NO302699B1 - Fremstilling av taxanderivater samt mellomprodukter til bruk ved fremstillingen - Google Patents

Fremstilling av taxanderivater samt mellomprodukter til bruk ved fremstillingen

Info

Publication number
NO302699B1
NO302699B1 NO931805A NO931805A NO302699B1 NO 302699 B1 NO302699 B1 NO 302699B1 NO 931805 A NO931805 A NO 931805A NO 931805 A NO931805 A NO 931805A NO 302699 B1 NO302699 B1 NO 302699B1
Authority
NO
Norway
Prior art keywords
aryl
protecting
taxane
intermediates
manufacture
Prior art date
Application number
NO931805A
Other languages
English (en)
Norwegian (no)
Other versions
NO931805L (no
NO931805D0 (no
Inventor
Jean-Dominique Bourzat
Alain Commercon
Jean-Marc Paris
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR909014635A external-priority patent/FR2669631B1/fr
Priority claimed from FR9109423A external-priority patent/FR2679557B1/fr
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of NO931805L publication Critical patent/NO931805L/no
Publication of NO931805D0 publication Critical patent/NO931805D0/no
Publication of NO302699B1 publication Critical patent/NO302699B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO931805A 1990-11-23 1993-05-18 Fremstilling av taxanderivater samt mellomprodukter til bruk ved fremstillingen NO302699B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR909014635A FR2669631B1 (fr) 1990-11-23 1990-11-23 Nouveaux derives de l'oxazolidine, leur preparation et leur emploi.
FR9109423A FR2679557B1 (fr) 1991-07-25 1991-07-25 Procede de preparation de derives du taxane, nouveaux derives obtenus et compositions pharmaceutiques qui les contiennent.
PCT/FR1991/000928 WO1992009589A1 (fr) 1990-11-23 1991-11-22 Procede de preparation de derives du taxane, nouveaux derives obtenus et compositions pharmaceutiques qui les contiennent

Publications (3)

Publication Number Publication Date
NO931805L NO931805L (no) 1993-05-18
NO931805D0 NO931805D0 (no) 1993-05-18
NO302699B1 true NO302699B1 (no) 1998-04-14

Family

ID=26228347

Family Applications (1)

Application Number Title Priority Date Filing Date
NO931805A NO302699B1 (no) 1990-11-23 1993-05-18 Fremstilling av taxanderivater samt mellomprodukter til bruk ved fremstillingen

Country Status (24)

Country Link
US (1) US5476954A (cs)
EP (2) EP0595370B1 (cs)
JP (1) JP3043411B2 (cs)
KR (1) KR100206457B1 (cs)
AT (2) ATE163415T1 (cs)
AU (1) AU655618B2 (cs)
CA (1) CA2096833C (cs)
CZ (1) CZ286749B6 (cs)
DE (2) DE69104223T2 (cs)
DK (2) DK0595370T3 (cs)
ES (2) ES2112377T3 (cs)
FI (2) FI105184B (cs)
GR (1) GR3026238T3 (cs)
HU (1) HU214332B (cs)
IE (2) IE80681B1 (cs)
MX (1) MX9102128A (cs)
NO (1) NO302699B1 (cs)
NZ (2) NZ247867A (cs)
PL (1) PL166893B1 (cs)
PT (2) PT99580B (cs)
RU (1) RU2095356C1 (cs)
SK (1) SK282162B6 (cs)
WO (1) WO1992009589A1 (cs)
YU (1) YU48150B (cs)

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* Cited by examiner, † Cited by third party
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