SK283193B6 - Spôsob prípravy purínových zlúčenín a medziprodukty - Google Patents

Spôsob prípravy purínových zlúčenín a medziprodukty Download PDF

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Publication number
SK283193B6
SK283193B6 SK1332-96A SK133296A SK283193B6 SK 283193 B6 SK283193 B6 SK 283193B6 SK 133296 A SK133296 A SK 133296A SK 283193 B6 SK283193 B6 SK 283193B6
Authority
SK
Slovakia
Prior art keywords
formula
compound
amino
preparation
hydrogen
Prior art date
Application number
SK1332-96A
Other languages
English (en)
Slovak (sk)
Other versions
SK133296A3 (en
Inventor
John Robert Mansfield Dales
Original Assignee
Novartis International Pharmaceutical Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis International Pharmaceutical Ltd. filed Critical Novartis International Pharmaceutical Ltd.
Publication of SK133296A3 publication Critical patent/SK133296A3/sk
Publication of SK283193B6 publication Critical patent/SK283193B6/sk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Chemical Treatment Of Metals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
SK1332-96A 1994-04-19 1995-04-19 Spôsob prípravy purínových zlúčenín a medziprodukty SK283193B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9407698A GB9407698D0 (en) 1994-04-19 1994-04-19 Pharmaceuticals
PCT/EP1995/001840 WO1995028402A2 (en) 1994-04-19 1995-04-19 Preparation of purines

Publications (2)

Publication Number Publication Date
SK133296A3 SK133296A3 (en) 1997-05-07
SK283193B6 true SK283193B6 (sk) 2003-03-04

Family

ID=10753741

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1332-96A SK283193B6 (sk) 1994-04-19 1995-04-19 Spôsob prípravy purínových zlúčenín a medziprodukty

Country Status (40)

Country Link
US (2) US6846927B1 (ja)
EP (1) EP0756597B1 (ja)
JP (1) JP3936734B2 (ja)
KR (1) KR100327147B1 (ja)
CN (1) CN1045963C (ja)
AP (2) AP582A (ja)
AT (1) ATE201209T1 (ja)
AU (1) AU691000B2 (ja)
BG (1) BG63464B1 (ja)
BR (1) BR9507494A (ja)
CA (1) CA2188181C (ja)
CZ (1) CZ287674B6 (ja)
DE (1) DE69520945T2 (ja)
DK (1) DK0756597T3 (ja)
DZ (1) DZ1872A1 (ja)
EG (1) EG20938A (ja)
ES (1) ES2158948T3 (ja)
FI (1) FI119691B (ja)
GB (1) GB9407698D0 (ja)
GR (1) GR3036338T3 (ja)
HK (1) HK1012348A1 (ja)
HU (1) HU226209B1 (ja)
IL (1) IL113409A (ja)
IN (1) IN183830B (ja)
MA (1) MA23518A1 (ja)
MX (1) MX9604942A (ja)
MY (1) MY128846A (ja)
NO (1) NO315000B1 (ja)
NZ (1) NZ287858A (ja)
OA (1) OA10376A (ja)
PL (1) PL181219B1 (ja)
PT (1) PT756597E (ja)
RO (1) RO118950B1 (ja)
RU (1) RU2158266C2 (ja)
SA (1) SA95150619B1 (ja)
SK (1) SK283193B6 (ja)
TW (1) TW311138B (ja)
UA (1) UA47401C2 (ja)
WO (1) WO1995028402A2 (ja)
ZA (1) ZA953110B (ja)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9615253D0 (en) * 1996-07-20 1996-09-04 Smithkline Beecham Plc Pharmaceuticals
GB9615276D0 (en) * 1996-07-20 1996-09-04 Smithkline Beecham Plc Pharmaceuticals
GB9807114D0 (en) * 1998-04-02 1998-06-03 Smithkline Beecham Plc Novel process
GB9807116D0 (en) * 1998-04-02 1998-06-03 Smithkline Beecham Plc Novel process
AU2003268213A1 (en) * 2002-08-26 2004-03-11 Teva Pharmaceutical Industries Ltd. Crystalline solid famciclovir forms i, ii, iii and preparation thereof
US20040266795A1 (en) * 2003-04-30 2004-12-30 Genny Shamai Process for the preparation of famciclovir
EP1556383A1 (en) * 2003-09-04 2005-07-27 Teva Pharmaceutical Industries Ltd. Process for preparing famciclovir
US7458839B2 (en) * 2006-02-21 2008-12-02 Fci Americas Technology, Inc. Electrical connectors having power contacts with alignment and/or restraining features
US20050215787A1 (en) * 2004-03-26 2005-09-29 Joshi Ramesh A An improved process for the preparation of purines
EP1747223A1 (en) * 2004-05-18 2007-01-31 Teva Pharmaceutical Industries Ltd. Drying process for preparing crystalline solid famciclovir
GB2426247A (en) * 2005-05-20 2006-11-22 Arrow Int Ltd Methods of preparing purine derivatives such as famciclovir
CN102070636B (zh) * 2011-01-17 2012-05-23 浙江大学 喷昔洛韦的制备方法
CN104086552B (zh) * 2014-07-31 2016-01-13 济南兆康医药科技有限公司 一种喷昔洛韦的精制方法
CN104496991A (zh) * 2014-11-04 2015-04-08 常州康丽制药有限公司 高品质2-氨基-6-氯-9-(4-羟基-3–羟甲基丁基)嘌呤的制备方法
CN104744472A (zh) * 2015-03-12 2015-07-01 常州康丽制药有限公司 高品质2-氨基-6-氯-9-(4-羟基-3-羟甲基丁基)嘌呤的制备方法
CN108314685B (zh) * 2018-03-16 2020-08-25 上药康丽(常州)药业有限公司 一种2-氨基-6-氯-9-(4-乙酰氧基-3-乙酰氧甲基丁基)嘌呤的制备方法
CN110713490A (zh) * 2018-07-12 2020-01-21 浙江医药股份有限公司新昌制药厂 一种喷昔洛韦的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3485225D1 (de) * 1983-08-18 1991-12-05 Beecham Group Plc Antivirale guanin-derivate.
EP0182024B1 (en) * 1984-09-20 1991-04-03 Beecham Group Plc Purine derivatives and their pharmaceutical use
EP0302644B1 (en) * 1987-08-01 1997-01-29 Beecham Group Plc Purine compounds and their preparation
GB8817607D0 (en) * 1988-07-23 1988-09-01 Beecham Group Plc Novel process
GB8822236D0 (en) * 1988-09-21 1988-10-26 Beecham Group Plc Chemical process

