilly And Company |
Anti-obesity proteins
|
US5521283A
(en)
|
1995-01-31 |
1996-05-28 |
Eli Lilly And Company |
Anti-obesity proteins
|
US5552524A
(en)
|
1995-01-31 |
1996-09-03 |
Eli Lilly And Company |
Anti-obesity proteins
|
US5605886A
(en)
|
1995-01-31 |
1997-02-25 |
Eli Lilly And Company |
Anti-obesity proteins
|
CA2211656A1
(en)
|
1995-01-31 |
1996-08-08 |
Margret B. Basinski |
Anti-obesity proteins
|
US5532237A
(en)
|
1995-02-15 |
1996-07-02 |
Merck Frosst Canada, Inc. |
Indole derivatives with affinity for the cannabinoid receptor
|
US5831115A
(en)
|
1995-04-21 |
1998-11-03 |
Abbott Laboratories |
Inhibitors of squalene synthase and protein farnesyltransferase
|
US20020006964A1
(en)
|
1995-05-16 |
2002-01-17 |
Young James W. |
Methods of using and compositions comprising (+) sibutramine optionally in combination with other pharmacologically active compounds
|
US5739106A
(en)
|
1995-06-07 |
1998-04-14 |
Rink; Timothy J. |
Appetite regulating compositions
|
FR2741621B1
(fr)
|
1995-11-23 |
1998-02-13 |
Sanofi Sa |
Nouveaux derives de pyrazole, procede pour leur preparation et compositions pharmaceutiques en contenant
|
AU7692996A
(en)
|
1995-12-01 |
1997-06-27 |
Ciba-Geigy Ag |
Receptor antagonists
|
AU7692696A
(en)
|
1995-12-01 |
1997-06-27 |
Novartis Ag |
Heteroaryl derivatives
|
WO1997020820A1
(en)
|
1995-12-01 |
1997-06-12 |
Novartis Ag |
Heteroaryl compounds
|
AU7692896A
(en)
|
1995-12-01 |
1997-06-27 |
Novartis Ag |
Quinazolin-2,4-diazirines as NPY receptor antagonist
|
AU1328197A
(en)
|
1995-12-01 |
1997-06-19 |
Synaptic Pharmaceutical Corporation |
Aryl sulfonamide and sulfamide derivatives and uses thereof
|
TW432073B
(en)
|
1995-12-28 |
2001-05-01 |
Pfizer |
Pyrazolopyridine compounds
|
KR19990082330A
(ko)
|
1996-02-06 |
1999-11-25 |
미즈노 마사루 |
신규 화합물 및 이의 의약 용도
|
IT1288388B1
(it)
|
1996-11-19 |
1998-09-22 |
Angeletti P Ist Richerche Bio |
Uso di sostanze che attivano il recettore del cntf ( fattore neurotrofico ciliare) per la preparazione di farmaci per la terapia
|
EP0945440B1
(en)
|
1996-12-16 |
2004-05-26 |
Banyu Pharmaceutical Co., Ltd. |
Aminopyrazole derivatives
|
CA2278307A1
(en)
|
1997-01-21 |
1998-07-23 |
Siegfried Benjamin Christensen Iv |
Novel cannabinoid receptor modulators
|
JP2001511147A
(ja)
|
1997-02-04 |
2001-08-07 |
ザ・ボード・オブ・トラステイーズ・オブ・ザ・ユニバーシテイ・オブ・アーカンソー |
殺菌・殺カビ性のカルボキサミド類
|
CA2470183C
(en)
|
1997-02-21 |
2008-01-29 |
Bayer Aktiengesellschaft |
Intermediates for preparing arylsulphonamides and analogues
|
WO1998041519A1
(en)
|
1997-03-18 |
1998-09-24 |
Smithkline Beecham Corporation |
Novel cannabinoid receptor agonists
|
FR2761265B1
(fr)
|
1997-03-28 |
1999-07-02 |
Sanofi Sa |
Composition pharmaceutique pour l'administration orale d'un derive du n-piperidino-3-pyrazolecarboxamide, de ses sels et de leurs solvates
|
