|
US3914250A
(en)
|
1974-08-01 |
1975-10-21 |
American Home Prod |
1,4-Diazepino{8 6,5,4-jk{9 carbazoles
|
|
JPS608117B2
(ja)
|
1977-02-08 |
1985-02-28 |
財団法人微生物化学研究会 |
新生理活性物質エステラスチンおよびその製造法
|
|
DE2928485A1
(de)
|
1979-07-14 |
1981-01-29 |
Bayer Ag |
Verwendung von harnstoffderivaten als arzneimittel bei der behandlung von fettstoffwechselstoerungen
|
|
ZA821577B
(en)
|
1981-04-06 |
1983-03-30 |
Boots Co Plc |
Therapeutic agents
|
|
US4452813A
(en)
|
1981-05-22 |
1984-06-05 |
Taiho Pharmaceutical Company Limited |
Sulfonate derivatives, process for preparing same and antilipemic compositions containing the derivative
|
|
CA1247547A
(en)
|
1983-06-22 |
1988-12-28 |
Paul Hadvary |
Leucine derivatives
|
|
EP0136976A3
(de)
|
1983-08-23 |
1985-05-15 |
Ciba-Geigy Ag |
Verwendung von Phenylpyrimidinen als Pflanzenregulatoren
|
|
IE61928B1
(en)
|
1988-11-29 |
1994-11-30 |
Boots Co Plc |
Treatment of obesity
|
|
US5391571A
(en)
|
1989-11-15 |
1995-02-21 |
American Home Products Corporation |
Cholesterol ester hydrolase inhibitors
|
|
US5081122A
(en)
|
1990-03-05 |
1992-01-14 |
Sterling Drug Inc. |
Antiglaucoma compositions containing 4-arylcarbonyl-1-(4-morpholinyl)-lower-alkyl)-1H-indoles and method of use thereof
|
|
US5112820A
(en)
|
1990-03-05 |
1992-05-12 |
Sterling Drug Inc. |
Anti-glaucoma compositions containing 2- and 3-aminomethyl-6-arylcarbonyl- or 6-phenylthio-2,3-dihydropyrrolo-(1,2,3-de)-1,4-benzoxazines and method of use thereof
|
|
US4973587A
(en)
|
1990-03-08 |
1990-11-27 |
Sterling Drug Inc. |
3-arylcarbonyl-1-aminoalkyl-1H-indole-containing antiglaucoma method
|
|
US5013837A
(en)
|
1990-03-08 |
1991-05-07 |
Sterling Drug Inc. |
3-Arylcarbonyl-1H-indole-containing compounds
|
|
FR2692575B1
(fr)
|
1992-06-23 |
1995-06-30 |
Sanofi Elf |
Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
|
|
US5349056A
(en)
|
1992-10-09 |
1994-09-20 |
Regeneron Pharmaceuticals |
Modified ciliary neurotrophic factors
|
|
US6472178B1
(en)
|
1998-02-27 |
2002-10-29 |
Regeneron Pharmaceuticals, Inc. |
Nucleic acids encoding a modified ciliary neurotrophic factor and method of making thereof
|
|
US5451677A
(en)
|
1993-02-09 |
1995-09-19 |
Merck & Co., Inc. |
Substituted phenyl sulfonamides as selective β 3 agonists for the treatment of diabetes and obesity
|
|
US5292736A
(en)
|
1993-02-26 |
1994-03-08 |
Sterling Winthrop Inc. |
Morpholinoalkylindenes as antiglaucoma agents
|
|
FR2714057B1
(fr)
|
1993-12-17 |
1996-03-08 |
Sanofi Elf |
Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant.
