NO316863B1 - Oral farmasoytisk, tablettert multippel enhetsdoseringsfom, fremgangsmate for dens fremstilling, anvendelse derav, og blaerepakning - Google Patents
Oral farmasoytisk, tablettert multippel enhetsdoseringsfom, fremgangsmate for dens fremstilling, anvendelse derav, og blaerepakning Download PDFInfo
- Publication number
- NO316863B1 NO316863B1 NO19960948A NO960948A NO316863B1 NO 316863 B1 NO316863 B1 NO 316863B1 NO 19960948 A NO19960948 A NO 19960948A NO 960948 A NO960948 A NO 960948A NO 316863 B1 NO316863 B1 NO 316863B1
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- NO
- Norway
- Prior art keywords
- dosage form
- coating layer
- enteric coating
- tableted
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- 150000003022 phthalic acids Chemical class 0.000 description 1
- 230000000704 physical effect Effects 0.000 description 1
- 229920000120 polyethyl acrylate Polymers 0.000 description 1
- 229940068917 polyethylene glycols Drugs 0.000 description 1
- 229920005597 polymer membrane Polymers 0.000 description 1
- 229950008882 polysorbate Drugs 0.000 description 1
- 229940068965 polysorbates Drugs 0.000 description 1
- 229940100467 polyvinyl acetate phthalate Drugs 0.000 description 1
- 239000011591 potassium Substances 0.000 description 1
- 229910052700 potassium Inorganic materials 0.000 description 1
- 230000002265 prevention Effects 0.000 description 1
- 239000000612 proton pump inhibitor Substances 0.000 description 1
- 239000008213 purified water Substances 0.000 description 1
- 238000011160 research Methods 0.000 description 1
- 230000000717 retained effect Effects 0.000 description 1
- 239000004208 shellac Substances 0.000 description 1
- 229940113147 shellac Drugs 0.000 description 1
- 235000013874 shellac Nutrition 0.000 description 1
- ZLGIYFNHBLSMPS-ATJNOEHPSA-N shellac Chemical compound OCCCCCC(O)C(O)CCCCCCCC(O)=O.C1C23[C@H](C(O)=O)CCC2[C@](C)(CO)[C@@H]1C(C(O)=O)=C[C@@H]3O ZLGIYFNHBLSMPS-ATJNOEHPSA-N 0.000 description 1
- 239000000377 silicon dioxide Substances 0.000 description 1
- 210000000813 small intestine Anatomy 0.000 description 1
- 239000007921 spray Substances 0.000 description 1
- 238000001694 spray drying Methods 0.000 description 1
- 239000008107 starch Substances 0.000 description 1
- 229940032147 starch Drugs 0.000 description 1
- 229910052717 sulfur Inorganic materials 0.000 description 1
- 125000004434 sulfur atom Chemical group 0.000 description 1
- 238000013268 sustained release Methods 0.000 description 1
- 239000012730 sustained-release form Substances 0.000 description 1
- 230000009747 swallowing Effects 0.000 description 1
- 238000009492 tablet coating Methods 0.000 description 1
- 239000002700 tablet coating Substances 0.000 description 1
- 239000007916 tablet composition Substances 0.000 description 1
- 230000009466 transformation Effects 0.000 description 1
- 230000032258 transport Effects 0.000 description 1
- 229960002622 triacetin Drugs 0.000 description 1
- 239000001069 triethyl citrate Substances 0.000 description 1
- VMYFZRTXGLUXMZ-UHFFFAOYSA-N triethyl citrate Natural products CCOC(=O)C(O)(C(=O)OCC)C(=O)OCC VMYFZRTXGLUXMZ-UHFFFAOYSA-N 0.000 description 1
- 235000013769 triethyl citrate Nutrition 0.000 description 1
- 125000005591 trimellitate group Chemical group 0.000 description 1
- 230000036269 ulceration Effects 0.000 description 1
- 238000005303 weighing Methods 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9402431A SE9402431D0 (sv) | 1994-07-08 | 1994-07-08 | New tablet formulation |
| PCT/SE1995/000678 WO1996001624A1 (en) | 1994-07-08 | 1995-06-07 | Multiple unit pharmaceutical preparation containing proton pump inhibitor |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO960948L NO960948L (no) | 1996-03-07 |
| NO960948D0 NO960948D0 (no) | 1996-03-07 |
| NO316863B1 true NO316863B1 (no) | 2004-06-07 |
Family
ID=20394685
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19960948A NO316863B1 (no) | 1994-07-08 | 1996-03-07 | Oral farmasoytisk, tablettert multippel enhetsdoseringsfom, fremgangsmate for dens fremstilling, anvendelse derav, og blaerepakning |
| NO960949A NO960949D0 (no) | 1994-07-08 | 1996-03-07 | Tablettert flerdoseenhetsform inneholdende protonpumpeinhibitor |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO960949A NO960949D0 (no) | 1994-07-08 | 1996-03-07 | Tablettert flerdoseenhetsform inneholdende protonpumpeinhibitor |
