AR053440A2 - Uso de una forma de dosificacion farmaceutica de liberacion sostenida para la manufactura de un medicamento, dicha forma de dosificacion farmaceutica y una tableta comprimida - Google Patents

Uso de una forma de dosificacion farmaceutica de liberacion sostenida para la manufactura de un medicamento, dicha forma de dosificacion farmaceutica y una tableta comprimida

Info

Publication number
AR053440A2
AR053440A2 ARP060100699A ARP060100699A AR053440A2 AR 053440 A2 AR053440 A2 AR 053440A2 AR P060100699 A ARP060100699 A AR P060100699A AR P060100699 A ARP060100699 A AR P060100699A AR 053440 A2 AR053440 A2 AR 053440A2
Authority
AR
Argentina
Prior art keywords
dosage form
pharmaceutical dosage
phthalate
manufacture
medicinal product
Prior art date
Application number
ARP060100699A
Other languages
English (en)
Original Assignee
Cv Therapeutics Inc
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26796494&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR053440(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Cv Therapeutics Inc, Syntex Inc filed Critical Cv Therapeutics Inc
Publication of AR053440A2 publication Critical patent/AR053440A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Saccharide Compounds (AREA)

Abstract

El uso de ranolazina y por lo menos un aglutinante dependiente del pH seleccionado entre copolímeros de ácido metacrilato, hidroxipropil celulosa ftalato, hidroxipropil metilcelulosa ftalato, celulosa acetato ftalato, polivinil acetato ftalato, polivinilpirrolidina ftalato y mezclas de los mismos, que es para la preparacion de una composicion farmacéutica de liberacion sostenida para tratar a un humano que sufre de una enfermedad cardiovascular seleccionada de arritmias, angina variante e inducida por ejercicio e infarto de miocardio, o claudicacion intermitente donde la composicion farmacéutica es para administracion una o dos veces al día.
ARP060100699A 1998-09-10 2006-02-24 Uso de una forma de dosificacion farmaceutica de liberacion sostenida para la manufactura de un medicamento, dicha forma de dosificacion farmaceutica y una tableta comprimida AR053440A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US9980498P 1998-09-10 1998-09-10
US09/321,522 US6303607B1 (en) 1998-09-10 1999-05-27 Method for administering a sustained release ranolanolazine formulation

Publications (1)

Publication Number Publication Date
AR053440A2 true AR053440A2 (es) 2007-05-09

Family

ID=26796494

Family Applications (3)

Application Number Title Priority Date Filing Date
ARP990104545A AR022085A1 (es) 1998-09-10 1999-09-09 Una forma de dosificacion farmaceutica de liberacion sostenida y una tableta comprimida
ARP060100700A AR052921A1 (es) 1998-09-10 2006-02-24 Uso de ranolazina para la preparacion de una composicion farmaceutica y composicion farmaceutica
ARP060100699A AR053440A2 (es) 1998-09-10 2006-02-24 Uso de una forma de dosificacion farmaceutica de liberacion sostenida para la manufactura de un medicamento, dicha forma de dosificacion farmaceutica y una tableta comprimida

Family Applications Before (2)

Application Number Title Priority Date Filing Date
ARP990104545A AR022085A1 (es) 1998-09-10 1999-09-09 Una forma de dosificacion farmaceutica de liberacion sostenida y una tableta comprimida
ARP060100700A AR052921A1 (es) 1998-09-10 2006-02-24 Uso de ranolazina para la preparacion de una composicion farmaceutica y composicion farmaceutica

Country Status (33)

Country Link
US (14) US6303607B1 (es)
EP (3) EP1096937B9 (es)
JP (2) JP3745621B2 (es)
KR (1) KR100475759B1 (es)
CN (2) CN1193757C (es)
AR (3) AR022085A1 (es)
AT (2) ATE217794T1 (es)
AU (4) AU760435B2 (es)
BR (2) BR9913553A (es)
CA (2) CA2343376C (es)
CY (1) CY2008020I1 (es)
CZ (2) CZ301375B6 (es)
DE (3) DE69901570T2 (es)
DK (2) DK1096937T3 (es)
ES (2) ES2234302T3 (es)
FR (1) FR09C0001I2 (es)
GE (1) GEP20053420B (es)
HK (2) HK1040060A1 (es)
HU (2) HU224215B1 (es)
IL (6) IL141893A0 (es)
LU (1) LU91504I2 (es)
MX (2) MXPA01002599A (es)
NL (1) NL300371I2 (es)
NO (4) NO320986B1 (es)
NZ (2) NZ510386A (es)
PL (3) PL196263B1 (es)
PT (2) PT1096937E (es)
RU (2) RU2207856C2 (es)
SI (2) SI1096937T1 (es)
TR (2) TR200101262T2 (es)
TW (1) TWI241911B (es)
UA (2) UA67793C2 (es)
WO (2) WO2000013687A2 (es)

