RS51873B - So fosforne kiseline i inhibitora dipeptidil peptidaze-iv - Google Patents

So fosforne kiseline i inhibitora dipeptidil peptidaze-iv

Info

Publication number
RS51873B
RS51873B YU20050947A YUP20050947A RS51873B RS 51873 B RS51873 B RS 51873B YU 20050947 A YU20050947 A YU 20050947A YU P20050947 A YUP20050947 A YU P20050947A RS 51873 B RS51873 B RS 51873B
Authority
RS
Serbia
Prior art keywords
phosphoric acid
dipeptidyl peptidase
inhibitor
acid salt
trifluorophenyl
Prior art date
Application number
YU20050947A
Other languages
English (en)
Inventor
Stephen Howard Cypes
Alex Minhua Chen
Russell R. Ferlita
Karl Hansen
Ivan Lee
Vicky K. Vydra
Robert M. Wenslow Jr.
Original Assignee
Merck Sharp & Dohme Corp.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33563839&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS51873(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck Sharp & Dohme Corp. filed Critical Merck Sharp & Dohme Corp.
Priority to MEP-2008-602A priority Critical patent/ME00405B/me
Publication of RS20050947A publication Critical patent/RS20050947A/sr
Publication of RS51873B publication Critical patent/RS51873B/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

SO FOSFORNE KISELINE I INHIBITORA DIPEPTIDIL PEPTIDAZE-IV. Dihidrogenfosfatna so 4-okso-4-[3-(trifluorometil)-5,6-dihidro[l,2,4]triazolo[4,3-a]pirazin-7(8H)-il]-l-(2,4,5-trifluorofenil)butan-2-amina strukturne formule II koja ima (R)-konfiguraciju na hiralnom centru označenom sa *ili njen farmaceutski prihvatljiv hidrat.Prijava sadrži još 19 patentnih zahteva.
YU20050947A 2003-06-24 2004-06-18 So fosforne kiseline i inhibitora dipeptidil peptidaze-iv RS51873B (sr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
MEP-2008-602A ME00405B (me) 2003-06-24 2004-06-18 So fosforne kiseline i inhibitora dipeptidil peptidaze-IV

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US48216103P 2003-06-24 2003-06-24
PCT/US2004/019683 WO2005003135A1 (en) 2003-06-24 2004-06-18 Phosphoric acid salt of a dipeptidyl peptidase-iv inhibitor

Publications (2)

Publication Number Publication Date
RS20050947A RS20050947A (en) 2008-04-04
RS51873B true RS51873B (sr) 2012-02-29

Family

ID=33563839

Family Applications (1)

Application Number Title Priority Date Filing Date
YU20050947A RS51873B (sr) 2003-06-24 2004-06-18 So fosforne kiseline i inhibitora dipeptidil peptidaze-iv

Country Status (41)

Country Link
US (1) US7326708B2 (sr)
EP (1) EP1654263B2 (sr)
JP (1) JP4463768B2 (sr)
KR (2) KR101016569B1 (sr)
CN (1) CN100430397C (sr)
AR (2) AR044705A1 (sr)
AT (1) ATE373003T1 (sr)
AU (1) AU2004253889B2 (sr)
BR (1) BRPI0411726B8 (sr)
CA (1) CA2529400C (sr)
CO (1) CO5660266A2 (sr)
CR (1) CR8117A (sr)
CY (1) CY1106936T1 (sr)
DE (1) DE602004008938T3 (sr)
DK (1) DK1654263T4 (sr)
DO (1) DOP2004000941A (sr)
EA (1) EA009042B1 (sr)
EC (1) ECSP056245A (sr)
ES (1) ES2291907T5 (sr)
GE (1) GEP20084489B (sr)
HK (1) HK1095144A1 (sr)
HR (1) HRP20070534T4 (sr)
IL (1) IL172563A (sr)
IS (1) IS2792B (sr)
JO (1) JO2625B1 (sr)
MA (1) MA27861A1 (sr)
ME (1) ME00405B (sr)
MX (1) MXPA05013931A (sr)
MY (1) MY139595A (sr)
NO (1) NO335371B1 (sr)
NZ (1) NZ544026A (sr)
PE (1) PE20050696A1 (sr)
PL (1) PL1654263T5 (sr)
PT (1) PT1654263E (sr)
RS (1) RS51873B (sr)
SI (1) SI1654263T2 (sr)
TN (1) TNSN05329A1 (sr)
TW (1) TWI347185B (sr)
UA (1) UA86026C2 (sr)
WO (1) WO2005003135A1 (sr)
ZA (1) ZA200509933B (sr)

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