NL193376C - 16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan. - Google Patents

16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan. Download PDF

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Publication number
NL193376C
NL193376C NL8701322A NL8701322A NL193376C NL 193376 C NL193376 C NL 193376C NL 8701322 A NL8701322 A NL 8701322A NL 8701322 A NL8701322 A NL 8701322A NL 193376 C NL193376 C NL 193376C
Authority
NL
Netherlands
Prior art keywords
group
formula
compounds
compound
carbon atoms
Prior art date
Application number
NL8701322A
Other languages
English (en)
Dutch (nl)
Other versions
NL8701322A (nl
NL193376B (nl
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB868613790A external-priority patent/GB8613790D0/en
Priority claimed from GB868625854A external-priority patent/GB8625854D0/en
Priority claimed from GB878708423A external-priority patent/GB8708423D0/en
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of NL8701322A publication Critical patent/NL8701322A/nl
Publication of NL193376B publication Critical patent/NL193376B/xx
Application granted granted Critical
Publication of NL193376C publication Critical patent/NL193376C/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N49/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds containing the group, wherein m+n>=1, both X together may also mean —Y— or a direct carbon-to-carbon bond, and the carbon atoms marked with an asterisk are not part of any ring system other than that which may be formed by the atoms X, the carbon atoms in square brackets being part of any acyclic or cyclic structure, or the group, wherein A means a carbon atom or Y, n>=0, and not more than one of these carbon atoms being a member of the same ring system, e.g. juvenile insect hormones or mimics thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biotechnology (AREA)
  • Insects & Arthropods (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NL8701322A 1986-06-06 1987-06-05 16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan. NL193376C (nl)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
GB868613790A GB8613790D0 (en) 1986-06-06 1986-06-06 Chemical compounds
GB8613790 1986-06-06
GB8625854 1986-10-29
GB868625854A GB8625854D0 (en) 1986-10-29 1986-10-29 Chemical process
GB878708423A GB8708423D0 (en) 1987-04-08 1987-04-08 Chemical compounds
GB8708423 1987-04-08

Publications (3)

Publication Number Publication Date
NL8701322A NL8701322A (nl) 1988-01-04
NL193376B NL193376B (nl) 1999-04-01
NL193376C true NL193376C (nl) 1999-08-03

Family

ID=27263057

Family Applications (2)

Application Number Title Priority Date Filing Date
NL8701322A NL193376C (nl) 1986-06-06 1987-06-05 16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan.
NL990026C NL990026I2 (nl) 1986-06-06 1999-08-18 16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan.

Family Applications After (1)

Application Number Title Priority Date Filing Date
NL990026C NL990026I2 (nl) 1986-06-06 1999-08-18 16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan.

Country Status (35)

