NO332383B1 - Makrosykliske forbindelser, anvendelse derav til fremstilling av et medikament, og farmasoytisk preparat som omfatter forbindelsen - Google Patents

Makrosykliske forbindelser, anvendelse derav til fremstilling av et medikament, og farmasoytisk preparat som omfatter forbindelsen Download PDF

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Publication number
NO332383B1
NO332383B1 NO20044256A NO20044256A NO332383B1 NO 332383 B1 NO332383 B1 NO 332383B1 NO 20044256 A NO20044256 A NO 20044256A NO 20044256 A NO20044256 A NO 20044256A NO 332383 B1 NO332383 B1 NO 332383B1
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Prior art keywords
mmol
compound
added
solution
formula
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Application number
NO20044256A
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English (en)
Norwegian (no)
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NO20044256L (no
Inventor
Hiroshi Shirota
Isao Tanaka
Kenichi Chiba
Kenzo Muramoto
Masaki Goto
Naoki Yoneda
Fabian Gusovsky
Yimin Jiang
Xiang-Yi Li
Mark Spyvee
Roch Boivin
Jesse Chow
Hong Du
Yoshihito Eguchi
Masanori Fujita
Jean-Christophe Harmange
Atsushi Inoue
Megumi Kawada
Takatoshi Kawai
Yoshiyuki Kawakami
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Jpkotake Makoto
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Application filed by Jpkotake Makoto filed Critical Jpkotake Makoto
Publication of NO20044256L publication Critical patent/NO20044256L/no
Publication of NO332383B1 publication Critical patent/NO332383B1/no

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    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D313/00Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A61K31/36Compounds containing methylenedioxyphenyl groups, e.g. sesamin
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    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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NO20044256A 2002-03-08 2004-10-07 Makrosykliske forbindelser, anvendelse derav til fremstilling av et medikament, og farmasoytisk preparat som omfatter forbindelsen NO332383B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US36288302P 2002-03-08 2002-03-08
US38071102P 2002-05-14 2002-05-14
PCT/US2003/007377 WO2003076424A1 (fr) 2002-03-08 2003-03-07 Composes macrocycliques utiles comme produits pharmaceutiques

Publications (2)

Publication Number Publication Date
NO20044256L NO20044256L (no) 2004-12-07
NO332383B1 true NO332383B1 (no) 2012-09-10

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Country Status (18)

Country Link
US (3) US7799827B2 (fr)
EP (2) EP1507773B1 (fr)
JP (3) JP4575667B2 (fr)
KR (1) KR101210018B1 (fr)
CN (2) CN104876904A (fr)
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CA2478065A1 (fr) 2003-09-18
TWI343916B (en) 2011-06-21
EP1507773A1 (fr) 2005-02-23
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NO20044256L (no) 2004-12-07
US20060247448A1 (en) 2006-11-02
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RU2334744C2 (ru) 2008-09-27
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PL221491B1 (pl) 2016-04-29
WO2003076424A1 (fr) 2003-09-18
AU2010201776A1 (en) 2010-05-27
JP2012193183A (ja) 2012-10-11
JP2005519954A (ja) 2005-07-07
BRPI0308113B8 (pt) 2021-05-25
PL373044A1 (en) 2005-08-08
CA2478065C (fr) 2013-01-08
CN1653059A (zh) 2005-08-10
NZ535101A (en) 2007-07-27
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RU2004129755A (ru) 2005-04-20
US8329742B2 (en) 2012-12-11
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IL163711A0 (en) 2005-12-18
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US20130196987A1 (en) 2013-08-01
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US7799827B2 (en) 2010-09-21
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