ATE265847T1 - Selbstemulgierbare formulierung enthaltend lipophile verbindungen - Google Patents

Selbstemulgierbare formulierung enthaltend lipophile verbindungen

Info

Publication number
ATE265847T1
ATE265847T1 AT98936889T AT98936889T ATE265847T1 AT E265847 T1 ATE265847 T1 AT E265847T1 AT 98936889 T AT98936889 T AT 98936889T AT 98936889 T AT98936889 T AT 98936889T AT E265847 T1 ATE265847 T1 AT E265847T1
Authority
AT
Austria
Prior art keywords
diglyceride
monoglyceride
self
emulsifable
formulation containing
Prior art date
Application number
AT98936889T
Other languages
English (en)
Inventor
Walter Morozowich
Ping Gao
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Application granted granted Critical
Publication of ATE265847T1 publication Critical patent/ATE265847T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4433Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
AT98936889T 1997-07-29 1998-07-27 Selbstemulgierbare formulierung enthaltend lipophile verbindungen ATE265847T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5407897P 1997-07-29 1997-07-29
US5401297P 1997-07-29 1997-07-29
PCT/US1998/014818 WO1999006024A1 (en) 1997-07-29 1998-07-27 Self-emulsifying formulation for lipophilic compounds

Publications (1)

Publication Number Publication Date
ATE265847T1 true ATE265847T1 (de) 2004-05-15

Family

ID=26732506

Family Applications (1)

Application Number Title Priority Date Filing Date
AT98936889T ATE265847T1 (de) 1997-07-29 1998-07-27 Selbstemulgierbare formulierung enthaltend lipophile verbindungen

Country Status (23)

Country Link
EP (1) EP0999826B1 (de)
JP (2) JP2002511099A (de)
KR (1) KR100509776B1 (de)
CN (1) CN1208047C (de)
AT (1) ATE265847T1 (de)
AU (1) AU728698B2 (de)
BR (1) BR9811058A (de)
CA (1) CA2294031E (de)
CZ (1) CZ297206B6 (de)
DE (1) DE69823663T2 (de)
DK (1) DK0999826T3 (de)
ES (1) ES2219895T3 (de)
FI (1) FI20000170A (de)
HK (1) HK1028883A1 (de)
HU (1) HU226114B1 (de)
NO (1) NO328591B1 (de)
NZ (1) NZ502569A (de)
PL (1) PL191780B1 (de)
PT (1) PT999826E (de)
RU (1) RU2211021C2 (de)
SI (1) SI0999826T1 (de)
SK (1) SK284511B6 (de)
WO (1) WO1999006024A1 (de)

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Also Published As

Publication number Publication date
DE69823663T2 (de) 2005-05-19
PL191780B1 (pl) 2006-07-31
EP0999826A1 (de) 2000-05-17
HU226114B1 (en) 2008-04-28
PT999826E (pt) 2004-09-30
SK172000A3 (en) 2000-07-11
AU728698B2 (en) 2001-01-18
AU8573998A (en) 1999-02-22
EP0999826B1 (de) 2004-05-06
KR100509776B1 (ko) 2005-08-24
NO328591B1 (no) 2010-03-29
CN1208047C (zh) 2005-06-29
SK284511B6 (sk) 2005-05-05
NO20000467D0 (no) 2000-01-28
NO20000467L (no) 2000-03-29
JP5227301B2 (ja) 2013-07-03
KR20010022365A (ko) 2001-03-15
NZ502569A (en) 2002-05-31
DK0999826T3 (da) 2004-07-26
BR9811058A (pt) 2000-09-05
CZ297206B6 (cs) 2006-10-11
CN1261790A (zh) 2000-08-02
FI20000170A (fi) 2000-01-28
DE69823663D1 (de) 2004-06-09
HUP0002486A1 (hu) 2000-12-28
JP2002511099A (ja) 2002-04-09
SI0999826T1 (en) 2004-12-31
CZ2000157A3 (cs) 2000-05-17
ES2219895T3 (es) 2004-12-01
CA2294031C (en) 2005-01-18
CA2294031E (en) 2012-04-03
WO1999006024A1 (en) 1999-02-11
HK1028883A1 (en) 2001-03-09
CA2294031A1 (en) 1999-02-11
PL338509A1 (en) 2000-11-06
RU2211021C2 (ru) 2003-08-27
HUP0002486A3 (en) 2001-03-28
JP2010070562A (ja) 2010-04-02

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