FR2761266B1
(fr)
|
1997-03-28 |
1999-07-02 |
Sanofi Sa |
Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates
|
EP0992239B1
(en)
|
1997-04-23 |
2003-03-12 |
Banyu Pharmaceutical Co., Ltd. |
Neuropeptide y receptor antagonist
|
US6001836A
(en)
|
1997-05-28 |
1999-12-14 |
Bristol-Myers Squibb Company |
Dihydropyridine NPY antagonists: cyanoguanidine derivatives
|
SE9702457D0
(sv)
|
1997-06-26 |
1997-06-26 |
Pharmacia & Upjohn Ab |
Screening
|
KR20010021696A
(ko)
|
1997-07-11 |
2001-03-15 |
미즈노 마사루 |
퀴놀린 화합물 및 그의 의약용도
|
WO1999027965A1
(fr)
|
1997-11-28 |
1999-06-10 |
Banyu Pharmaceutical Co., Ltd. |
Agents anti-hyperlipemiques
|
WO1999051600A1
(en)
|
1998-04-02 |
1999-10-14 |
Neurogen Corporation |
AMINOALKYL SUBSTITUTED 9H-PYRIDINO[2,3-b]INDOLE AND 9H-PYRIMIDINO[4,5-b]INDOLE DERIVATIVES
|
US6140354A
(en)
|
1998-04-29 |
2000-10-31 |
Ortho-Mcneil Pharmaceutical, Inc. |
N-substituted aminotetralins as ligands for the neuropeptide Y Y5 receptor useful in the treatment of obesity and other disorders
|
US6329395B1
(en)
|
1998-06-08 |
2001-12-11 |
Schering Corporation |
Neuropeptide Y5 receptor antagonists
|
WO1999064002A1
(en)
|
1998-06-11 |
1999-12-16 |
Merck & Co., Inc. |
Spiropiperidine derivatives as melanocortin receptor agonists
|
DE19837627A1
(de)
|
1998-08-19 |
2000-02-24 |
Bayer Ag |
Neue Aminosäureester von Arylsulfonamiden und Analoga
|
HN1998000027A
(es)
|
1998-08-19 |
1999-06-02 |
Bayer Ip Gmbh |
Arilsulfonamidas y analagos
|
US6358951B1
(en)
|
1998-08-21 |
2002-03-19 |
Pfizer Inc. |
Growth hormone secretagogues
|
US6337332B1
(en)
|
1998-09-17 |
2002-01-08 |
Pfizer Inc. |
Neuropeptide Y receptor antagonists
|
DK1121111T3
(da)
|
1998-10-15 |
2010-05-31 |
Imp Innovations Ltd |
Forbindelser til behandling af vægttab
|
WO2000027845A1
(en)
|
1998-11-10 |
2000-05-18 |
Merck & Co., Inc. |
Spiro-indolines as y5 receptor antagonists
|
ES2161594B1
(es)
|
1998-12-17 |
2003-04-01 |
Servier Lab |
Nuevos derivados de la hidrazida, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.
|
US6344481B1
(en)
|
1999-03-01 |
2002-02-05 |
Pfizer Inc. |
Thyromimetic antiobesity agents
|
AU773188C
(en)
|
1999-03-19 |
2006-01-05 |
Abbott Gmbh & Co. Kg |
Method of treating eating disorders
|
FR2792314B1
(fr)
|
1999-04-15 |
2001-06-01 |
Adir |
Nouveaux composes aminotriazoles, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
|
DE60034783T2
(de)
|
1999-04-22 |
2008-01-31 |
H. Lundbeck A/S, Valby |
Selektive npy(y5)-antagonisten
|
US6340683B1
(en)
|
1999-04-22 |
2002-01-22 |
Synaptic Pharmaceutical Corporation |
Selective NPY (Y5) antagonists (triazines)
|
MXPA01011321A
(es)
|
1999-05-05 |
2003-08-01 |
Johnson & Johnson |
Neuropeptidos y ligandos de receptores 3a, 4, 5, 9b-tetrahidro-1h-benz(e)indol-2-il amino derivados utiles en el tratamiento de obesidad y otros trastornos.
