NL7709092A - Werkwijze ter bereiding van cefalosporinever- bindingen met antibacteriele activiteit als- mede farmaceutische preparaten die deze ver- bindingen als actieve component bevatten. - Google Patents

Werkwijze ter bereiding van cefalosporinever- bindingen met antibacteriele activiteit als- mede farmaceutische preparaten die deze ver- bindingen als actieve component bevatten.

Info

Publication number
NL7709092A
NL7709092A NL7709092A NL7709092A NL7709092A NL 7709092 A NL7709092 A NL 7709092A NL 7709092 A NL7709092 A NL 7709092A NL 7709092 A NL7709092 A NL 7709092A NL 7709092 A NL7709092 A NL 7709092A
Authority
NL
Netherlands
Prior art keywords
preparation
components
active component
pharmaceutical preparations
antibacterial activity
Prior art date
Application number
NL7709092A
Other languages
English (en)
Original Assignee
Fujisawa Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB3430276A external-priority patent/GB1556438A/en
Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co
Publication of NL7709092A publication Critical patent/NL7709092A/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/69—Two or more oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/60—Three or more oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/18—Oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30—Oxygen atoms, e.g. delta-lactones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/34—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D309/36—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C07D309/40—Oxygen atoms attached in positions 3 and 4, e.g. maltol

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NL7709092A 1976-08-17 1977-08-17 Werkwijze ter bereiding van cefalosporinever- bindingen met antibacteriele activiteit als- mede farmaceutische preparaten die deze ver- bindingen als actieve component bevatten. NL7709092A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB3430276A GB1556438A (en) 1976-08-17 1976-08-17 Cephalosporin derivatives and the preparation thereof
GB4974876 1976-11-29

Publications (1)

Publication Number Publication Date
NL7709092A true NL7709092A (nl) 1978-02-21

Family

ID=26262231

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7709092A NL7709092A (nl) 1976-08-17 1977-08-17 Werkwijze ter bereiding van cefalosporinever- bindingen met antibacteriele activiteit als- mede farmaceutische preparaten die deze ver- bindingen als actieve component bevatten.

Country Status (7)

Country Link
US (2) US4172198A (nl)
JP (1) JPS5323993A (nl)
CH (1) CH634848A5 (nl)
DE (1) DE2737066A1 (nl)
ES (2) ES461688A1 (nl)
FR (1) FR2362146A1 (nl)
NL (1) NL7709092A (nl)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4343938A (en) * 1978-03-24 1982-08-10 American Cyanamid Company 7-[Dα-(Coumarin-3-carboxamido)arylacetamido]-cephalosporanic acids or salts
IT1141286B (it) * 1980-04-17 1986-10-01 Dob Far Spa Esteri delle desacetossi cefalosporine loro sali e procedimenti per il loro ottenimento
JPS5855491A (ja) * 1981-09-29 1983-04-01 Eisai Co Ltd ３−カルバモイルオキシメチルセフエム誘導体およびその製造法
KR20020085180A (ko) * 2001-05-07 2002-11-16 주식회사 엘지생명과학 신규 세팔로스포린계 항생제 및 이의 제조 방법
KR20020085176A (ko) * 2001-05-07 2002-11-16 주식회사 엘지생명과학 신규 세팔로스포린계 항생제 및 이의 제조 방법
GB0116142D0 (en) * 2001-07-02 2001-08-22 Astrazeneca Ab Method

