TW209174B - - Google Patents
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- TW209174B TW209174B TW081102828A TW81102828A TW209174B TW 209174 B TW209174 B TW 209174B TW 081102828 A TW081102828 A TW 081102828A TW 81102828 A TW81102828 A TW 81102828A TW 209174 B TW209174 B TW 209174B
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- GLDOVTGHNKAZLK-UHFFFAOYSA-N octadecan-1-ol Chemical compound CCCCCCCCCCCCCCCCCCO GLDOVTGHNKAZLK-UHFFFAOYSA-N 0.000 claims description 6
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- DCXXMTOCNZCJGO-UHFFFAOYSA-N Glycerol trioctadecanoate Natural products CCCCCCCCCCCCCCCCCC(=O)OCC(OC(=O)CCCCCCCCCCCCCCCCC)COC(=O)CCCCCCCCCCCCCCCCC DCXXMTOCNZCJGO-UHFFFAOYSA-N 0.000 claims description 5
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- KIUKXJAPPMFGSW-DNGZLQJQSA-N (2S,3S,4S,5R,6R)-6-[(2S,3R,4R,5S,6R)-3-Acetamido-2-[(2S,3S,4R,5R,6R)-6-[(2R,3R,4R,5S,6R)-3-acetamido-2,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-2-carboxy-4,5-dihydroxyoxan-3-yl]oxy-5-hydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-3,4,5-trihydroxyoxane-2-carboxylic acid Chemical compound CC(=O)N[C@H]1[C@H](O)O[C@H](CO)[C@@H](O)[C@@H]1O[C@H]1[C@H](O)[C@@H](O)[C@H](O[C@H]2[C@@H]([C@@H](O[C@H]3[C@@H]([C@@H](O)[C@H](O)[C@H](O3)C(O)=O)O)[C@H](O)[C@@H](CO)O2)NC(C)=O)[C@@H](C(O)=O)O1 KIUKXJAPPMFGSW-DNGZLQJQSA-N 0.000 claims 1
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- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
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- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
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- Oncology (AREA)
- Communicable Diseases (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| JP11674591 | 1991-04-19 | ||
| JP22515591 | 1991-08-09 |
Publications (1)
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| TW209174B true TW209174B (en:Method) | 1993-07-11 |
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| TW081102828A TW209174B (en:Method) | 1991-04-19 | 1992-04-11 |
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| EP (1) | EP0514008B1 (en:Method) |
| JP (4) | JP3272029B2 (en:Method) |
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| GR (1) | GR3023383T3 (en:Method) |
| SG (1) | SG50480A1 (en:Method) |
| TW (1) | TW209174B (en:Method) |
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-
1992
- 1992-04-11 TW TW081102828A patent/TW209174B/zh active
- 1992-04-14 SG SG1996002366A patent/SG50480A1/en unknown
- 1992-04-14 DK DK92303357.5T patent/DK0514008T3/da active
- 1992-04-14 EP EP92303357A patent/EP0514008B1/en not_active Expired - Lifetime
- 1992-04-14 AT AT92303357T patent/ATE149348T1/de not_active IP Right Cessation
- 1992-04-14 ES ES92303357T patent/ES2098447T3/es not_active Expired - Lifetime
- 1992-04-14 DE DE69217711T patent/DE69217711T2/de not_active Expired - Fee Related
- 1992-04-15 JP JP12268192A patent/JP3272029B2/ja not_active Expired - Fee Related
- 1992-04-16 CA CA002066384A patent/CA2066384C/en not_active Expired - Fee Related
- 1992-04-18 KR KR1019920006554A patent/KR100217165B1/ko not_active Expired - Fee Related
-
1995
- 1995-03-29 US US08/412,591 patent/US5576025A/en not_active Expired - Lifetime
-
1996
- 1996-08-20 US US08/697,166 patent/US5731006A/en not_active Expired - Fee Related
-
1997
- 1997-05-09 GR GR970401036T patent/GR3023383T3/el unknown
- 1997-12-18 US US08/993,314 patent/US6368635B1/en not_active Expired - Fee Related
-
2001
- 2001-05-11 JP JP2001141178A patent/JP2001354593A/ja active Pending
- 2001-05-11 JP JP2001141179A patent/JP4084000B2/ja not_active Expired - Fee Related
-
2002
- 2002-02-20 US US10/077,896 patent/US20020142041A1/en not_active Abandoned
-
2007
- 2007-07-09 JP JP2007179258A patent/JP2007246547A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| KR920019336A (ko) | 1992-11-19 |
| US20020142041A1 (en) | 2002-10-03 |
| GR3023383T3 (en) | 1997-08-29 |
| CA2066384C (en) | 2007-04-03 |
| EP0514008A1 (en) | 1992-11-19 |
| JP2001354593A (ja) | 2001-12-25 |
| JP3272029B2 (ja) | 2002-04-08 |
| CA2066384A1 (en) | 1992-10-20 |
| JP4084000B2 (ja) | 2008-04-30 |
| JP2001354550A (ja) | 2001-12-25 |
| US5576025A (en) | 1996-11-19 |
| SG50480A1 (en) | 1998-07-20 |
| KR100217165B1 (ko) | 1999-09-01 |
| US6368635B1 (en) | 2002-04-09 |
| EP0514008B1 (en) | 1997-03-05 |
| DK0514008T3 (da) | 1997-05-12 |
| DE69217711T2 (de) | 1997-07-17 |
| JPH05132416A (ja) | 1993-05-28 |
| ATE149348T1 (de) | 1997-03-15 |
| ES2098447T3 (es) | 1997-05-01 |
| JP2007246547A (ja) | 2007-09-27 |
| DE69217711D1 (de) | 1997-04-10 |
| US5731006A (en) | 1998-03-24 |
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