LU88323A1 - Comprimes solubles dans l'eau - Google Patents
Comprimes solubles dans l'eau Download PDFInfo
- Publication number
- LU88323A1 LU88323A1 LU88323A LU88323A LU88323A1 LU 88323 A1 LU88323 A1 LU 88323A1 LU 88323 A LU88323 A LU 88323A LU 88323 A LU88323 A LU 88323A LU 88323 A1 LU88323 A1 LU 88323A1
- Authority
- LU
- Luxembourg
- Prior art keywords
- tablet
- water
- tablet according
- granules
- tablets
- Prior art date
Links
- 239000004554 water soluble tablet Substances 0.000 title 1
- 239000003826 tablet Substances 0.000 claims abstract description 226
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- 239000006185 dispersion Substances 0.000 claims abstract description 57
- 229960004150 aciclovir Drugs 0.000 claims abstract description 56
- MKUXAQIIEYXACX-UHFFFAOYSA-N aciclovir Chemical compound N1C(N)=NC(=O)C2=C1N(COCCO)C=N2 MKUXAQIIEYXACX-UHFFFAOYSA-N 0.000 claims abstract description 56
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims abstract description 50
- PYZRQGJRPPTADH-UHFFFAOYSA-N lamotrigine Chemical compound NC1=NC(N)=NN=C1C1=CC=CC(Cl)=C1Cl PYZRQGJRPPTADH-UHFFFAOYSA-N 0.000 claims abstract description 49
- 229960001848 lamotrigine Drugs 0.000 claims abstract description 47
- 239000004565 water dispersible tablet Substances 0.000 claims abstract description 25
- 239000000440 bentonite Substances 0.000 claims abstract description 17
- 229910000278 bentonite Inorganic materials 0.000 claims abstract description 17
- SVPXDRXYRYOSEX-UHFFFAOYSA-N bentoquatam Chemical compound O.O=[Si]=O.O=[Al]O[Al]=O SVPXDRXYRYOSEX-UHFFFAOYSA-N 0.000 claims abstract description 17
- 229960003459 allopurinol Drugs 0.000 claims abstract description 13
- OFCNXPDARWKPPY-UHFFFAOYSA-N allopurinol Chemical compound OC1=NC=NC2=C1C=NN2 OFCNXPDARWKPPY-UHFFFAOYSA-N 0.000 claims abstract description 12
- XBDQKXXYIPTUBI-UHFFFAOYSA-N dimethylselenoniopropionate Natural products CCC(O)=O XBDQKXXYIPTUBI-UHFFFAOYSA-N 0.000 claims abstract description 12
- FGEANDFKBDCXNV-UHFFFAOYSA-N 9h-purine-2,8-dione Chemical compound O=C1N=CC2=NC(=O)NC2=N1 FGEANDFKBDCXNV-UHFFFAOYSA-N 0.000 claims abstract description 9
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- IEDVJHCEMCRBQM-UHFFFAOYSA-N trimethoprim Chemical compound COC1=C(OC)C(OC)=CC(CC=2C(=NC(N)=NC=2)N)=C1 IEDVJHCEMCRBQM-UHFFFAOYSA-N 0.000 claims abstract description 9
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- 239000000080 wetting agent Substances 0.000 claims description 4
- BSJMWHQBCZFXBR-UHFFFAOYSA-N 3-[4-(p-chlorophenyl)cyclohexyl]-4-hydroxy-1,2-naphthoquinone Chemical compound O=C1C(=O)C2=CC=CC=C2C(O)=C1C(CC1)CCC1C1=CC=C(Cl)C=C1 BSJMWHQBCZFXBR-UHFFFAOYSA-N 0.000 claims description 3
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- HSRJKNPTNIJEKV-UHFFFAOYSA-N Guaifenesin Chemical compound COC1=CC=CC=C1OCC(O)CO HSRJKNPTNIJEKV-UHFFFAOYSA-N 0.000 claims description 3
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
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- A—HUMAN NECESSITIES