Family Cites Families (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3769281A (en) * 1970-07-09 1973-10-30 Lilly Co Eli Deblocking process for cephalosporin antibiotics
US3867380A (en) * 1971-02-18 1975-02-18 Smithkline Corp 3-Heterocyclic thiomethylcephalosporins
IL38099A (en) * 1970-12-17 1976-01-30 Smith Kline French Lab 3-heterocyclyl thiomethylcephalosporins
CH606016A5 (en) * 1973-08-01 1978-10-13 Ciba Geigy Ag Antibacterial 3-pyridino-cephalosporin cpds.
AR208171A1 (es) * 1972-09-29 1976-12-09 Ciba Geigy Ag Procedimiento para la obtencion de nuevos derivados del acido cef-3-em-4-carboxilico
JPS551273B2 (nl) * 1972-12-21 1980-01-12
CA1022544A (en) * 1972-12-21 1977-12-13 Yukiyasu Murakami Process of preparing a heterocyclic acyl group-substituted cephalosporin derivative
JPS5143785A (en) * 1974-10-11 1976-04-14 Yamanouchi Pharma Co Ltd Shinsefuarosuhorinkanrenkagobutsuno goseiho
GB1479711A (en) * 1973-06-12 1977-07-13 Beecham Group Ltd Acylureido cephalosporins
US4058610A (en) * 1973-09-13 1977-11-15 Pfizer Inc. 7-D-(α-Acylamino-arylacetamido)-cephalosporanic acid derivatives
JPS4970990A (nl) * 1973-09-29 1974-07-09
DE2407715C2 (de) * 1974-02-18 1982-12-02 Bayer Ag, 5090 Leverkusen Cephalosporine, Verfahren zu ihrer Herstellung sowie Arzneimittel
US4107304A (en) * 1974-02-18 1978-08-15 Bayer Aktiengesellschaft Oxo-imidazolidine substituted cephalosporins and antibacterial compositions and methods of combatting bacteria employing them
DE2512284A1 (de) * 1974-03-28 1975-10-09 Fujisawa Pharmaceutical Co Cephalosporansaeurederivate, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische mittel
US4068074A (en) * 1974-04-05 1978-01-10 Yamanouchi Pharmaceutical Co., Ltd. Cephalosporin derivatives having at the 3-position of the cephem ring a heterocyclic thiomethyl group with a carboxy or sulfo group and at the 7-position of the cephem ring an α-heterocylic acylaminophenyl-acetamide group
US4110327A (en) * 1974-05-09 1978-08-29 Toyama Chemical Co., Ltd. 2,3 Diketo-piperazinocarbonylamino alkanoic acids and derivatives
JPS5170788A (en) * 1974-12-13 1976-06-18 Toyama Chemical Co Ltd Shinkina sefuarosuhorinruino seizoho
US4154831A (en) * 1974-05-13 1979-05-15 Ciba-Geigy Corporation Cephalosporins having an α-acylaminoacetic acid side chain
CH606001A5 (nl) * 1974-05-13 1978-10-13 Ciba Geigy Ag
JPS50151895A (nl) * 1974-05-31 1975-12-06
JPS50157387A (nl) * 1974-06-06 1975-12-19
US3985740A (en) * 1974-07-26 1976-10-12 Bristol-Myers Company 7-[D-(α-amino-α-phenyl-, 2-thienyl- and 3-thienylacetamido)]-3-(5-methylthiazol-2-yl)carbonylthiomethyl-3-cephem-4-carboxylic acids
CA1074784A (en) * 1974-09-06 1980-04-01 Sumitomo Chemical Company N-ACYLAMINO-.alpha.-ARYLACETAMIDO CEPHALOSPORINS
JPS5132576A (en) * 1974-09-06 1976-03-19 Sumitomo Chemical Co Nn ashiruamino arufua ariiruasetoamidosefuarosuhorinruinoseiho
GB1498025A (en) * 1975-10-01 1978-01-18 Beecham Group Ltd 3-carbamoyloxymethyl-7-8-(substituted acetamido)-3-cephem-4-carboxylic acid derivatives and methods for their preparation
GB1469797A (en) * 1974-11-07 1977-04-06 Pfizer Ltd Antibacterial cephalosporin derivatives
US4053470A (en) * 1974-12-23 1977-10-11 Parke, Davis & Company Substituted-1,2-dihydro-2-oxonicotinyl-cephalosporins
US4224442A (en) * 1975-03-03 1980-09-23 Eli Lilly And Company 7-Ureido acetamido substituted cephalosporin antibiotics
JPS5293790A (en) * 1976-02-02 1977-08-06 Sumitomo Chem Co Ltd 7-(n-acylamino-alpha-arylacetamide) cephalosporins
US4061630A (en) * 1976-02-20 1977-12-06 Eli Lilly And Company 7-Substituted-ureido-3-carbamoyloxymethyl cephalosporin antibiotics
AU498968B2 (en) * 1976-03-03 1979-03-29 Sumitomo Chemical Company, Limited Cephalosporins
US4103008A (en) * 1976-04-07 1978-07-25 Ishimaru Toshiyasu 7[2(2,3 Dioxopiperazin-1-yl-carbonylamino)substituted 2 phenylacetamido]-3-2'-thiadiazolyl cephalosporanic acid derivatives
US4048161A (en) * 1976-05-20 1977-09-13 Eli Lilly And Company 7-[α-(Benzimidazol-2-ylcarbonylamino)-arylacetamido]ephalosporins

Also Published As

Publication number Publication date
JPS6337794B2 (nl) 1988-07-27
FR2362146B1 (nl) 1982-10-15
ES472240A1 (es) 1979-10-16
CH634848A5 (de) 1983-02-28
JPS5323993A (en) 1978-03-06
US4324892A (en) 1982-04-13
US4172198A (en) 1979-10-23
DE2737066A1 (de) 1978-02-23
FR2362146A1 (fr) 1978-03-17
ES461688A1 (es) 1978-12-01