|
CA2373510A1
(en)
|
1999-05-12 |
2000-11-23 |
Ortho-Mcneil Pharmaceutical, Inc. |
Pyrazole carboxamides useful for the treatment of obesity and other disorders
|
WO2000074679A1
(en)
|
1999-06-04 |
2000-12-14 |
Merck & Co., Inc. |
Substituted piperidines as melanocortin-4 receptor agonists
|
AU773892B2
(en)
|
1999-06-30 |
2004-06-10 |
H. Lundbeck A/S |
Selective NPY (Y5) antagonists
|
WO2001007409A1
(en)
|
1999-07-23 |
2001-02-01 |
Astrazeneca Uk Limited |
Carbazole derivatives and their use as neuropeptide y5 receptor ligands
|
RU2228927C2
(ru)
|
1999-07-28 |
2004-05-20 |
Орто-Макнейл Фармасьютикал, Инк. |
Производные аминов или амидов, фармацевтическая композиция на их основе и способ антагонизирования рецептора y5 нейропептида npy
|
TWI279402B
(en)
|
1999-08-20 |
2007-04-21 |
Banyu Pharma Co Ltd |
Spiro compounds having NPY antagonistic activities and agents containing the same
|
IL148904A0
(en)
|
1999-09-30 |
2002-09-12 |
Neurogen Corp |
Amino substituted pyrazolo {1,5,-a}-1,5- pyrimidines and pyrazolo{1,5,-a}-1,3,5-triazines
|
DE60026155T2
(de)
|
1999-09-30 |
2006-08-10 |
Neurogen Corp., Branford |
Einige alkylendiamin-substituierte heterocyclen
|
YU23802A
(sh)
|
1999-09-30 |
2004-09-03 |
Neurogen Corporation |
Određeni alkilen diamin-supstituisani pirazolo/1,5-a/-1,5- piramidini i pirazolo/1,5-a/1,3,5-triazini
|
DE19949319A1
(de)
|
1999-10-13 |
2001-06-13 |
Ruetgers Vft Ag |
Verfahren zur Herstellung von Arylalkylethern
|
SK4732002A3
(en)
|
1999-10-13 |
2002-12-03 |
Pfizer Prod Inc |
Biaryl ether derivatives useful as monoamine reuptake inhibitors
|
US6444687B1
(en)
|
1999-12-16 |
2002-09-03 |
Schering Corporation |
Substituted imidazole neuropeptide Y Y5 receptor antagonists
|
AU2001228325A1
(en)
|
2000-02-01 |
2001-08-14 |
Novo-Nordisk A/S |
Use of compounds for the regulation of food intake
|
WO2001058869A2
(en)
|
2000-02-11 |
2001-08-16 |
Bristol-Myers Squibb Company |
Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators in treating respiratory and non-respiratory diseases
|
JP2001226269A
(ja)
|
2000-02-18 |
2001-08-21 |
Takeda Chem Ind Ltd |
メラニン凝集ホルモン拮抗剤
|
ATE292119T1
(de)
|
2000-02-22 |
2005-04-15 |
Banyu Pharma Co Ltd |
Imidazolin-verbindungen
|
GB0004003D0
(en)
|
2000-02-22 |
2000-04-12 |
Knoll Ag |
Therapeutic agents
|
US6531478B2
(en)
|
2000-02-24 |
2003-03-11 |
Cheryl P. Kordik |
Amino pyrazole derivatives useful for the treatment of obesity and other disorders
|
FR2805810B1
(fr)
|
2000-03-03 |
2002-04-26 |
Aventis Pharma Sa |
Compositions pharmaceutiques contenant des derives de 3- amino-azetidine, les nouveaux derives et leur preparation
|
FR2805817B1
(fr)
|
2000-03-03 |
2002-04-26 |
Aventis Pharma Sa |
Compositions pharmaceutiques contenant des derives d'azetidine, les nouveaux derives d'azetidine et leur preparation
|
FR2805818B1
(fr)
|
2000-03-03 |
2002-04-26 |
Aventis Pharma Sa |
Derives d'azetidine, leur preparation et les compositions pharmaceutiques les contenant
|
EP1132389A1
(en)
|
2000-03-06 |
2001-09-12 |
Vernalis Research Limited |
New aza-indolyl derivatives for the treatment of obesity
|
HU227811B1
(en)
|
2000-03-14 |
2012-03-28 |
Actelion Pharmaceuticals Ltd |
1,2,3,4-tetrahydroisquinoline derivatives, pharmaceutical compositions containing them and their preparation processes
|
US6472398B1
(en)
|
2000-03-23 |
2002-10-29 |
Merck & Co., Inc. |
Spiropiperidine derivatives as melanocortin receptor agonists
|
CA2403686C
(en)
|
2000-03-23 |
2010-01-26 |
Merck & Co., Inc. |
Substituted piperidines as melanocortin receptor agonists
|
US6600015B2
(en)
|
2000-04-04 |
2003-07-29 |
Hoffmann-La Roche Inc. |
Selective linear peptides with melanocortin-4 receptor (MC4-R) agonist activity
