LU91220I2 - Tipranavir ou un de ses sels pharmaceutiques (aptivus) - Google Patents

Tipranavir ou un de ses sels pharmaceutiques (aptivus)

Info

Publication number
LU91220I2
LU91220I2 LU91220C LU91220C LU91220I2 LU 91220 I2 LU91220 I2 LU 91220I2 LU 91220 C LU91220 C LU 91220C LU 91220 C LU91220 C LU 91220C LU 91220 I2 LU91220 I2 LU 91220I2
Authority
LU
Luxembourg
Prior art keywords
aptivus
tipranavir
ones
pharmaceutical salt
pyran
Prior art date
Application number
LU91220C
Other languages
English (en)
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of LU91220I2 publication Critical patent/LU91220I2/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/32Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/34Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D309/36Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C07D309/38Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms one oxygen atom in position 2 or 4, e.g. pyrones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/74Benzo[b]pyrans, hydrogenated in the carbocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pyrane Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
LU91220C 1994-05-06 2006-02-08 Tipranavir ou un de ses sels pharmaceutiques (aptivus) LU91220I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23881794A 1994-05-06 1994-05-06
US34936194A 1994-12-02 1994-12-02

Publications (1)

Publication Number Publication Date
LU91220I2 true LU91220I2 (fr) 2006-04-10

Family

ID=26931995

Family Applications (1)

Application Number Title Priority Date Filing Date
LU91220C LU91220I2 (fr) 1994-05-06 2006-02-08 Tipranavir ou un de ses sels pharmaceutiques (aptivus)

Country Status (33)

Country Link
US (2) US5852195A (fr)
EP (1) EP0758327B1 (fr)
JP (1) JP3883206B2 (fr)
KR (1) KR100445929B1 (fr)
CN (2) CN1329378C (fr)
AT (1) ATE236894T1 (fr)
AU (2) AU701965B2 (fr)
BR (1) BR9507615A (fr)
CA (2) CA2560489C (fr)
CO (1) CO4810313A1 (fr)
CZ (1) CZ296515B6 (fr)
DE (2) DE122006000014I2 (fr)
DK (1) DK0758327T3 (fr)
ES (1) ES2192201T3 (fr)
FI (1) FI117387B (fr)
FR (1) FR05C0047I2 (fr)
HK (2) HK1066796A1 (fr)
HU (1) HU228057B1 (fr)
IL (3) IL129871A (fr)
LU (1) LU91220I2 (fr)
MX (1) MX9605391A (fr)
MY (2) MY149862A (fr)
NL (1) NL300216I2 (fr)
NO (2) NO315799B1 (fr)
NZ (1) NZ285510A (fr)
PE (1) PE23196A1 (fr)
PL (1) PL190540B1 (fr)
PT (1) PT758327E (fr)
RU (1) RU2139284C1 (fr)
SI (1) SI0758327T1 (fr)
SK (1) SK284407B6 (fr)
TW (1) TW504507B (fr)
WO (1) WO1995030670A2 (fr)

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CZ317296A3 (en) 1997-04-16
AU718117B2 (en) 2000-04-06
EP0758327B1 (fr) 2003-04-09
US5852195A (en) 1998-12-22
CN1329378C (zh) 2007-08-01
CA2560489C (fr) 2010-01-12
CN1150424A (zh) 1997-05-21
NZ285510A (en) 1998-03-25
FR05C0047I1 (fr) 2006-03-10
NO315799B1 (no) 2003-10-27
US6169181B1 (en) 2001-01-02
IL129871A0 (en) 2000-02-29
CN1539825A (zh) 2004-10-27
DE122006000014I2 (de) 2007-03-29
WO1995030670A3 (fr) 1996-04-25
CA2187523C (fr) 2006-11-21
SK138496A3 (en) 1997-06-04
PT758327E (pt) 2003-08-29
HK1066796A1 (en) 2005-04-01
FR05C0047I2 (fr) 2007-10-19
SK284407B6 (sk) 2005-03-04
PL190540B1 (pl) 2005-12-30
WO1995030670A2 (fr) 1995-11-16
HUT77601A (hu) 1998-06-29
HU9603074D0 (en) 1997-01-28
CZ296515B6 (cs) 2006-04-12
JPH09512821A (ja) 1997-12-22
DE69530294T2 (de) 2003-12-24
JP3883206B2 (ja) 2007-02-21
DE69530294D1 (de) 2003-05-15
IL129871A (en) 2003-11-23
DK0758327T3 (da) 2003-07-28
CO4810313A1 (es) 1999-06-30
FI964441A (fi) 1996-11-05
NO964676D0 (no) 1996-11-05
HK1084667A1 (en) 2006-08-04
KR100445929B1 (ko) 2005-09-30
TW504507B (en) 2002-10-01
MY149862A (en) 2013-10-31
KR970702858A (ko) 1997-06-10
NL300216I2 (nl) 2006-06-01
MY127701A (en) 2006-12-29
AU2462695A (en) 1995-11-29
AU2368699A (en) 1999-06-03
PE23196A1 (es) 1996-06-07
MX9605391A (es) 1997-12-31
NO2006003I1 (no) 2006-03-13
BR9507615A (pt) 1997-09-09
EP0758327A1 (fr) 1997-02-19
PL317061A1 (en) 1997-03-03
CN1154642C (zh) 2004-06-23
NO964676L (no) 1997-01-06
ATE236894T1 (de) 2003-04-15
AU701965B2 (en) 1999-02-11
CA2187523A1 (fr) 1995-11-16
FI117387B (fi) 2006-09-29
DE122006000014I1 (de) 2006-11-16
RU2139284C1 (ru) 1999-10-10
CA2560489A1 (fr) 1995-11-16
SI0758327T1 (en) 2003-08-31
NL300216I1 (nl) 2006-04-03
ES2192201T3 (es) 2003-10-01
IL113567A (en) 2003-05-29
NO2006003I2 (no) 2008-10-20
HU228057B1 (en) 2012-09-28
FI964441A0 (fi) 1996-11-05

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