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- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
- A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/06—Aluminium, calcium or magnesium; Compounds thereof, e.g. clay
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2009—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Oncology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- General Preparation And Processing Of Foods (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Glanulating (AREA)
Applications Claiming Priority (10)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB919102019A GB9102019D0 (en) | 1991-01-30 | 1991-01-30 | Pharmaceutical formulations |
| GB9102019 | 1991-01-31 | ||
| GB919124803A GB9124803D0 (en) | 1991-11-22 | 1991-11-22 | Pharmaceutical formulations |
| GB9124807 | 1991-11-22 | ||
| GB9124803 | 1991-11-22 | ||
| GB919124807A GB9124807D0 (en) | 1991-11-22 | 1991-11-22 | Pharmaceutical formulations |
| GB9125005 | 1991-11-25 | ||
| GB919125005A GB9125005D0 (en) | 1991-11-25 | 1991-11-25 | Pharmaceutical formulations |
| GB9200163 | 1992-01-29 | ||
| PCT/GB1992/000163 WO1992013527A1 (en) | 1991-01-30 | 1992-01-29 | Water-dispersible tablets |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| LU88323A1 true LU88323A1 (fr) | 1994-01-05 |
Family
ID=27450613
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LU88323A LU88323A1 (fr) | 1991-01-30 | 1993-06-22 | Comprimes solubles dans l'eau |
Country Status (37)
| Country | Link |
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| US (2) | US5556639A (de) |
| EP (1) | EP0522128B1 (de) |
| JP (2) | JP3118255B2 (de) |
| KR (1) | KR100190254B1 (de) |
| AT (1) | ATE133068T1 (de) |
| AU (2) | AU653203B2 (de) |
| BE (1) | BE1004461A5 (de) |
| BG (1) | BG61665B2 (de) |
| CA (1) | CA2098108C (de) |
| CH (1) | CH685978A5 (de) |
| CY (1) | CY2007A (de) |
| CZ (1) | CZ286723B6 (de) |
| DE (2) | DE69207656T2 (de) |
| DK (2) | DK0522128T3 (de) |
| ES (2) | ES2089498T3 (de) |
| FI (2) | FI111605B (de) |
| FR (1) | FR2671970B1 (de) |
| GB (1) | GB2257363B (de) |
| GR (1) | GR3019545T3 (de) |
| HK (1) | HK78597A (de) |
| HU (2) | HU221677B1 (de) |
| IE (1) | IE77165B1 (de) |
| IL (1) | IL100796A (de) |
| IT (1) | IT1257473B (de) |
| LU (1) | LU88323A1 (de) |
| MX (1) | MX9200412A (de) |
| MY (2) | MY110880A (de) |
| NL (1) | NL9220009A (de) |
| NO (1) | NO306697B1 (de) |
| PA (1) | PA7695401A1 (de) |
| PL (1) | PL169106B1 (de) |
| RU (1) | RU2106861C1 (de) |
| SA (1) | SA92120365B1 (de) |
| SE (1) | SE9302363L (de) |
| SK (2) | SK282071B6 (de) |
| UA (1) | UA37214C2 (de) |
| WO (1) | WO1992013527A1 (de) |
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| GB8613183D0 (en) * | 1986-05-30 | 1986-07-02 | Wellcome Found | Triazine salt |
| DE3635864A1 (de) * | 1986-06-26 | 1988-05-05 | Gerhard Gergely | Verfahren zum herstellen eines brausegranulates, danach hergestelltes brausegranulat sowie dessen verwendung |
| US4757090A (en) * | 1986-07-14 | 1988-07-12 | Mallinckrodt, Inc. | Direct tableting acetaminophen compositions |