Country Status (36)
| Country | Link |
|---|---|
| US (1) | US5753265A (pl) |
| EP (3) | EP0723437B1 (pl) |
| JP (2) | JPH09502741A (pl) |
| KR (1) | KR100384961B1 (pl) |
| CN (2) | CN1152671C (pl) |
| AT (1) | ATE275396T1 (pl) |
| AU (1) | AU695971B2 (pl) |
| BR (2) | BR9506029A (pl) |
| CA (2) | CA2170644C (pl) |
| CZ (1) | CZ294380B6 (pl) |
| DE (1) | DE69533470T2 (pl) |
| DK (1) | DK0723437T3 (pl) |
| EE (1) | EE03292B1 (pl) |
| ES (1) | ES2227556T3 (pl) |
| FI (2) | FI961059A0 (pl) |
| HK (1) | HK1008298A1 (pl) |
| HU (2) | HUT75934A (pl) |
| IL (2) | IL114449A0 (pl) |
| IS (3) | IS4326A (pl) |
| MA (1) | MA23608A1 (pl) |
| MY (1) | MY114388A (pl) |
| NO (2) | NO316863B1 (pl) |
| NZ (1) | NZ289949A (pl) |
| PL (2) | PL313389A1 (pl) |
| PT (1) | PT723437E (pl) |
| RU (2) | RU2166935C2 (pl) |
| SA (1) | SA95160092B1 (pl) |
| SE (1) | SE9402431D0 (pl) |
| SI (1) | SI0723437T1 (pl) |
| SK (1) | SK283841B6 (pl) |
| TN (1) | TNSN95076A1 (pl) |
| TR (2) | TR199500826A2 (pl) |
| TW (1) | TW421599B (pl) |
| UA (1) | UA47390C2 (pl) |
| WO (2) | WO1996001624A1 (pl) |
| ZA (2) | ZA955546B (pl) |
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| DE29522419U1 (de) * | 1994-07-08 | 2003-07-03 | AstraZeneca AB, Södertälje | Tablettierte Mehrfacheinheits-Dosisform |
| SE9402431D0 (sv) * | 1994-07-08 | 1994-07-08 | Astra Ab | New tablet formulation |
| ES2094694B1 (es) * | 1995-02-01 | 1997-12-16 | Esteve Quimica Sa | Nueva formulacion farmaceuticamente estable de un compuesto de bencimidazol y su proceso de obtencion. |
| SE9500422D0 (sv) * | 1995-02-06 | 1995-02-06 | Astra Ab | New oral pharmaceutical dosage forms |
| SE9500478D0 (sv) * | 1995-02-09 | 1995-02-09 | Astra Ab | New pharmaceutical formulation and process |
| ATE262332T1 (de) * | 1995-09-21 | 2004-04-15 | Pharma Pass Ii Llc | Lansoprazolhaltige arzneizusammensetzung und herstellungsverfahren |
| US6489346B1 (en) | 1996-01-04 | 2002-12-03 | The Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and method of using same |
| US6645988B2 (en) * | 1996-01-04 | 2003-11-11 | Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and method of using same |
| US6699885B2 (en) | 1996-01-04 | 2004-03-02 | The Curators Of The University Of Missouri | Substituted benzimidazole dosage forms and methods of using same |
| US5840737A (en) | 1996-01-04 | 1998-11-24 | The Curators Of The University Of Missouri | Omeprazole solution and method for using same |
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| SE9600071D0 (sv) | 1996-01-08 | 1996-01-08 | Astra Ab | New oral formulation of two active ingredients I |
| SE9600070D0 (sv) * | 1996-01-08 | 1996-01-08 | Astra Ab | New oral pharmaceutical dosage forms |
| SE9600072D0 (sv) * | 1996-01-08 | 1996-01-08 | Astra Ab | New oral formulation of two active ingredients II |
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| HUP0100179A3 (en) | 1997-07-03 | 2002-12-28 | Bristol Myers Squibb Pharma Co | Imidazopyrimidine and imidazopyridine derivatives and pharmaceutical compositions thereof |
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1994
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- 1995-06-07 RU RU96107040/14A patent/RU2166935C2/ru not_active IP Right Cessation
- 1995-06-07 EP EP95926055A patent/EP0723437B1/en not_active Revoked
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- 1995-06-07 EP EP04011147A patent/EP1452172A3/en not_active Withdrawn
- 1995-06-07 AU AU29938/95A patent/AU695971B2/en not_active Expired
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- 1995-06-07 PT PT95926055T patent/PT723437E/pt unknown
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- 1995-06-07 CN CN95190816A patent/CN1134667A/zh active Pending
- 1995-06-07 BR BR9506028A patent/BR9506028A/pt active Search and Examination
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- 1995-06-07 JP JP8504250A patent/JPH09502741A/ja active Pending
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- 1995-07-07 EP EP95926056A patent/EP0724434A1/en not_active Withdrawn
- 1995-07-07 TN TNTNSN95076A patent/TNSN95076A1/fr unknown
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1996
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| MK1K | Patent expired |