|
|
US5705515A
(en)
|
1994-04-26 |
1998-01-06 |
Merck & Co., Inc. |
Substituted sulfonamides as selective β-3 agonists for the treatment of diabetes and obesity
|
|
PL321136A1
(en)
|
1994-11-07 |
1997-11-24 |
Pfizer |
Some substituted derivatives of bencylamine as a new class of specific ligands of neuropeptide y1
|
|
US5602024A
(en)
|
1994-12-02 |
1997-02-11 |
Synaptic Pharmaceutical Corporation |
DNA encoding a hypothalamic atypical neuropeptide Y/peptide YY receptor (Y5) and uses thereof
|
|
US5552522A
(en)
|
1995-01-31 |
1996-09-03 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
WO1996023515A1
(en)
|
1995-01-31 |
1996-08-08 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5552523A
(en)
|
1995-01-31 |
1996-09-03 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5521283A
(en)
|
1995-01-31 |
1996-05-28 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
WO1996023514A1
(en)
|
1995-01-31 |
1996-08-08 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5559208A
(en)
|
1995-01-31 |
1996-09-24 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5554727A
(en)
|
1995-01-31 |
1996-09-10 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5605886A
(en)
|
1995-01-31 |
1997-02-25 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5552524A
(en)
|
1995-01-31 |
1996-09-03 |
Eli Lilly And Company |
Anti-obesity proteins
|
|
US5532237A
(en)
|
1995-02-15 |
1996-07-02 |
Merck Frosst Canada, Inc. |
Indole derivatives with affinity for the cannabinoid receptor
|
|
US5831115A
(en)
|
1995-04-21 |
1998-11-03 |
Abbott Laboratories |
Inhibitors of squalene synthase and protein farnesyltransferase
|
|
US20020006964A1
(en)
|
1995-05-16 |
2002-01-17 |
Young James W. |
Methods of using and compositions comprising (+) sibutramine optionally in combination with other pharmacologically active compounds
|
|
US5739106A
(en)
|
1995-06-07 |
1998-04-14 |
Rink; Timothy J. |
Appetite regulating compositions
|
|
FR2741621B1
(fr)
|
1995-11-23 |
1998-02-13 |
Sanofi Sa |
Nouveaux derives de pyrazole, procede pour leur preparation et compositions pharmaceutiques en contenant
|
|
AU1328197A
(en)
|
1995-12-01 |
1997-06-19 |
Synaptic Pharmaceutical Corporation |
Aryl sulfonamide and sulfamide derivatives and uses thereof
|
|
WO1997020822A1
(en)
|
1995-12-01 |
1997-06-12 |
Novartis Ag |
Quinazolin-2,4-diazirines as npy receptor antagonist
|
|
WO1997020823A2
(en)
|
1995-12-01 |
1997-06-12 |
Novartis Ag |
2-amino quinazoline derivatives as npy receptor antagonists
|
|
WO1997020821A1
(en)
|
1995-12-01 |
1997-06-12 |
Novartis Ag |
Heteroaryl derivatives
|
|
AU7626496A
(en)
|
1995-12-01 |
1997-06-27 |
Ciba-Geigy Ag |
Heteroaryl compounds
|
|
TW432073B
(en)
|
1995-12-28 |
2001-05-01 |
Pfizer |
Pyrazolopyridine compounds
|
|
AU1618697A
(en)
|
1996-02-06 |
1997-08-28 |
Japan Tobacco Inc. |
Novel compounds and pharmaceutical use thereof
|
|
IT1288388B1
(it)
|
1996-11-19 |
1998-09-22 |
Angeletti P Ist Richerche Bio |