Also Published As

Publication number Publication date
CN1150427A (zh) 1997-05-21
FI119691B (fi) 2009-02-13
WO1995028402A3 (en) 1996-01-25
US6846927B1 (en) 2005-01-25
ATE201209T1 (de) 2001-06-15
IL113409A0 (en) 1995-07-31
SA95150619B1 (ar) 2005-05-04
FI964193A0 (fi) 1996-10-18
SK133296A3 (en) 1997-05-07
AU691000B2 (en) 1998-05-07
US20050101570A1 (en) 2005-05-12
MY128846A (en) 2007-02-28
GB9407698D0 (en) 1994-06-15
AP703A (en) 1998-12-04
MX9604942A (es) 1998-05-31
RU2158266C2 (ru) 2000-10-27
CZ287674B6 (en) 2001-01-17
OA10376A (en) 2001-11-20
PL316943A1 (en) 1997-02-17
AP582A (en) 1997-04-09
CA2188181C (en) 2007-04-17
GR3036338T3 (en) 2001-11-30
DE69520945T2 (de) 2002-03-28
BR9507494A (pt) 1997-08-12
BG63464B1 (bg) 2002-02-28
HU226209B1 (en) 2008-06-30
FI964193A (fi) 1996-12-18
NZ287858A (en) 1998-06-26
DK0756597T3 (da) 2001-08-20
PT756597E (pt) 2001-11-30
TW311138B (ja) 1997-07-21
DE69520945D1 (de) 2001-06-21
HK1012348A1 (en) 1999-07-30
CZ305396A3 (en) 1997-06-11
DZ1872A1 (fr) 2002-02-17
AP9500730A0 (en) 1995-04-30
AP9600870A0 (en) 1996-10-31
HU9602891D0 (en) 1996-12-30
JP3936734B2 (ja) 2007-06-27
NO964395D0 (no) 1996-10-15
NO964395L (no) 1996-10-15
CN1045963C (zh) 1999-10-27
AU2670695A (en) 1995-11-10
EP0756597A1 (en) 1997-02-05
CA2188181A1 (en) 1995-10-26
IN183830B (ja) 2000-04-29
JPH09512000A (ja) 1997-12-02
EG20938A (en) 2000-06-28
BG100926A (en) 1997-07-31
ZA953110B (en) 1996-05-20
NO315000B1 (no) 2003-06-23
ES2158948T3 (es) 2001-09-16
US7355043B2 (en) 2008-04-08
HUT75339A (en) 1997-05-28
PL181219B1 (pl) 2001-06-29
UA47401C2 (uk) 2002-07-15
RO118950B1 (ro) 2004-01-30
EP0756597B1 (en) 2001-05-16
WO1995028402A2 (en) 1995-10-26
KR970702280A (ko) 1997-05-13
MA23518A1 (fr) 1995-12-31
IL113409A (en) 1999-08-17
KR100327147B1 (ko) 2002-07-27

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MK4A Patent expired

Expiry date: 20150419