AP2015008277A0 - Novel bicyclic pyridinones - Google Patents

Novel bicyclic pyridinones

Info

Publication number
AP2015008277A0
AP2015008277A0 AP2015008277A AP2015008277A AP2015008277A0 AP 2015008277 A0 AP2015008277 A0 AP 2015008277A0 AP 2015008277 A AP2015008277 A AP 2015008277A AP 2015008277 A AP2015008277 A AP 2015008277A AP 2015008277 A0 AP2015008277 A0 AP 2015008277A0
Authority
AP
ARIPO
Prior art keywords
novel bicyclic
pyridinones
bicyclic pyridinones
novel
bicyclic
Prior art date
Application number
AP2015008277A
Other languages
English (en)
Inventor
Michael Eric Green
Christopher John O'donnell
Martin Youngjin Pettersson
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of AP2015008277A0 publication Critical patent/AP2015008277A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Epidemiology (AREA)
AP2015008277A 2012-09-21 2013-09-06 Novel bicyclic pyridinones AP2015008277A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261703969P 2012-09-21 2012-09-21
PCT/IB2013/058347 WO2014045156A1 (en) 2012-09-21 2013-09-06 Novel bicyclic pyridinones

Publications (1)

Publication Number Publication Date
AP2015008277A0 true AP2015008277A0 (en) 2015-02-28

Family

ID=49585452

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2015008277A AP2015008277A0 (en) 2012-09-21 2013-09-06 Novel bicyclic pyridinones

Country Status (46)

Country Link
US (3) US8916564B2 (forum.php)
EP (1) EP2897956B1 (forum.php)
JP (1) JP5844018B2 (forum.php)
KR (1) KR101725696B1 (forum.php)
CN (1) CN104662021B (forum.php)
AP (1) AP2015008277A0 (forum.php)
AR (1) AR092628A1 (forum.php)
AU (1) AU2013319845B2 (forum.php)
BR (1) BR112015006436A2 (forum.php)
CA (1) CA2882386C (forum.php)
CL (1) CL2015000717A1 (forum.php)
CR (1) CR20150053A (forum.php)
CU (1) CU20150021A7 (forum.php)
CY (1) CY1118662T1 (forum.php)
DK (1) DK2897956T3 (forum.php)
DO (1) DOP2015000069A (forum.php)
EA (1) EA026668B1 (forum.php)
EC (1) ECSP15015594A (forum.php)
ES (1) ES2609987T3 (forum.php)
GE (1) GEP201706659B (forum.php)
GT (1) GT201500069A (forum.php)
HR (1) HRP20161558T1 (forum.php)
HU (1) HUE031248T2 (forum.php)
IL (1) IL237163A (forum.php)
IN (1) IN2015DN01119A (forum.php)
LT (1) LT2897956T (forum.php)
MA (1) MA37886B1 (forum.php)
MD (1) MD4583B1 (forum.php)
ME (1) ME02571B (forum.php)
MX (1) MX360599B (forum.php)
MY (1) MY181891A (forum.php)
NI (1) NI201500038A (forum.php)
NZ (1) NZ704863A (forum.php)
PE (1) PE20150686A1 (forum.php)
PH (1) PH12015500376A1 (forum.php)
PL (1) PL2897956T3 (forum.php)
PT (1) PT2897956T (forum.php)
RS (1) RS55426B1 (forum.php)
SG (1) SG11201501074WA (forum.php)
SI (1) SI2897956T1 (forum.php)
TN (1) TN2015000084A1 (forum.php)
TW (1) TWI500616B (forum.php)
UA (1) UA110688C2 (forum.php)
UY (1) UY35039A (forum.php)
WO (1) WO2014045156A1 (forum.php)
ZA (1) ZA201501195B (forum.php)

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CN104936958B (zh) 2013-01-17 2019-07-26 詹森药业有限公司 作为γ分泌酶调节剂的新颖的经取代的吡啶并-哌嗪酮衍生物
JP6425717B2 (ja) * 2013-10-04 2018-11-21 ファイザー・インク ガンマセクレターゼモジュレーターとしての新規二環式ピリジノン
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PH12021552572A1 (en) 2019-04-08 2022-06-20 Frequency Therapeutics Inc Combination of chir99021 and valproic acid for treating hearing loss
JOP20220130A1 (ar) 2019-12-06 2023-01-30 Vertex Pharma مجموعات تترا هيدروفيوران بها استبدال في صورة عوامل تعديل لقنوات الصوديوم
CN113402490B (zh) * 2021-03-29 2023-01-03 白银京宇新药业有限公司 一种1，2，6，7-四氢-8H-茚并[5，4-b]呋喃-8-酮的制备方法
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