Uso di sostanze che attivano il recettore del cntf ( fattore neurotrofico ciliare) per la preparazione di farmaci per la terapia
|
|
US6180653B1
(en)
|
1996-12-16 |
2001-01-30 |
Banyu Pharmaceutical Co., Ltd. |
Aminopyrazole derivatives
|
|
DE69822449T2
(de)
|
1997-01-21 |
2005-01-27 |
Smithkline Beecham Corp. |
Neue cannabinoidrezeptor-modulatoren
|
|
US6251947B1
(en)
|
1997-02-04 |
2001-06-26 |
Board Of Trustees Of The University Of Arkansas |
Fungicidal carboxamides
|
|
ATE229502T1
(de)
|
1997-02-21 |
2002-12-15 |
Bayer Ag |
Arylsulfonamide und analoga und ihre verwendung zur behandlung von neurodegenerativen erkrankungen
|
|
CA2283797A1
(en)
|
1997-03-18 |
1998-09-24 |
Paul Elliot Bender |
Novel cannabinoid receptor agonists
|
|
FR2761265B1
(fr)
|
1997-03-28 |
1999-07-02 |
Sanofi Sa |
Composition pharmaceutique pour l'administration orale d'un derive du n-piperidino-3-pyrazolecarboxamide, de ses sels et de leurs solvates
|
|
FR2761266B1
(fr)
|
1997-03-28 |
1999-07-02 |
Sanofi Sa |
Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates
|
|
US6258837B1
(en)
|
1997-04-23 |
2001-07-10 |
Banyu Pharmaceutical Co., Ltd. |
Neuropeptide Y receptor antagonist
|
|
US6001836A
(en)
|
1997-05-28 |
1999-12-14 |
Bristol-Myers Squibb Company |
Dihydropyridine NPY antagonists: cyanoguanidine derivatives
|
|
SE9702457D0
(sv)
|
1997-06-26 |
1997-06-26 |
Pharmacia & Upjohn Ab |
Screening
|
|
KR20010021696A
(ko)
|
1997-07-11 |
2001-03-15 |
미즈노 마사루 |
퀴놀린 화합물 및 그의 의약용도
|
|
WO1999027965A1
(en)
|
1997-11-28 |
1999-06-10 |
Banyu Pharmaceutical Co., Ltd. |
Antihyperlipemic agents
|
|
JP2002510688A
(ja)
|
1998-04-02 |
2002-04-09 |
ニューロゲン コーポレイション |
アミノアルキル置換9H−ピリジノ[2,3−b]インドールおよび9H−ピリミジノ[4,5−b]インドール誘導体
|
|
DK1076644T3
(da)
|
1998-04-29 |
2004-08-30 |
Ortho Mcneil Pharm Inc |
N-Substituerede aminotetraliner som ligander for neutopeptid Y Y5-receptoren, der er nyttig til behandling af fedme og andre lidelser
|
|
US6329395B1
(en)
|
1998-06-08 |
2001-12-11 |
Schering Corporation |
Neuropeptide Y5 receptor antagonists
|
|
WO1999064002A1
(en)
|
1998-06-11 |
1999-12-16 |
Merck & Co., Inc. |
Spiropiperidine derivatives as melanocortin receptor agonists
|
|
DE19837627A1
(de)
|
1998-08-19 |
2000-02-24 |
Bayer Ag |
Neue Aminosäureester von Arylsulfonamiden und Analoga
|
|
HN1998000027A
(es)
|
1998-08-19 |
1999-06-02 |
Bayer Ip Gmbh |
Arilsulfonamidas y analagos
|
|
US6358951B1
(en)
|
1998-08-21 |
2002-03-19 |
Pfizer Inc. |
Growth hormone secretagogues
|
|
US6337332B1
(en)
|
1998-09-17 |
2002-01-08 |
Pfizer Inc. |
Neuropeptide Y receptor antagonists
|
|
JP2002527378A
(ja)
|
1998-10-15 |
2002-08-27 |
インペリアル・カレッジ・イノベイションズ・リミテッド |
治療方法
|
|
DE69929235T2
(de)
|
1998-11-10 |
2006-08-24 |
Merck & Co., Inc. |
Spiro-indole als y5-rezeptor antagonisten
|
|
ES2161594B1
(es)
|
1998-12-17 |
2003-04-01 |
Servier Lab |
Nuevos derivados de la hidrazida, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.
