PE23196A1 - Compuesto util para tratar infecciones por retrovirus - Google Patents

Compuesto util para tratar infecciones por retrovirus

Info

Publication number
PE23196A1
PE23196A1 PE1995268036A PE26803695A PE23196A1 PE 23196 A1 PE23196 A1 PE 23196A1 PE 1995268036 A PE1995268036 A PE 1995268036A PE 26803695 A PE26803695 A PE 26803695A PE 23196 A1 PE23196 A1 PE 23196A1
Authority
PE
Peru
Prior art keywords
het
cyclopropyl
zero
useful compound
nr12so2
Prior art date
Application number
PE1995268036A
Other languages
English (en)
Spanish (es)
Inventor
Joseph Walter Strohbach
Karen Rene Romines
Ruben A Tommasi
Suvit Thaisrivongs
Harvey Irving Skulnick
Joel Morris
Gordon L Bundy
George P Luke
Paul Adrian Aristoff
Louis L Skaletzky
Ronald B Gammill
Theresa M Schwartz
Steven Ronald Turner
Paul D Johnson
David John Anderson
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of PE23196A1 publication Critical patent/PE23196A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/32—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/34—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D309/36—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C07D309/38—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms one oxygen atom in position 2 or 4, e.g. pyrones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/74—Benzo[b]pyrans, hydrogenated in the carbocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pyrane Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PE1995268036A 1994-05-06 1995-05-08 Compuesto util para tratar infecciones por retrovirus PE23196A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23881794A 1994-05-06 1994-05-06
US34936194A 1994-12-02 1994-12-02

Publications (1)

Publication Number Publication Date
PE23196A1 true PE23196A1 (es) 1996-06-07

Family

ID=26931995

Family Applications (1)

Application Number Title Priority Date Filing Date
PE1995268036A PE23196A1 (es) 1994-05-06 1995-05-08 Compuesto util para tratar infecciones por retrovirus

Country Status (32)

Country Link
US (2) US5852195A (OSRAM)
EP (1) EP0758327B1 (OSRAM)
JP (1) JP3883206B2 (OSRAM)
KR (1) KR100445929B1 (OSRAM)
CN (2) CN1154642C (OSRAM)
AT (1) ATE236894T1 (OSRAM)
AU (2) AU701965B2 (OSRAM)
BR (1) BR9507615A (OSRAM)
CA (2) CA2187523C (OSRAM)
CO (1) CO4810313A1 (OSRAM)
CZ (1) CZ296515B6 (OSRAM)
DE (2) DE122006000014I2 (OSRAM)
DK (1) DK0758327T3 (OSRAM)
ES (1) ES2192201T3 (OSRAM)
FI (1) FI117387B (OSRAM)
FR (1) FR05C0047I2 (OSRAM)
HU (1) HU228057B1 (OSRAM)
IL (3) IL129871A (OSRAM)
LU (1) LU91220I2 (OSRAM)
MX (1) MX9605391A (OSRAM)
MY (2) MY127701A (OSRAM)
NL (1) NL300216I2 (OSRAM)
NO (2) NO315799B1 (OSRAM)
NZ (1) NZ285510A (OSRAM)
PE (1) PE23196A1 (OSRAM)
PL (1) PL190540B1 (OSRAM)
PT (1) PT758327E (OSRAM)
RU (1) RU2139284C1 (OSRAM)
SI (1) SI0758327T1 (OSRAM)
SK (1) SK284407B6 (OSRAM)
TW (1) TW504507B (OSRAM)
WO (1) WO1995030670A2 (OSRAM)

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SI0999826T1 (en) * 1997-07-29 2004-12-31 Pharmacia & Upjohn Company Self-emulsifying formulation for lipophilic compounds
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IL129871A (en) 2003-11-23
NO315799B1 (no) 2003-10-27
KR970702858A (ko) 1997-06-10
RU2139284C1 (ru) 1999-10-10
FI964441L (fi) 1996-11-05
NO964676D0 (no) 1996-11-05
NO964676L (no) 1997-01-06
JP3883206B2 (ja) 2007-02-21
ATE236894T1 (de) 2003-04-15
HU228057B1 (en) 2012-09-28
CN1154642C (zh) 2004-06-23
US5852195A (en) 1998-12-22
HUT77601A (hu) 1998-06-29
MX9605391A (es) 1997-12-31
FR05C0047I2 (OSRAM) 2007-10-19
EP0758327B1 (en) 2003-04-09
DE122006000014I1 (de) 2006-11-16
HU9603074D0 (en) 1997-01-28
NL300216I1 (nl) 2006-04-03
CA2560489C (en) 2010-01-12
HK1084667A1 (en) 2006-08-04
CN1150424A (zh) 1997-05-21
SK138496A3 (en) 1997-06-04
CA2187523A1 (en) 1995-11-16
TW504507B (en) 2002-10-01
SI0758327T1 (en) 2003-08-31
IL129871A0 (en) 2000-02-29
EP0758327A1 (en) 1997-02-19
NO2006003I2 (no) 2008-10-20
NZ285510A (en) 1998-03-25
NL300216I2 (nl) 2006-06-01
KR100445929B1 (ko) 2005-09-30
WO1995030670A3 (en) 1996-04-25
AU718117B2 (en) 2000-04-06
FR05C0047I1 (OSRAM) 2006-03-10
BR9507615A (pt) 1997-09-09
PL190540B1 (pl) 2005-12-30
IL113567A (en) 2003-05-29
MY127701A (en) 2006-12-29
DE69530294T2 (de) 2003-12-24
FI117387B (fi) 2006-09-29
LU91220I2 (fr) 2006-04-10
ES2192201T3 (es) 2003-10-01
CZ317296A3 (en) 1997-04-16
CA2560489A1 (en) 1995-11-16
NO2006003I1 (no) 2006-03-13
PL317061A1 (en) 1997-03-03
CN1329378C (zh) 2007-08-01
HK1066796A1 (zh) 2005-04-01
MY149862A (en) 2013-10-31
AU2368699A (en) 1999-06-03
SK284407B6 (sk) 2005-03-04
CZ296515B6 (cs) 2006-04-12
JPH09512821A (ja) 1997-12-22
DE69530294D1 (de) 2003-05-15
DK0758327T3 (da) 2003-07-28
AU2462695A (en) 1995-11-29
FI964441A0 (fi) 1996-11-05
DE122006000014I2 (de) 2007-03-29
PT758327E (pt) 2003-08-29
US6169181B1 (en) 2001-01-02
CA2187523C (en) 2006-11-21
CO4810313A1 (es) 1999-06-30
AU701965B2 (en) 1999-02-11
CN1539825A (zh) 2004-10-27
WO1995030670A2 (en) 1995-11-16

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