NO2015014I2 - Paritaprevir - Google Patents

Paritaprevir

Info

Publication number
NO2015014I2
NO2015014I2 NO2015014C NO2015014C NO2015014I2 NO 2015014 I2 NO2015014 I2 NO 2015014I2 NO 2015014 C NO2015014 C NO 2015014C NO 2015014 C NO2015014 C NO 2015014C NO 2015014 I2 NO2015014 I2 NO 2015014I2
Authority
NO
Norway
Prior art keywords
paritaprevir
Prior art date
Application number
NO2015014C
Other languages
English (en)
Other versions
NO2015014I1 (no
Original Assignee
Abbvie Bahamas Ltd
Enanta Pharm Inc
Filing date
Publication date
Family has litigation
Priority to US19172508P priority Critical
Priority to US20968909P priority
Priority to PCT/US2009/005082 priority patent/WO2010030359A2/en
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42005677&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO2015014(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Publication of NO2015014I2 publication Critical patent/NO2015014I2/no
Application filed by Abbvie Bahamas Ltd, Enanta Pharm Inc filed Critical Abbvie Bahamas Ltd
Publication of NO2015014I1 publication Critical patent/NO2015014I1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C07K1/113—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides without change of the primary structure
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
NO2015014C 2008-09-11 2015-04-22 Paritaprevir, eller et farmasøytisk akseptabelt salt eller ester derav NO2015014I1 (no)

Priority Applications (3)

Application Number Priority Date Filing Date Title
US19172508P true 2008-09-11 2008-09-11
US20968909P true 2009-03-10 2009-03-10
PCT/US2009/005082 WO2010030359A2 (en) 2008-09-11 2009-09-10 Macrocyclic hepatitis c serine protease inhibitors

Publications (2)

Publication Number Publication Date
NO2015014I2 true NO2015014I2 (no) 2015-04-22
NO2015014I1 NO2015014I1 (no) 2015-05-04

Family

ID=42005677

Family Applications (1)

Application Number Title Priority Date Filing Date
NO2015014C NO2015014I1 (no) 2008-09-11 2015-04-22 Paritaprevir, eller et farmasøytisk akseptabelt salt eller ester derav

Country Status (41)

Country Link
US (3) US8420596B2 (no)
EP (5) EP2468285B1 (no)
JP (4) JP5259537B2 (no)
KR (3) KR101379365B1 (no)
CN (3) CN101775017B (no)
AR (3) AR073568A1 (no)
AU (1) AU2009292182B2 (no)
BR (2) BRPI0918724B1 (no)
CA (1) CA2736895C (no)
CL (2) CL2011000512A1 (no)
CO (1) CO6341565A2 (no)
CR (1) CR20140180A (no)
CY (5) CY1115137T1 (no)
DK (5) DK2468286T3 (no)
DO (1) DOP2011000077A (no)
EA (2) EA022891B1 (no)
EC (2) ECSP11010879A (no)
ES (5) ES2677644T3 (no)
GT (2) GT201100056AA (no)
HK (4) HK1170937A1 (no)
HR (5) HRP20140492T1 (no)
HU (2) HUE039478T2 (no)
IL (2) IL218441A (no)
LT (2) LT2805726T (no)
LU (1) LU92667I2 (no)
MX (1) MX2011002486A (no)
MY (1) MY159820A (no)
NL (1) NL300730I1 (no)
NO (1) NO2015014I1 (no)
NZ (2) NZ605550A (no)
PA (1) PA8842201A1 (no)
PE (3) PE20140961A1 (no)
PL (5) PL2468286T3 (no)
PT (5) PT2805726T (no)
SG (1) SG179414A1 (no)
SI (5) SI2468287T1 (no)
TR (1) TR201809771T4 (no)
TW (3) TWI450723B (no)
UY (3) UY32099A (no)
WO (1) WO2010030359A2 (no)
ZA (2) ZA201101558B (no)