|
|
US6344481B1
(en)
|
1999-03-01 |
2002-02-05 |
Pfizer Inc. |
Thyromimetic antiobesity agents
|
|
CA2367666C
(en)
|
1999-03-19 |
2008-11-25 |
Carl M. Mendel |
Method of treating eating disorders
|
|
FR2792314B1
(fr)
|
1999-04-15 |
2001-06-01 |
Adir |
Nouveaux composes aminotriazoles, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
|
|
WO2000064880A1
(en)
|
1999-04-22 |
2000-11-02 |
Synaptic Pharmaceutical Corporation |
Selective npy (y5) antagonists
|
|
US6340683B1
(en)
|
1999-04-22 |
2002-01-22 |
Synaptic Pharmaceutical Corporation |
Selective NPY (Y5) antagonists (triazines)
|
|
WO2000068197A1
(en)
|
1999-05-05 |
2000-11-16 |
Ortho-Mcneil Pharmaceutical, Inc. |
3a,4,5,9b-TETRAHYDRO-1H-BENZ[e]INDOL-2-YL AMINE-DERIVED NEUROPEPTIDE Y RECEPTORS LIGANDS USEFUL IN THE TREATMENT OF OBESITY AND OTHER DISORDERS
|
|
US6291476B1
(en)
|
1999-05-12 |
2001-09-18 |
Ortho-Mcneil Pharmaceutical, Inc. |
Pyrazole carboxamides useful for the treatment of obesity and other disorders
|
|
AU766191B2
(en)
|
1999-06-04 |
2003-10-09 |
Merck & Co., Inc. |
Substituted piperidines as melanocortin-4 receptor agonists
|
|
DK1194421T3
(da)
|
1999-06-30 |
2006-02-13 |
Lundbeck & Co As H |
Selektive NPY (Y5) antagonister
|
|
WO2001007409A1
(en)
|
1999-07-23 |
2001-02-01 |
Astrazeneca Uk Limited |
Carbazole derivatives and their use as neuropeptide y5 receptor ligands
|
|
HUP0202143A3
(en)
|
1999-07-28 |
2003-12-29 |
Ortho Mcneil Pharm Inc |
Amine and amide derivatives as ligands for the neuropeptide y y5 receptor pharmaceutical compositions containing them and their use
|
|
TWI279402B
(en)
|
1999-08-20 |
2007-04-21 |
Banyu Pharma Co Ltd |
Spiro compounds having NPY antagonistic activities and agents containing the same
|
|
EP1224187B1
(en)
|
1999-09-30 |
2006-02-22 |
Neurogen Corporation |
Certain alkylene diamine-substituted heterocycles
|
|
YU23802A
(sh)
|
1999-09-30 |
2004-09-03 |
Neurogen Corporation |
Određeni alkilen diamin-supstituisani pirazolo/1,5-a/-1,5- piramidini i pirazolo/1,5-a/1,3,5-triazini
|
|
CA2379633C
(en)
|
1999-09-30 |
2006-06-20 |
Neurogen Corporation |
Amino substituted pyrazolo[1,5,-a]-1,5-pyrimidines and pyrazolo[1,5-a]-1,3,5-triazines
|
|
DE19949319A1
(de)
|
1999-10-13 |
2001-06-13 |
Ruetgers Vft Ag |
Verfahren zur Herstellung von Arylalkylethern
|
|
CZ20021180A3
(cs)
|
1999-10-13 |
2002-11-13 |
Pfizer Products Inc. |
Biaryletherové deriváty uľitečné jako inhibitory zpětného vychytávání monoaminu
|
|
DE60022386T2
(de)
|
1999-12-16 |
2006-06-22 |
Schering Corp. |
Substituierte imidazole als neuropeptide y y5 rezeptor antagonisten
|
|
WO2001056592A1
(en)
|
2000-02-01 |
2001-08-09 |
Novo Nordisk A/S |
Use of compounds for the regulation of food intake
|
|
CA2399791A1
(en)
|
2000-02-11 |
2001-08-16 |
Bristol-Myers Squibb Company |
Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators in treating respiratory and non-respiratory diseases
|
|
JP2001226269A
(ja)
|
2000-02-18 |
2001-08-21 |
Takeda Chem Ind Ltd |
メラニン凝集ホルモン拮抗剤
|
|
GB0004003D0
(en)
|
2000-02-22 |
2000-04-12 |
Knoll Ag |
Therapeutic agents
|
|
ES2236178T3
(es)
|
2000-02-22 |
2005-07-16 |
Banyu Pharmaceutical Co., Ltd. |
Nuevos compuestos de imidazolina.