Country Link
US (1) US4900753A (fi)
JP (1) JP2648147B2 (fi)
KR (1) KR950010077B1 (fi)
CN (1) CN1023858C (fi)
AR (1) AR244691A1 (fi)
AT (1) AT398571B (fi)
AU (1) AU609399B2 (fi)
BE (1) BE1000201A4 (fi)
BR (1) BR8702866A (fi)
CA (1) CA1296329C (fi)
CH (1) CH677670A5 (fi)
DE (3) DE19875029I2 (fi)
DK (1) DK166498B1 (fi)
EG (1) EG18752A (fi)
ES (1) ES2006479A6 (fi)
FI (2) FI90663C (fi)
FR (1) FR2599742B1 (fi)
GB (1) GB2192630B (fi)
GE (1) GEP19981388B (fi)
GR (1) GR870891B (fi)
HU (1) HU199847B (fi)
IE (1) IE60411B1 (fi)
IL (1) IL82776A (fi)
IT (1) IT1206015B (fi)
LU (2) LU86908A1 (fi)
LV (2) LV10280A (fi)
NL (2) NL193376C (fi)
NZ (1) NZ220587A (fi)
OA (1) OA08606A (fi)
PH (1) PH23948A (fi)
PL (3) PL153036B1 (fi)
PT (1) PT85018B (fi)
SE (1) SE503399C2 (fi)
TR (1) TR28970A (fi)
UA (1) UA45300C2 (fi)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0260537A1 (en) * 1986-09-12 1988-03-23 American Cyanamid Company 13-Deoxy-23-oxo(keto) and 23-imino derivatives of 13-deoxy C-076-aglycone compounds
ES2058082T3 (es) * 1986-09-12 1994-11-01 American Cyanamid Co Derivados 23-oxo (ceto) y 23-imino de compuestos ll-f28249.
US4886828A (en) * 1986-09-12 1989-12-12 American Cyanamid Company Δ22 -derivatives of LL-F28249 compounds
GB8721377D0 (en) * 1987-09-11 1987-10-21 Glaxo Group Ltd Chemical compounds
GB8811036D0 (en) * 1988-05-10 1988-06-15 Glaxo Group Ltd Chemical compounds
GB8813150D0 (en) * 1988-06-03 1988-07-06 American Cyanamid Co Chemical compounds
GB8905605D0 (en) * 1989-03-11 1989-04-26 Beecham Group Plc Novel compounds
NZ233680A (en) * 1989-05-17 1995-02-24 Beecham Group Plc Avermectins and milbemycins and compositions thereof
US4988824A (en) * 1989-09-11 1991-01-29 Maulding Donald R Process for the preparation of 23-(C1-C6 alkyloxime)-LL-F28249 compounds
CA2097918C (en) * 1990-12-07 2002-07-16 Frank N. Chang Stabilized insect nematode compositions
JP2855181B2 (ja) 1993-12-10 1999-02-10 敏雄 鈴木 松類の枯損防止用組成物及び防止方法
DK1197215T3 (da) 2000-10-10 2006-07-10 Wyeth Corp Anthelmintiske sammensætninger
US7348417B2 (en) * 2003-08-07 2008-03-25 Wyeth Method of purifying moxidectin through crystallization
WO2006119174A1 (en) 2005-04-30 2006-11-09 Ocular Surface Center, P.A. Method for treating ocular demodex
JP4939025B2 (ja) * 2005-09-30 2012-05-23 三菱電線工業株式会社 電熱ヒータ付きハンドル用グリップ部材
EP1849363A1 (en) * 2006-03-09 2007-10-31 Cheminova A/S Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin
US8128968B2 (en) * 2007-08-29 2012-03-06 Tissuetech, Inc. Compositions and methods for treating Demodex infestations
DK3351546T5 (da) 2011-12-02 2024-08-12 Boehringer Ingelheim Vetmedica Gmbh Langtidsvirkende injicerbare moxidectinformuleringer
FR2995605B1 (fr) * 2012-09-18 2014-09-19 Sanofi Sa Derives de macrolides, leur preparation et leur application therapeutique.

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH15982A (en) * 1977-10-03 1983-05-18 Merck & Co Inc Selective hydrogenation producta of c-076 compounds and derivatives thereof
US4289760A (en) * 1980-05-02 1981-09-15 Merck & Co., Inc. 23-Keto derivatives of C-076 compounds
US4423209A (en) * 1982-02-26 1983-12-27 Merck & Co., Inc. Processes for the interconversion of avermectin compounds
JPS59108785A (ja) * 1982-11-25 1984-06-23 Sankyo Co Ltd ミルベマイシン類の５−オキシム誘導体
JPS60126289A (ja) * 1983-11-14 1985-07-05 Sankyo Co Ltd ミルベマイシン類の５−カ−ボネ−ト誘導体
EP0170006B1 (en) * 1984-06-05 1992-07-08 American Cyanamid Company Method and compositions for helmintic, arthropod ectoparasitic and acaridal infections with novel agents
US4579864A (en) * 1984-06-11 1986-04-01 Merck & Co., Inc. Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives
IT1182857B (it) * 1984-09-14 1987-10-05 Glaxo Group Ltd Composti antibiotici, composizioni antiparassitarie che li contengono e procedimento per prepararli ed applicarli
ES8802229A1 (es) * 1985-04-30 1988-04-16 Glaxo Group Ltd Un procedimiento para preparar nuevos derivados lactonicos macrociclicos.
ES2058082T3 (es) * 1986-09-12 1994-11-01 American Cyanamid Co Derivados 23-oxo (ceto) y 23-imino de compuestos ll-f28249.