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Also Published As

Publication number Publication date
EP1096937B1 (en) 2004-12-29
IL141893A (en) 2008-08-07
HUP0103844A2 (hu) 2002-04-29
AU6036499A (en) 2000-03-27
LU91504I2 (fr) 2009-02-03
US6864258B2 (en) 2005-03-08
DK1096937T3 (da) 2005-05-09
DE69901570D1 (de) 2002-06-27
PL347073A1 (en) 2002-03-11
WO2000013686A2 (en) 2000-03-16
IL141892A0 (en) 2002-03-10
US20060217397A1 (en) 2006-09-28
NL300371I2 (nl) 2009-10-01
DK1109558T3 (da) 2002-08-26
AU760435B2 (en) 2003-05-15
ATE285774T1 (de) 2005-01-15
US20030100566A1 (en) 2003-05-29
NO20011191L (no) 2001-04-30
CZ301341B6 (cs) 2010-01-20
HU224215B1 (hu) 2005-06-28
UA67793C2 (uk) 2004-07-15
NO20011192L (no) 2001-04-30
AR022085A1 (es) 2002-09-04
HK1044284A1 (en) 2002-10-18
US20060147521A1 (en) 2006-07-06
US20030166659A1 (en) 2003-09-04
WO2000013687A2 (en) 2000-03-16
NO20011192D0 (no) 2001-03-08
RU2207856C2 (ru) 2003-07-10
CN1354665A (zh) 2002-06-19
US6562826B1 (en) 2003-05-13
NO20011191D0 (no) 2001-03-08
UA75027C2 (uk) 2006-03-15
ES2234302T3 (es) 2005-06-16
HK1044284B (zh) 2005-07-15
CA2342390A1 (en) 2000-03-16
BR9913626A (pt) 2001-12-04
GEP20053420B (en) 2005-01-25
FR09C0001I2 (es) 2009-12-18
PL202207B1 (pl) 2009-06-30
CZ2001879A3 (cs) 2001-08-15
NO2009005I2 (es) 2010-06-28
PL348249A1 (en) 2002-05-20
PL196263B1 (pl) 2007-12-31
US20020090396A1 (en) 2002-07-11
JP2006096757A (ja) 2006-04-13
PT1096937E (pt) 2005-04-29
NZ510386A (en) 2003-08-29
CY2008020I2 (el) 2010-07-28
WO2000013687A3 (en) 2000-06-29
TR200101262T2 (tr) 2001-12-21
CA2343376C (en) 2007-01-09
EP1527779A1 (en) 2005-05-04
HUP0103844A3 (en) 2002-11-28
US6525057B2 (en) 2003-02-25
CN1193757C (zh) 2005-03-23
ES2177346T3 (es) 2002-12-01
US6620814B2 (en) 2003-09-16
HUP0104088A3 (en) 2002-12-28
BR9913553A (pt) 2001-10-23
DE122008000065I1 (de) 2009-04-09
CN1211086C (zh) 2005-07-20
HK1040060A1 (en) 2002-05-24
US20040029890A1 (en) 2004-02-12
NZ510384A (en) 2002-10-25
IL141892A (en) 2006-08-20
CN1321088A (zh) 2001-11-07
TR200101261T2 (tr) 2002-05-21
KR100475759B1 (ko) 2005-03-10
NO20054324L (no) 2001-04-30
CA2343376A1 (en) 2000-03-16
CA2342390C (en) 2006-08-29
AU744071B2 (en) 2002-02-14
MXPA01002598A (es) 2002-04-08
RU2214233C2 (ru) 2003-10-20
LU91504I9 (es) 2019-01-02
ATE217794T1 (de) 2002-06-15
US20050153982A1 (en) 2005-07-14
US6852724B2 (en) 2005-02-08
CY2008020I1 (el) 2010-07-28
NO319434B1 (no) 2005-08-15
DE69901570T2 (de) 2003-01-09
PT1109558E (pt) 2002-10-31
NO2009005I1 (no) 2009-03-16
US20040097514A1 (en) 2004-05-20
IL180864A0 (en) 2007-07-04
EP1096937A2 (en) 2001-05-09
IL175371A0 (en) 2006-09-05
JP2002524416A (ja) 2002-08-06
AR052921A1 (es) 2007-04-11
EP1109558A2 (en) 2001-06-27
DE69922964D1 (de) 2005-02-03
EP1109558B1 (en) 2002-05-22
US20020004506A1 (en) 2002-01-10
HUP0104088A2 (hu) 2002-05-29
DE69922964T2 (de) 2005-12-08
KR20010089874A (ko) 2001-10-12
US20030099705A1 (en) 2003-05-29
TWI241911B (en) 2005-10-21
MXPA01002599A (es) 2005-02-17
JP3745621B2 (ja) 2006-02-15
US6617328B2 (en) 2003-09-09
SI1109558T1 (en) 2002-10-31
AU2008207703A1 (en) 2008-09-25
SI1096937T1 (en) 2005-04-30
NO320986B1 (no) 2006-02-20
NL300371I1 (nl) 2009-02-02
US20050059667A1 (en) 2005-03-17
FR09C0001I1 (es) 2009-02-27
PL196668B1 (pl) 2008-01-31
AU2008207707A1 (en) 2008-09-25
IL141893A0 (en) 2002-03-10
CZ301375B6 (cs) 2010-02-03
US6503911B2 (en) 2003-01-07
US6369062B1 (en) 2002-04-09
WO2000013686A3 (en) 2000-07-06
CZ2001880A3 (cs) 2001-08-15
AU6142599A (en) 2000-03-27
EP1096937B9 (en) 2007-02-28
US6303607B1 (en) 2001-10-16

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