|
|
US6531478B2
(en)
|
2000-02-24 |
2003-03-11 |
Cheryl P. Kordik |
Amino pyrazole derivatives useful for the treatment of obesity and other disorders
|
|
FR2805810B1
(fr)
|
2000-03-03 |
2002-04-26 |
Aventis Pharma Sa |
Compositions pharmaceutiques contenant des derives de 3- amino-azetidine, les nouveaux derives et leur preparation
|
|
FR2805817B1
(fr)
|
2000-03-03 |
2002-04-26 |
Aventis Pharma Sa |
Compositions pharmaceutiques contenant des derives d'azetidine, les nouveaux derives d'azetidine et leur preparation
|
|
FR2805818B1
(fr)
|
2000-03-03 |
2002-04-26 |
Aventis Pharma Sa |
Derives d'azetidine, leur preparation et les compositions pharmaceutiques les contenant
|
|
EP1132389A1
(en)
|
2000-03-06 |
2001-09-12 |
Vernalis Research Limited |
New aza-indolyl derivatives for the treatment of obesity
|
|
US6703392B2
(en)
|
2000-03-14 |
2004-03-09 |
Actelion Pharmaceuticals Ltd. |
1,2,3,4-tetrahydroisoquinoline derivatives
|
|
AU2001249296B2
(en)
|
2000-03-23 |
2005-03-24 |
Merck Sharp & Dohme Corp. |
Substituted piperidines as melanocortin receptor agonists
|
|
AU4928101A
(en)
|
2000-03-23 |
2001-10-03 |
Merck & Co Inc |
Spiropiperidine derivatives as melanocortin receptor agonists
|
|
US6600015B2
(en)
|
2000-04-04 |
2003-07-29 |
Hoffmann-La Roche Inc. |
Selective linear peptides with melanocortin-4 receptor (MC4-R) agonist activity
|
|
EP1142886A1
(en)
|
2000-04-07 |
2001-10-10 |
Aventis Pharma Deutschland GmbH |
Percyquinnin, a process for its production and its use as a pharmaceutical
|
|
WO2001082925A1
(en)
|
2000-04-28 |
2001-11-08 |
Takeda Chemical Industries, Ltd. |
Melanin concentrating hormone antagonists
|
|
GB0010757D0
(en)
|
2000-05-05 |
2000-06-28 |
Astrazeneca Ab |
Chemical compounds
|
|
GB0011013D0
(en)
|
2000-05-09 |
2000-06-28 |
Astrazeneca Ab |
Chemical compounds
|
|
US6432960B2
(en)
|
2000-05-10 |
2002-08-13 |
Bristol-Myers Squibb Company |
Squarate derivatives of dihydropyridine NPY antagonists
|
|
US6444675B2
(en)
|
2000-05-10 |
2002-09-03 |
Bristol-Myers Squibb Company |
4-alkyl and 4-cycloalkyl derivatives of dihydropyridine NPY antagonists
|
|
WO2001085173A1
(en)
|
2000-05-10 |
2001-11-15 |
Bristol-Myers Squibb Company |
Alkylamine derivatives of dihydropyridine npy antagonists
|
|
ES2252230T3
(es)
|
2000-05-11 |
2006-05-16 |
Bristol-Myers Squibb Company |
Analogos de tetrahidroisoquinolina utiles como secretores de la hormona del crecimiento.
