NL182401C - Farmaceutisch preparaat met antimicrobiele activiteit, alsmede syn-isomeer van een 7-(2-(2-aminothiazool-4-yl)-2-(alkoxyimino)-aceetamido)-3-cefem-4-carbonzuur derivaat. - Google Patents

Farmaceutisch preparaat met antimicrobiele activiteit, alsmede syn-isomeer van een 7-(2-(2-aminothiazool-4-yl)-2-(alkoxyimino)-aceetamido)-3-cefem-4-carbonzuur derivaat.

Info

Publication number
NL182401C
NL182401C NLAANVRAGE7802792,A NL7802792A NL182401C NL 182401 C NL182401 C NL 182401C NL 7802792 A NL7802792 A NL 7802792A NL 182401 C NL182401 C NL 182401C
Authority
NL
Netherlands
Prior art keywords
aminothiazol
alkoxyimino
cephem
acetamido
acid derivative
Prior art date
Application number
NLAANVRAGE7802792,A
Other languages
English (en)
Other versions
NL182401B (nl
NL7802792A (nl
Original Assignee
Fujisawa Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB10699/77A external-priority patent/GB1600735A/en
Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co
Priority claimed from KR7802782A external-priority patent/KR820001285B1/ko
Publication of NL7802792A publication Critical patent/NL7802792A/nl
Priority claimed from KR1019820000231A external-priority patent/KR830000455B1/ko
Publication of NL182401B publication Critical patent/NL182401B/nl
Application granted granted Critical
Publication of NL182401C publication Critical patent/NL182401C/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/06—1,2,3-Thiadiazoles; Hydrogenated 1,2,3-thiadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NLAANVRAGE7802792,A 1977-03-14 1978-03-14 Farmaceutisch preparaat met antimicrobiele activiteit, alsmede syn-isomeer van een 7-(2-(2-aminothiazool-4-yl)-2-(alkoxyimino)-aceetamido)-3-cefem-4-carbonzuur derivaat. NL182401C (nl)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
GB10699/77A GB1600735A (en) 1977-03-14 1977-03-14 Cephem and cephem compounds and processes for preparation thereof
GB2924577 1977-07-12
GB4231577 1977-10-11
GB7578 1978-01-03
KR7802782A KR820001285B1 (ko) 1977-03-14 1978-09-13 세펨화합물의 제조방법
KR1019820000231A KR830000455B1 (ko) 1977-03-14 1982-01-18 세펨화합물의 제조방법

Publications (3)

Publication Number Publication Date
NL7802792A NL7802792A (nl) 1978-09-18
NL182401B NL182401B (nl) 1987-10-01
NL182401C true NL182401C (nl) 1988-03-01

Family

ID=27546433

Family Applications (2)

Application Number Title Priority Date Filing Date
NLAANVRAGE7802792,A NL182401C (nl) 1977-03-14 1978-03-14 Farmaceutisch preparaat met antimicrobiele activiteit, alsmede syn-isomeer van een 7-(2-(2-aminothiazool-4-yl)-2-(alkoxyimino)-aceetamido)-3-cefem-4-carbonzuur derivaat.
NL8501475A NL8501475A (nl) 1977-03-14 1985-05-23 Cefem- en cefam-verbindingen met antimicrobiele werking, werkwijzen ter bereiding daarvan, alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten.

Family Applications After (1)

Application Number Title Priority Date Filing Date
NL8501475A NL8501475A (nl) 1977-03-14 1985-05-23 Cefem- en cefam-verbindingen met antimicrobiele werking, werkwijzen ter bereiding daarvan, alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten.

Country Status (21)

Country Link
US (7) US4425341A (nl)
JP (7) JPS53137988A (nl)
AR (2) AR230452A1 (nl)
AT (1) AT364456B (nl)
BE (1) BE864810A (nl)
CA (1) CA1321580C (nl)
CH (1) CH637138A5 (nl)
CS (1) CS217961B2 (nl)
DD (2) DD144772A5 (nl)
DE (1) DE2810922C2 (nl)
DK (1) DK163832C (nl)
ES (8) ES467828A1 (nl)
FI (1) FI65779C (nl)
FR (1) FR2383951A1 (nl)
GR (1) GR63619B (nl)
NL (2) NL182401C (nl)
NZ (2) NZ186679A (nl)
PH (2) PH17188A (nl)
PT (1) PT67773A (nl)
SE (3) SE438677B (nl)
YU (3) YU41586B (nl)