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PL2468287T3 (pl) 2014-09-30
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ES2525922T3 (es) 2015-01-02
NL300730I2 (no) 2016-01-07
GT201100056AA (es) 2014-09-26
UY35259A (es) 2015-08-31
PE20110704A1 (es) 2011-11-12
HK1171184A1 (zh) 2013-03-22
AR086181A2 (es) 2013-11-27
CY1115379T1 (el) 2017-01-04
WO2010030359A2 (en) 2010-03-18
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JP2012136546A (ja) 2012-07-19
PT2805726T (pt) 2018-07-23
NZ592170A (en) 2013-02-22
SG179414A1 (en) 2012-04-27
HRP20140493T1 (xx) 2014-07-18
EP2340029B1 (en) 2014-03-05
JP5902123B2 (ja) 2016-04-13
HK1170936A1 (zh) 2013-03-15
PT2468287E (pt) 2014-07-15
JP5259537B2 (ja) 2013-08-07
US8642538B2 (en) 2014-02-04
NL300730I1 (no) 2016-01-07
EP2468285B1 (en) 2014-10-15
KR20120044316A (ko) 2012-05-07
EP2468286B1 (en) 2014-04-23
SI2340029T1 (sl) 2014-08-29
JP5534533B2 (ja) 2014-07-02
DK2468286T3 (da) 2014-07-28
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CY1115137T1 (xx) 2016-04-13
PL2468286T3 (pl) 2014-09-30
EP2805726B1 (en) 2018-05-02
BR122012005261A2 (pt) 2015-07-14
PL2340029T3 (pl) 2014-12-31
UY32099A (es) 2010-04-30
AR073568A1 (es) 2010-11-17
SI2468285T1 (sl) 2015-01-30
PT2468286E (pt) 2014-07-15
ES2677644T3 (es) 2018-08-06
HRP20141169T1 (en) 2015-02-13
TW201417826A (zh) 2014-05-16
SI2468286T1 (sl) 2014-08-29
DK2340029T3 (da) 2014-06-10
KR20100031092A (ko) 2010-03-19
TWI450723B (zh) 2014-09-01
MY159820A (en) 2017-02-15
NO2015014I1 (no) 2015-05-04
EP2340029A4 (en) 2012-06-13
CA2736895A1 (en) 2010-03-18
DOP2011000077A (es) 2011-04-30
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EA020580B1 (ru) 2014-12-30
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TW201023875A (en) 2010-07-01
AU2009292182A1 (en) 2010-03-18
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IL234969D0 (en) 2014-11-30
SI2468287T1 (sl) 2014-08-29
EP2468286A1 (en) 2012-06-27
PT2468285E (pt) 2015-02-04
SI2805726T1 (sl) 2018-09-28
CR20140180A (es) 2014-06-03
DK2468285T3 (en) 2015-01-19
CN101775017A (zh) 2010-07-14
US8420596B2 (en) 2013-04-16
HRP20140492T1 (en) 2014-09-12
ES2459390T3 (es) 2014-05-09
CL2011000512A1 (es) 2011-06-17
GT201100056BA (es) 2015-04-22
NZ605550A (en) 2014-06-27
BRPI0918724B1 (pt) 2019-12-03
PA8842201A1 (es) 2010-04-21
PT2340029E (pt) 2014-05-13
EP2468285A1 (en) 2012-06-27
JP5801342B2 (ja) 2015-10-28
EA022891B1 (ru) 2016-03-31
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ES2475163T3 (es) 2014-07-10
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DK2468287T3 (da) 2014-07-28
LT2805726T (lt) 2018-08-10
EA201170434A1 (ru) 2011-10-31
ES2475815T3 (es) 2014-07-11
CY1115844T1 (el) 2017-01-25
HK1159515A1 (zh) 2012-08-03
CN102641271B (zh) 2013-12-25
PE20140961A1 (es) 2014-08-24
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PL2468285T3 (pl) 2015-03-31
KR101487726B1 (ko) 2015-01-29
CO6341565A2 (es) 2011-11-21
ECSP12011947A (es) 2012-07-31
PL2805726T3 (pl) 2018-11-30
KR101379365B1 (ko) 2014-03-31
CN103896950A (zh) 2014-07-02
BRPI0918724A2 (pt) 2013-06-18
TWI429449B (zh) 2014-03-11
CL2012001495A1 (es) 2013-07-12
IL218441D0 (en) 2012-04-30
CA2736895C (en) 2016-02-09
CN101775017B (zh) 2014-04-30
MX2011002486A (es) 2011-04-26
US20120196792A1 (en) 2012-08-02
HK1170937A1 (zh) 2013-03-15
DK2805726T3 (en) 2018-07-30
EA201200390A1 (ru) 2012-12-28
US9309279B2 (en) 2016-04-12
UY33981A (es) 2013-10-31
JP2013227314A (ja) 2013-11-07
EP2805726A1 (en) 2014-11-26
JP2010065035A (ja) 2010-03-25
US20140148573A1 (en) 2014-05-29
PE20121312A1 (es) 2012-10-28
IL218441A (en) 2015-09-24
HUE039478T2 (hu) 2019-01-28
TW201231064A (en) 2012-08-01
HRP20140494T1 (xx) 2014-07-04
TR201809771T4 (tr) 2018-07-23
JP2013163680A (ja) 2013-08-22

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