|
|
CA2408913A1
(en)
|
2000-05-16 |
2001-11-22 |
Takeda Chemical Industries, Ltd. |
Melanin-concentrating hormone antagonist
|
|
AU2001259056A1
(en)
|
2000-05-17 |
2001-11-26 |
Eli Lilly And Company |
Method for selectively inhibiting ghrelin action
|
|
US6391881B2
(en)
|
2000-05-19 |
2002-05-21 |
Bristol-Myers Squibb Company |
Thiourea derivatives of dihydropyridine NPY antagonists
|
|
SE0001899D0
(sv)
|
2000-05-22 |
2000-05-22 |
Pharmacia & Upjohn Ab |
New compounds
|
|
JP2003534377A
(ja)
|
2000-05-30 |
2003-11-18 |
メルク エンド カムパニー インコーポレーテッド |
メラノコルチン受容体作働薬
|
|
EP1294714B1
(en)
|
2000-06-15 |
2007-08-01 |
Schering Corporation |
Thrombin receptor antagonists
|
|
WO2001096302A1
(en)
|
2000-06-16 |
2001-12-20 |
Smithkline Beecham P.L.C. |
Piperidines for use as orexin receptor antagonists
|
|
WO2002006245A1
(en)
|
2000-07-05 |
2002-01-24 |
Synaptic Pharmarceutical Corporation |
Selective melanin concentrating hormone-1 (mch1) receptor antagonists and uses thereof
|
|
EP1366030A2
(en)
|
2000-07-06 |
2003-12-03 |
Neurogen Corporation |
Melanin concentrating hormone receptor ligands
|
|
GB0019357D0
(en)
|
2000-08-07 |
2000-09-27 |
Melacure Therapeutics Ab |
Novel phenyl guanidines
|
|
MXPA03000738A
(es)
|
2000-07-24 |
2003-06-04 |
Ardana Bioscience Ltd |
Antagonistas de grelina.
|
|
DE60113865T2
(de)
|
2000-07-31 |
2006-07-20 |
Vernalis Research Ltd., Winnersh |
Piperazin derivate
|
|
US6768024B1
(en)
|
2000-08-04 |
2004-07-27 |
Lion Bioscience Ag |
Triamine derivative melanocortin receptor ligands and methods of using same
|
|
GB0019359D0
(en)
|
2000-08-07 |
2000-09-27 |
Melacure Therapeutics Ab |
Novel guanidines
|
|
WO2002015845A2
(en)
|
2000-08-21 |
2002-02-28 |
Merck & Co., Inc. |
Anti-hypercholesterolemic drug combination
|
|
JP2004506685A
(ja)
|
2000-08-21 |
2004-03-04 |
グリアテツク・インコーポレイテツド |
食欲の制御と肥満の治療のためのヒスタミンh3受容体逆アゴニストの使用
|
|
WO2002015909A1
(en)
|
2000-08-23 |
2002-02-28 |
Merck & Co., Inc. |
Substituted piperidines as melanocortin receptor agonists
|
|
US6900226B2
(en)
|
2000-09-06 |
2005-05-31 |
Hoffman-La Roche Inc. |
Neuropeptide Y antagonists
|
|
US20020165223A1
(en)
|
2000-09-14 |
2002-11-07 |
Greenlee William J. |
Substituted urea neuropeptide Y Y5 receptor antagonists
|
|
TR200402046T4
(tr)
|
2000-10-13 |
2004-10-21 |
Eli Lilly And Company |
Büyüme hormonu salgılanmasını uyarıcı maddeler olarak ikameli dipeptitler.
|
|
ATE403647T1
(de)
|
2000-10-16 |
2008-08-15 |
Hoffmann La Roche |
Indolinderivate und deren verwendung als 5-ht2 rezeptor liganden
|
|
AP2001002307A0
(en)
|
2000-10-20 |
2001-12-31 |
Pfizer Prod Inc |
B3 adrenergic receptor agonists and uses thereof.