Also Published As

Publication number Publication date
CA1296329C (en) 1992-02-25
FI923445A0 (fi) 1992-07-30
EG18752A (en) 1993-12-30
GB8713239D0 (en) 1987-07-08
NL8701322A (nl) 1988-01-04
LU86908A1 (fr) 1988-01-20
LV10781B (en) 1996-10-20
GEP19981388B (en) 1998-11-10
IL82776A (en) 1992-02-16
KR880000441A (ko) 1988-03-25
NL990026I1 (nl) 1999-11-01
GB2192630A (en) 1988-01-20
JP2648147B2 (ja) 1997-08-27
SE8702361L (sv) 1987-12-07
DK290287A (da) 1987-12-07
FI923445A (fi) 1992-07-30
SE503399C2 (sv) 1996-06-10
IT1206015B (it) 1989-04-05
FI872517A0 (fi) 1987-06-04
SE8702361D0 (sv) 1987-06-05
NZ220587A (en) 1990-05-28
FR2599742B1 (fr) 1989-05-19
PH23948A (en) 1990-01-23
IL82776A0 (en) 1987-12-20
IE871496L (en) 1987-12-06
AU7387387A (en) 1987-12-10
GR870891B (en) 1987-10-02
AR244691A1 (es) 1993-11-30
PL266100A1 (en) 1988-07-21
FI90663C (fi) 1994-03-10
OA08606A (en) 1988-11-30
KR950010077B1 (ko) 1995-09-06
LV10280A (lv) 1994-10-20
DK290287D0 (da) 1987-06-04
BR8702866A (pt) 1988-03-01
FI90549C (fi) 1994-02-25
PT85018A (en) 1987-07-01
CN87104431A (zh) 1987-12-30
UA45300C2 (uk) 2002-04-15
LV10781A (lv) 1995-08-20
AT398571B (de) 1994-12-27
DK166498B1 (da) 1993-06-01
GB2192630B (en) 1990-05-23
ES2006479A6 (es) 1989-05-01
NL193376B (nl) 1999-04-01
DE3745133C2 (de) 1998-01-02
AU609399B2 (en) 1991-05-02
DE3718926A1 (de) 1987-12-10
CH677670A5 (fi) 1991-06-14
FI872517A (fi) 1987-12-07
LU88790I2 (fr) 1997-03-18
FI90549B (fi) 1993-11-15
HU199847B (en) 1990-03-28
ATA143887A (de) 1994-05-15
DE19875029I2 (de) 2001-11-22
DE3718926C2 (de) 1998-01-15
NL990026I2 (nl) 1999-12-01
TR28970A (tr) 1997-07-21
CN1023858C (zh) 1994-02-23
FI90663B (fi) 1993-11-30
HUT44254A (en) 1988-02-29
FR2599742A1 (fr) 1987-12-11
PL155723B1 (en) 1991-12-31
IT8748023A0 (it) 1987-06-05
PL153226B1 (en) 1991-03-29
PT85018B (pt) 1990-03-08
US4900753A (en) 1990-02-13
BE1000201A4 (fr) 1988-08-23
JPS6354375A (ja) 1988-03-08
PL153036B1 (en) 1991-02-28
IE60411B1 (en) 1994-07-13

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Legal Events

Date Code Title Description
CNR Transfer of rights (patent application after its laying open for public inspection)

Free format text: AMERICAN CYANAMID COMPANY TE WAYNE

BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
KC1 Grant of a supplementary protection certificate

Free format text: 990026, 20070605, EXPIRES: 20091229

TNT Modifications of names of proprietors of patents or applicants of examined patent applications

Owner name: WYETH HOLDINGS CORPORATION

V4 Discontinued because of reaching the maximum lifetime of a patent

Effective date: 20070605