|
EP1142886A1
(en)
|
2000-04-07 |
2001-10-10 |
Aventis Pharma Deutschland GmbH |
Percyquinnin, a process for its production and its use as a pharmaceutical
|
WO2001082925A1
(fr)
|
2000-04-28 |
2001-11-08 |
Takeda Chemical Industries, Ltd. |
Antagonistes de l'hormone concentrant la melanine
|
GB0010757D0
(en)
|
2000-05-05 |
2000-06-28 |
Astrazeneca Ab |
Chemical compounds
|
GB0011013D0
(en)
|
2000-05-09 |
2000-06-28 |
Astrazeneca Ab |
Chemical compounds
|
US6432960B2
(en)
|
2000-05-10 |
2002-08-13 |
Bristol-Myers Squibb Company |
Squarate derivatives of dihydropyridine NPY antagonists
|
US6444675B2
(en)
|
2000-05-10 |
2002-09-03 |
Bristol-Myers Squibb Company |
4-alkyl and 4-cycloalkyl derivatives of dihydropyridine NPY antagonists
|
WO2001085173A1
(en)
|
2000-05-10 |
2001-11-15 |
Bristol-Myers Squibb Company |
Alkylamine derivatives of dihydropyridine npy antagonists
|
AU5959201A
(en)
|
2000-05-11 |
2001-11-20 |
Bristol Myers Squibb Co |
Tetrahydroisoquinoline analogs useful as growth hormone secretagogues
|
AU2001256733A1
(en)
|
2000-05-16 |
2001-11-26 |
Takeda Chemical Industries Ltd. |
Melanin-concentrating hormone antagonist
|
AU2001259056A1
(en)
|
2000-05-17 |
2001-11-26 |
Eli Lilly And Company |
Method for selectively inhibiting ghrelin action
|
US6391881B2
(en)
|
2000-05-19 |
2002-05-21 |
Bristol-Myers Squibb Company |
Thiourea derivatives of dihydropyridine NPY antagonists
|
SE0001899D0
(sv)
|
2000-05-22 |
2000-05-22 |
Pharmacia & Upjohn Ab |
New compounds
|
EP1289526A4
(en)
|
2000-05-30 |
2005-03-16 |
Merck & Co Inc |
MELANOCORTIN RECEPTOR AGONISTS
|
MXPA02012447A
(es)
|
2000-06-15 |
2003-04-25 |
Schering Corp |
Antagonistas receptores de trombina.
|
ES2238458T3
(es)
|
2000-06-16 |
2005-09-01 |
Smithkline Beecham Plc |
Piperidinas para uso como antagonistas de los receptores de orexina.
|
EP1299362A4
(en)
|
2000-07-05 |
2004-11-03 |
Synaptic Pharma Corp |
SELECTIVE RECEPTOR ANTAGONISTS OF MELANINE CONCENTRATING HORMON-1 (MCH1) AND THEIR USE
|
CA2414198A1
(en)
|
2000-07-06 |
2002-01-17 |
Neurogen Corporation |
Melanin concentrating hormone receptor ligands
|
GB0019357D0
(en)
|
2000-08-07 |
2000-09-27 |
Melacure Therapeutics Ab |
Novel phenyl guanidines
|
AU2001283938A1
(en)
|
2000-07-24 |
2002-02-05 |
Ardana Bioscience Limited |
Ghrelin antagonists
|
DK1325008T3
(da)
|
2000-07-31 |
2006-02-13 |
Hoffmann La Roche |
Piperazinderivater
|
US6768024B1
(en)
|
2000-08-04 |
2004-07-27 |
Lion Bioscience Ag |
Triamine derivative melanocortin receptor ligands and methods of using same
|
GB0019359D0
(en)
|
2000-08-07 |
2000-09-27 |
Melacure Therapeutics Ab |
Novel guanidines
|
EP1320364A1
(en)
|
2000-08-21 |
2003-06-25 |
Gliatech, Inc. |
The use of histamine h3-receptor inverse agonists for the control of appetite and treatment of obesity
|
WO2002015845A2
(en)
|
2000-08-21 |
2002-02-28 |
Merck & Co., Inc. |
Anti-hypercholesterolemic drug combination
|
AU2001288285B2
(en)
|
2000-08-23 |
2005-09-29 |
Merck & Co., Inc. |
Substituted piperidines as melanocortin receptor agonists
|
US6900226B2
(en)
|
2000-09-06 |
2005-05-31 |
Hoffman-La Roche Inc. |
Neuropeptide Y antagonists
|
US20020165223A1
(en)
|
2000-09-14 |
2002-11-07 |
Greenlee William J. |
Substituted urea neuropeptide Y Y5 receptor antagonists
|
IL154809A0
(en)
|
2000-10-13 |
2003-10-31 |
Lilly Co Eli |
Substituted dipeptides as growth hormone secretagogues
|
EP1328515B1
(en)
|
2000-10-16 |
2008-08-06 |
F. Hoffmann-La Roche AG |
Indoline derivatives and their use as 5-ht2 receptor ligands
|
MXPA03003455A
(es)
|
2000-10-20 |
2003-07-14 |
Pfizer Prod Inc |
Agonistas del receptor beta3-adrenergico y usos de los mismos.