|
|
WO2002036596A2
(en)
|
2000-11-03 |
2002-05-10 |
Wyeth |
CYCLOALKYL[b][1,4]DIAZEPINO[6,7,1-hi]INDOLES AND DERIVATIVES
|
|
DE60142355D1
(de)
|
2000-11-20 |
2010-07-22 |
Biovitrum Ab Publ |
Piperazinylpyrazinverbindungen als agonisten oder antagonisten am serotonin-5ht-2-rezeptor
|
|
AU1529402A
(en)
|
2000-11-20 |
2002-05-27 |
Biovitrum Ab |
Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor
|
|
BR0116113A
(pt)
*
|
2000-12-12 |
2004-08-03 |
Neurogen Corp |
Espiro[isobenzofuran-1,4'-piperidin]-3-onas e 3h-espiroisoben-zofuran-1,4'-piperidinas
|
|
GB0030710D0
(en)
|
2000-12-15 |
2001-01-31 |
Hoffmann La Roche |
Piperazine derivatives
|
|
MXPA03005745A
(es)
|
2000-12-21 |
2003-09-05 |
Schering Corp |
Neuropeptidos heteroarilo urea y antagonista de los receptores y5 del neuropeptido y.
|
|
JP4025200B2
(ja)
|
2000-12-22 |
2007-12-19 |
シェーリング コーポレイション |
ピペリジンmchアンタゴニストおよび肥満の処置におけるそれらの使用
|
|
WO2002051232A2
(en)
|
2000-12-27 |
2002-07-04 |
Actelion Pharmaceuticals Ltd. |
Novel benzazepines and related heterocyclic derivatives
|
|
ES2291374T3
(es)
|
2000-12-27 |
2008-03-01 |
F. Hoffmann-La Roche Ag |
Derivados de indol y su empleo como ligandos receptores de 5-ht2b y 5-ht2c.
|
|
US7157463B2
(en)
|
2001-01-23 |
2007-01-02 |
Eli Lilly And Company |
Substituted piperidines/piperazines as melanocortin receptor agonists
|
|
EP1358163A1
(en)
|
2001-01-23 |
2003-11-05 |
Eli Lilly And Company |
Melanocortin receptor agonists
|
|
ES2247298T3
(es)
|
2001-01-23 |
2006-03-01 |
Eli Lilly And Company |
Derivados de piperazina y piperidina como agonistas del receptor de melanocortina.
|
|
ATE366724T1
(de)
|
2001-02-02 |
2007-08-15 |
Takeda Pharmaceutical |
Kondensierte heterocyclische derivate
|
|
WO2002067869A2
(en)
|
2001-02-28 |
2002-09-06 |
Merck & Co., Inc. |
Acylated piperidine derivatives as melanocortin-4 receptor agonists
|
|
RS63203A
(sr)
|
2001-02-28 |
2006-12-15 |
Merck & Co.Inc. |
Acilovani derivati piperidina kao agonisti receptora melanokortina-4
|
|
US7015235B2
(en)
|
2001-02-28 |
2006-03-21 |
Merck & Co., Inc. |
Acylated piperidine derivatives as melanocortin-4 receptor agonists
|
|
US6900329B2
(en)
|
2001-03-21 |
2005-05-31 |
Schering Corporation |
MCH antagonists and their use in the treatment of obesity
|
|
HUP0400252A3
(en)
|
2001-03-21 |
2011-09-28 |
Pharmacopeia Drug Discovery |
Aryl and biaryl compounds having mch modulatory activity, pharmaceutical compositions containing them and process for producing them
|
|
CN100366614C
(zh)
|
2001-03-22 |
2008-02-06 |
索尔瓦药物有限公司 |
具有cb1-拮抗活性的4,5-二氢-1h-吡唑衍生物
|
|
EP1373212A4
(en)
|
2001-03-29 |
2004-06-23 |
Molecular Design Int |
ADRENERGIC-BETA-3 RECEPTOR AGONISTS, AGONIST COMPOSITIONS AND METHODS OF PREPARING AND USING THE SAME
|
|
MXPA03009353A
(es)
|
2001-04-12 |
2004-02-12 |
Pharmacopeia Inc |
Aril y biaril piperidinas utilizadas como antagonistas de mch.