Similar Documents

Publication Publication Date Title
NL7714329A (nl) Werkwijze ter bereiding van 3-de-0-methylforti- micinen alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten.
NL7708741A (nl) Werkwijze ter bereiding van prostaanzuurderiva- ten alsmede farmaceutische preparaten die deze derivaten als actieve component bevatten.
BE826260A (nl) Werkwijze voor het bereiden van werkzame cyclohexanolderivaten en van preparaten, die deze bevatten
NL7803195A (nl) Heterocyclische verbindingen met farmaceutische activiteit, werkwijzen ter bereiding daarvan, alsmede farmaceutische preparaten, die deze verbindingen als actieve component bevatten.
NL7709697A (nl) Werkwijze ter bereiding van thiazolidinederivaten, alsmede farmaceutische preparaten die deze ver- bindingen als actieve component bevatten.
NL7603193A (nl) Werkwijze ter bereiding van acyclische, alicycli- sche en aromatische n-gesubstitueerde halogeen-2- -pyrrolidinonen met herbicidewerking alsmede her- bicidepreparaten die deze verbindingen als actie- ve component bevatten.
NL7706064A (nl) Werkwijze ter bereiding van heterocyclische verbindingen alsmede van farmaceutische pre- paraten die deze verbindingen als actieve component omvatten.
NL7700379A (nl) Werkwijze ter bereiding van anthracyclinegly- cosiden, alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten.
NL7614538A (nl) Werkwijze ter bereiding van farmacologisch actieve heterocyclische verbindingen en farmaceutische preparaten die deze verbindingen bevatten.
NL7713470A (nl) Werkwijze ter bereiding van 2-gesubstitueerde benzimidazoolverbindingen en de zuuradditiezou- ten daarvan alsmede farmaceutische preparaten die deze verbindingen als actieve component be- vatten.
BE857181A (nl) Werkwijze ter bereiding van n-alkynyl-&-(gesugstitueerde fenoxy) alkylamiden met herbicidewerking alsmede herbicide-preparaten die deze verbindingen als actieve component bevatten
NL7604797A (nl) Werkwijze ter bereiding van nieuwe antibacteriele middelen alsmede preparaten die deze verbindingen als actieve component bevatten.
NL7610480A (nl) Werkwijze ter bereiding van hypolipemische ver- bindingen alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten.
NL7607337A (nl) Werkwijze ter bereiding van spirocycloalkyl- prostaanzuren en derivaten daarvan, alsmede geneeskundige preparaten die deze verbindingen als actieve component bevatten.
NL7609559A (nl) Werkwijze ter bereiding van oxazolidinonen alsmede geneeskrachtige middelen die deze ver- bindingen als actieve component bevatten.
NL7702180A (nl) Werkwijze ter bereiding van 9-gesubstitueerde- -8-azapurinen alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten.
NL7711414A (nl) Werkwijze ter bereiding van n-gesubstitueerde lactamen, alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten.
NL7707150A (nl) Werkwijze ter bereiding van 2-lagere alkyl-7-ge- substitueerde-2 of 3-cefem-4-carbonzuurverbin- dingen, alsmede farmaceutische preparaten die deze verbindingen als actieve component bevatten.
NL7709092A (nl) Werkwijze ter bereiding van cefalosporinever- bindingen met antibacteriele activiteit als- mede farmaceutische preparaten die deze ver- bindingen als actieve component bevatten.
NL155827B (nl) Werkwijze voor de bereiding van antibacterieel werkzame benzylpyrimidinen, alsmede voor de bereiding van antibacterieel werkzame preparaten, die deze verbindingen bevatten, en de gevormde preparaten.
NL7515085A (nl) Werkwijze ter bereiding van cefalosporinederiva- ten als antimicrobiele preparaten die deze deri- vaten als actieve componenten bevatten.
NL7807890A (nl) Pyranochromoonderivaten, alsmede preparaten voor de be- handeling van allergische aandoeningen, die deze ver- bindingen bevatten.
NL7714063A (nl) Werkwijze ter bereiding van imidazolinen alsmede pesticidepreparaten die deze verbindingen als actieve component bevatten.
NL7505961A (nl) Werkwijze ter bereiding van een antibacterieel middel, alsmede preparaten die dit middel als actieve component bevatten.
NL7707751A (nl) Werkwijze ter bereiding van cefalosporineverbin- dingen alsmede antibacteriele preparaten die deze componenten bevatten.

Legal Events

Date Code Title Description
BV The patent application has lapsed