|
WO2002036596A2
(en)
|
2000-11-03 |
2002-05-10 |
Wyeth |
CYCLOALKYL[b][1,4]DIAZEPINO[6,7,1-hi]INDOLES AND DERIVATIVES
|
EP1335907B1
(en)
|
2000-11-20 |
2010-06-09 |
Biovitrum AB (publ) |
Piperazinylpyrazine compounds as agonist or antagonist of serotonin 5ht-2 receptor
|
ATE433962T1
(de)
|
2000-11-20 |
2009-07-15 |
Biovitrum Ab Publ |
Piperazinylpyrazinverbindungen als antagonisten des serotonin-5-ht2-rezeptors
|
US6566367B2
(en)
|
2000-12-12 |
2003-05-20 |
Pfizer Inc. |
Spiro[isobenzofuran-1,4′-piperidin]-3-ones and 3H-spiroisobenzofuran-1,4′-piperidines
|
GB0030710D0
(en)
|
2000-12-15 |
2001-01-31 |
Hoffmann La Roche |
Piperazine derivatives
|
AR035520A1
(es)
|
2000-12-21 |
2004-06-02 |
Schering Corp |
Compuestos heteroarilo urea que son neuropeptidos y antagonistas de los receptores y5 del neuropeptido y, composiciones farmaceuticas, un proceso para su preparacion, uso de dichos compuestos y composiciones para la manufactura de medicamentos
|
JP4025200B2
(ja)
|
2000-12-22 |
2007-12-19 |
シェーリング コーポレイション |
ピペリジンmchアンタゴニストおよび肥満の処置におけるそれらの使用
|
AU2002228007B2
(en)
|
2000-12-27 |
2007-06-21 |
F. Hoffmann-La Roche Ag |
Indole derivatives and their use as 5-HT2b and 5-HT2c receptor ligands
|
WO2002051232A2
(en)
|
2000-12-27 |
2002-07-04 |
Actelion Pharmaceuticals Ltd. |
Novel benzazepines and related heterocyclic derivatives
|
EP1368339A1
(en)
|
2001-01-23 |
2003-12-10 |
Eli Lilly & Company |
Substituted piperidines/piperazines as melanocortin receptor agonists
|
DE60205465T2
(de)
|
2001-01-23 |
2006-04-20 |
Eli Lilly And Co., Indianapolis |
Piperazinderivate als agonisten des melanocortin-rezeptors
|
JP2004524297A
(ja)
|
2001-01-23 |
2004-08-12 |
イーライ・リリー・アンド・カンパニー |
メラノコルチン受容体アゴニスト
|
CN1500080A
(zh)
|
2001-02-02 |
2004-05-26 |
����ҩƷ��ҵ��ʽ���� |
稠合杂环化合物
|
WO2002068387A2
(en)
|
2001-02-28 |
2002-09-06 |
Merck & Co., Inc. |
Acylated piperidine derivatives as melanocortin-4 receptor agonists
|
ES2283550T3
(es)
|
2001-02-28 |
2007-11-01 |
MERCK & CO., INC. |
Derivados de piperidina acilados como antagonistas del receptor de.