|
|
US6573287B2
(en)
|
2001-04-12 |
2003-06-03 |
Bristo-Myers Squibb Company |
2,1-oxazoline and 1,2-pyrazoline-based inhibitors of dipeptidyl peptidase IV and method
|
|
FR2824825B1
(fr)
|
2001-05-15 |
2005-05-06 |
Servier Lab |
Nouveaux derives d'alpha-amino-acides, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
|
|
DE60225274T2
(de)
|
2001-05-21 |
2009-03-26 |
F. Hoffmann-La Roche Ag |
Chinolinderivate als liganden für den neuropeptid-y-rezeptor
|
|
WO2002094799A2
(en)
|
2001-05-22 |
2002-11-28 |
Neurogen Corporation |
Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
|
|
US7098239B2
(en)
|
2001-06-20 |
2006-08-29 |
Merck & Co., Inc |
Dipeptidyl peptidase inhibitors for the treatment of diabetes
|
|
US7253172B2
(en)
|
2001-06-20 |
2007-08-07 |
Merck & Co., Inc. |
Dipeptidyl peptidase inhibitors for the treatment of diabetes
|
|
GB0115517D0
(en)
|
2001-06-25 |
2001-08-15 |
Ferring Bv |
Novel antidiabetic agents
|
|
WO2003002593A2
(en)
|
2001-06-27 |
2003-01-09 |
Probiodrug Ag |
Peptide structures useful for competitive modulation of dipeptidyl peptidase iv catalysis
|
|
DE60221983T2
(de)
|
2001-06-27 |
2008-05-15 |
Smithkline Beecham Corp. |
Fluorpyrrolidine als dipeptidyl-peptidase inhibitoren
|
|
ES2296962T3
(es)
|
2001-06-27 |
2008-05-01 |
Smithkline Beecham Corporation |
Pirrolidinas como inhibidores de dipeptidil peptidasa.
|
|
WO2003002531A2
(en)
|
2001-06-27 |
2003-01-09 |
Smithkline Beecham Corporation |
Fluoropyrrolidines as dipeptidyl peptidase inhibitors
|
|
ATE388951T1
(de)
|
2001-07-03 |
2008-03-15 |
Novo Nordisk As |
Dpp-iv-inhibierende purin-derivative zur behandlung von diabetes
|
|
EP1411942A4
(en)
|
2001-07-05 |
2005-01-26 |
Synaptic Pharma Corp |
SUBSTITUTED ANILINPIPERIDINES AS MCH-SELECTIVE ANTAGONISTS
|
|
UA74912C2
(en)
|
2001-07-06 |
2006-02-15 |
Merck & Co Inc |
Beta-aminotetrahydroimidazo-(1,2-a)-pyrazines and tetratriazolo-(4,3-a)-pyrazines as inhibitors of dipeptylpeptidase for the treatment or prevention of diabetes
|
|
ITMI20011483A1
(it)
|
2001-07-11 |
2003-01-11 |
Res & Innovation Soc Coop A R |
Uso di composti come antagonisti funzionali ai recettori centrali deicannabinoidi
|
|
ATE411021T1
(de)
|
2001-07-18 |
2008-10-15 |
Merck & Co Inc |
Überbrückte piperidinderivate als melanocortin- rezeptor-agonisten
|
|
AU2002319627A1
(en)
|
2001-07-20 |
2003-03-03 |
Merck And Co., Inc. |
Substituted imidazoles as cannabinoid receptor modulators
|
|
US6977264B2
(en)
|
2001-07-25 |
2005-12-20 |
Amgen Inc. |
Substituted piperidines and methods of use
|
|
US6915444B2
(en)
|
2001-09-12 |
2005-07-05 |
Rockwell Automation Technologies, Inc. |
Network independent safety protocol for industrial controller using data manipulation techniques
|
|
AU2003302640B2
(en)
*
|
2002-11-29 |
2009-09-24 |
Banyu Pharmaceutical Co., Ltd. |
Novel azole derivatives
|