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FR2399418A1 (fr) * 1977-03-14 1979-03-02 Fujisawa Pharmaceutical Co Procede de preparation d'acides iminoacetiques et nouveaux produits ainsi obtenus, utilises pour la synthese d'acides cepham- ou cephem-carboxyliques
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JPS53103493A (en) 1977-02-18 1978-09-08 Takeda Chem Ind Ltd Cephalosporin derivatives and process for their preparation
FR2384779A1 (fr) * 1977-03-25 1978-10-20 Roussel Uclaf Nouvelles oximes derivees de l'acide 3-chloro ou 3-methoxy 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
SE439312B (sv) 1977-03-25 1985-06-10 Roussel Uclaf Sett att framstella nya oximderivat av 3-acetoximetyl-7-aminotiazolylacetamido cefalosporansyra
DE2714880A1 (de) * 1977-04-02 1978-10-26 Hoechst Ag Cephemderivate und verfahren zu ihrer herstellung
DE2716677C2 (de) 1977-04-15 1985-10-10 Hoechst Ag, 6230 Frankfurt Cephemderivate und Verfahren zu ihrer Herstellung
FR2410655A1 (fr) 1977-12-05 1979-06-29 Roussel Uclaf Nouvelles oximes derivees de l'acide 3-substitue 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
US4284631A (en) 1978-07-31 1981-08-18 Fujisawa Pharmaceutical Co., Ltd. 7-Substituted cephem compounds and pharmaceutical antibacterial compositions containing them
US4379922A (en) * 1978-09-12 1983-04-12 Fujisawa Pharmaceutical Co., Ltd. Cepham compounds
JPS5543011A (en) * 1978-09-20 1980-03-26 Shionogi & Co Ltd 7-halothiazolylalkoxyiminoacetamido-3-cephem compound
FR2448543A1 (fr) 1979-02-09 1980-09-05 Roussel Uclaf Nouvelles oximes o-substituees par un radical comportant un ammonium quaternaire et derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR2461713A1 (fr) * 1979-07-19 1981-02-06 Roussel Uclaf Nouvelles alcoyloximes substituees derivees de l'acide 7-(2-amino 4-thiazolyl) acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
JPS56125392A (en) * 1980-03-06 1981-10-01 Fujisawa Pharmaceut Co Ltd Cepham and cephem compound and preparation thereof
JPS6238569A (ja) * 1985-08-13 1987-02-19 Nec Corp 磁気デイスク制御装置
US5059611A (en) * 1988-11-18 1991-10-22 Allergan, Inc. Anti-inflammatory 5-hydroxy-2-furanones

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ES8203865A1 (es) 1982-04-01
JPH03115256A (ja) 1991-05-16
US4294960A (en) 1981-10-13
US4460583A (en) 1984-07-17
SE7802933L (sv) 1978-09-15
US4425341A (en) 1984-01-10
SE456909B (sv) 1988-11-14
DD144772A5 (de) 1980-11-05
PH17064A (en) 1984-05-24
YU42061B (en) 1988-04-30
JPS53137988A (en) 1978-12-01
YU274582A (en) 1983-06-30
SE438677B (sv) 1985-04-29
JPH03115288A (ja) 1991-05-16
DE2810922A1 (de) 1978-09-21
NL182401B (nl) 1987-10-01
US4447430A (en) 1984-05-08
ES8101077A1 (es) 1980-12-01
DD136839A5 (de) 1979-08-01
FR2383951B1 (nl) 1983-02-11
FR2383951A1 (fr) 1978-10-13
ES491184A0 (es) 1981-03-16
SE8304670D0 (sv) 1983-08-29
PH17188A (en) 1984-06-14
YU41586B (en) 1987-10-31
CA1321580C (en) 1993-08-24
JPS6434974A (en) 1989-02-06
US4822888A (en) 1989-04-18
SE8304670L (sv) 1983-08-29
CH637138A5 (de) 1983-07-15
ES8103752A1 (es) 1981-03-16
GR63619B (en) 1979-11-27
NL7802792A (nl) 1978-09-18
JPH052666B2 (nl) 1993-01-13
ES491183A0 (es) 1981-03-16
ATA181378A (de) 1981-03-15
JPH0639464B2 (ja) 1994-05-25
NL8501475A (nl) 1985-09-02
DE2810922C2 (de) 1985-08-29
ES480598A1 (es) 1980-07-01
FI780801A (fi) 1978-09-15
ES8103751A1 (es) 1981-03-16
JPH0517230B2 (nl) 1993-03-08
JPH03135972A (ja) 1991-06-10
SE8304671D0 (sv) 1983-08-29
PT67773A (en) 1978-04-01
ES487736A0 (es) 1980-11-01
ES497084A0 (es) 1982-04-01
NZ186679A (en) 1982-12-21
BE864810A (fr) 1978-09-13
DK163832B (da) 1992-04-06
FI65779B (fi) 1984-03-30
JPH03135973A (ja) 1991-06-10
NZ199860A (en) 1984-07-31
DK163832C (da) 1992-09-21
ES8100665A1 (es) 1980-11-01
ES487737A0 (es) 1980-12-01
AT364456B (de) 1981-10-27
AR230452A1 (es) 1984-04-30
YU274682A (en) 1983-10-31
JPS6134435B2 (nl) 1986-08-07
ES467828A1 (es) 1979-09-01
US4604456A (en) 1986-08-05
FI65779C (fi) 1984-07-10
YU60878A (en) 1983-04-30
ES491182A0 (es) 1981-03-16
DK114878A (da) 1978-09-15
US4563522A (en) 1986-01-07
JPH03135971A (ja) 1991-06-10
JPH0720947B2 (ja) 1995-03-08
ES8103753A1 (es) 1981-03-16
CS217961B2 (en) 1983-02-25
AR226423A1 (es) 1982-07-15

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