|
AU2002250343B2
(en)
|
2001-02-28 |
2006-05-25 |
Merck Sharp & Dohme Corp. |
Acylated piperidine derivatives as melanocortin-4 receptor agonists
|
EP1370520A1
(en)
|
2001-03-21 |
2003-12-17 |
Pharmacopeia, Inc. |
Aryl and biaryl compounds having mch modulatory activity
|
US6900329B2
(en)
|
2001-03-21 |
2005-05-31 |
Schering Corporation |
MCH antagonists and their use in the treatment of obesity
|
IL153508A
(en)
|
2001-03-22 |
2008-07-08 |
Solvay Pharm Bv |
Derivatives of 4,5 - Dihydro-1H-pyrazole with antagonistic activity to the 1CB receptor
|
EP1373212A4
(en)
|
2001-03-29 |
2004-06-23 |
Molecular Design Int |
ADRENERGIC-BETA-3 RECEPTOR AGONISTS, AGONIST COMPOSITIONS AND METHODS OF PREPARING AND USING THE SAME
|
US6573287B2
(en)
|
2001-04-12 |
2003-06-03 |
Bristo-Myers Squibb Company |
2,1-oxazoline and 1,2-pyrazoline-based inhibitors of dipeptidyl peptidase IV and method
|
PE20021081A1
(es)
|
2001-04-12 |
2002-12-18 |
Pharmacopeia Drug Discovery |
Aril y biaril piperidinas con actividad moduladora mch
|
FR2824825B1
(fr)
|
2001-05-15 |
2005-05-06 |
Servier Lab |
Nouveaux derives d'alpha-amino-acides, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
|
ES2300478T3
(es)
|
2001-05-21 |
2008-06-16 |
F. Hoffmann-La Roche Ag |
Derivados de quinolina como ligandos para el receptor de neuropeptido y.
|
MXPA03010612A
(es)
|
2001-05-22 |
2004-04-02 |
Neurogen Corp |
Ligandos receptores de la hormona concentradora de melanina: analogos de 1-bencil-4-aril piperazina substiruidos.
|
CA2450475A1
(en)
|
2001-06-20 |
2003-01-03 |
Linda Brockunier |
Dipeptidyl peptidase inhibitors for the treatment of diabetes
|
DE60224189T2
(de)
|
2001-06-20 |
2008-12-11 |
Merck & Co., Inc. |
Dipeptidylpeptidase-hemmer zur behandlung von diabetes
|
GB0115517D0
(en)
|
2001-06-25 |
2001-08-15 |
Ferring Bv |
Novel antidiabetic agents
|
PL367527A1
(en)
|
2001-06-27 |
2005-02-21 |
Smithkline Beecham Corporation |
Fluoropyrrolidines as dipeptidyl peptidase inhibitors
|
ZA200300833B
(en)
|
2001-06-27 |
2004-02-10 |
Probiodrug Ag |
Dipeptidyl peptidase IV inhibitors and their uses as anti-cancer agents.
|
JP4357293B2
(ja)
|
2001-06-27 |
2009-11-04 |
スミスクライン ビーチャム コーポレーション |
ジペプチジルペプチダーゼ阻害剤としてのフルオロピロリジン類
|
AU2002316437A1
(en)
|
2001-06-27 |
2003-03-03 |
Smithkline Beecham Corporation |
Pyrrolidines as dipeptidyl peptidase inhibitors
|
JP2005502624A
(ja)
|
2001-07-03 |
2005-01-27 |
ノボ ノルディスク アクティーゼルスカブ |
糖尿病を治療するための、dpp−ivを阻害するプリン誘導体
|
EP1411942A4
(en)
|
2001-07-05 |
2005-01-26 |
Synaptic Pharma Corp |
SUBSTITUTED ANILINE PIPERIDINES AS SELECTIVE MCH ANTAGONISTS
|
UA74912C2
(en)
|
2001-07-06 |
2006-02-15 |
Merck & Co Inc |
Beta-aminotetrahydroimidazo-(1,2-a)-pyrazines and tetratriazolo-(4,3-a)-pyrazines as inhibitors of dipeptylpeptidase for the treatment or prevention of diabetes
|
ITMI20011483A1
(it)
|
2001-07-11 |
2003-01-11 |
Res & Innovation Soc Coop A R |
Uso di composti come antagonisti funzionali ai recettori centrali deicannabinoidi
|
EP1411940B1
(en)
|
2001-07-18 |
2008-10-15 |
Merck & Co., Inc. |
Bridged piperidine derivatives as melanocortin receptor agonists
|
AU2002319627A1
(en)
|
2001-07-20 |
2003-03-03 |
Merck And Co., Inc. |
Substituted imidazoles as cannabinoid receptor modulators
|
US6977264B2
(en)
|
2001-07-25 |
2005-12-20 |
Amgen Inc. |
Substituted piperidines and methods of use
|
US6915444B2
(en)
|
2001-09-12 |
2005-07-05 |
Rockwell Automation Technologies, Inc. |
Network independent safety protocol for industrial controller using data manipulation techniques
|
DE60328035D1
(de)
*
|
2002-11-29 |
2009-07-30 |
Banyu Pharma Co Ltd |
Neue azolderivate
|