ZA201209381B - The use of inhibitors of bruton's tyrosine kinase (btk) - Google Patents

The use of inhibitors of bruton's tyrosine kinase (btk)

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Publication number
ZA201209381B
ZA201209381B ZA2012/09381A ZA201209381A ZA201209381B ZA 201209381 B ZA201209381 B ZA 201209381B ZA 2012/09381 A ZA2012/09381 A ZA 2012/09381A ZA 201209381 A ZA201209381 A ZA 201209381A ZA 201209381 B ZA201209381 B ZA 201209381B
Authority
ZA
South Africa
Prior art keywords
bruton
btk
inhibitors
tyrosine kinase
tyrosine
Prior art date
Application number
ZA2012/09381A
Other languages
English (en)
Inventor
Joseph J Buggy
Gwen Fyfe
David J Loury
Eric Hedrick
Laurence Elias
Tarak D Mody
Original Assignee
Pharmacylics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45067334&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA201209381(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacylics Inc filed Critical Pharmacylics Inc
Publication of ZA201209381B publication Critical patent/ZA201209381B/en

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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
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