| KR960001372B1 (ko) * | 1986-09-24 | 1996-01-26 | 예일 유니버시티 | 레트로비루스로 감염된 환자의 치료에 사용되는 2',3'-디디옥시사이티딘-2'-엔(2',3'-디디옥시-2',3'-디디하이드로사이티딘)의 항생물질 |
| GB8624628D0 (en) * | 1986-10-14 | 1986-11-19 | Scras | Soluble/splitable tablets |
| US4771077A (en) * | 1986-10-21 | 1988-09-13 | American Home Products Corporation (Del.) | Spray dried acetaminophen |
| GB8628359D0 (en) * | 1986-11-27 | 1986-12-31 | Zyma Sa | Galenical formulation |
| DE3887179T2 (de) * | 1987-03-02 | 1994-06-16 | Brocades Pharma Bv | Pharmazeutische Zusammensetzung, pharmazeutisches Granulat und Verfahren zu ihrer Herstellung. |
| ATE73328T1 (de) * | 1987-05-08 | 1992-03-15 | Smith Kline French Lab | Pharmazeutische zusammensetzungen. |
| US4904477A (en) * | 1987-07-08 | 1990-02-27 | American Home Products Corporation | Spray dried ibuprofen compositions |
| ES2026198T3 (es) * | 1987-07-22 | 1992-04-16 | Farvalsa Ag | Compuesto a base de acido valproico solido, estable a la humedad y metodo para su preparacion. |
| JP2527973B2 (ja) * | 1987-08-05 | 1996-08-28 | 株式会社資生堂 | 球状粘土鉱物及びその製造方法 |
| DE3806633A1 (de) * | 1987-09-01 | 1989-03-09 | Bayer Ag | Antivirales mittel |
| US4837031A (en) * | 1987-09-17 | 1989-06-06 | Mallinckrodt, Inc. | Compositions containing ibuprofen |
| JP2537062B2 (ja) * | 1987-10-02 | 1996-09-25 | 株式会社資生堂 | 薬剤組成物 |
| US4999200A (en) * | 1987-12-09 | 1991-03-12 | Marion Laboratories | Psyllium tablet composition, method of manufacture and method of use |
| ES2060737T3 (es) * | 1988-02-25 | 1994-12-01 | Yamanouchi Europ Bv | Procedimiento de preparacion de un granulado farmaceutico. |
| US4910023A (en) * | 1988-06-09 | 1990-03-20 | Warner-Lambert Company | Drug in combination with flavor masking agent and method for making same |
| YU120988A (en) * | 1988-06-23 | 1990-06-30 | Lek Tovarna Farmacevtskih | Process for preparing new dispersion pills of cimetidine |
| IT1226549B (it) * | 1988-07-12 | 1991-01-24 | Resa Farma | Composizioni farmaceutiche ad attivita' analgesica ed antiinfiammatoria per uso orale, dotate di ottima palatabilita' ed esenti da effetti irritanti sulle mucose. |
| YU183988A (en) * | 1988-09-30 | 1990-08-31 | Lek Tovarna Farmacevtskih | Process for preparing dispersion pills of dihydroergotoxine |
| JPH02111620A (ja) * | 1988-10-21 | 1990-04-24 | Kunimine Kogyo Kk | 水中分散性粒剤 |
| US4965072A (en) * | 1988-11-03 | 1990-10-23 | Miles Inc. | Granulating composition and method |
| US5073377A (en) * | 1988-11-03 | 1991-12-17 | Miles Inc. | Method of preparing oral dosage forms with a granulating composition |
| JPH02145501A (ja) * | 1988-11-25 | 1990-06-05 | Sanyo Chem Ind Ltd | 殺生剤粒剤組成物 |
| FI895821A0 (fi) * | 1988-12-07 | 1989-12-05 | Wellcome Found | Farmaceutiskt aktiva cns foereningar. |
| US4927639A (en) * | 1989-02-02 | 1990-05-22 | Warner-Lambert Company | Modified release gemfibrozil composition |
| US4925676A (en) * | 1989-02-02 | 1990-05-15 | Warner-Lambert Company | Extended release gemfibrozil composition |
| ES2055894T3 (es) * | 1989-04-07 | 1994-09-01 | Ciba Geigy Ag | Concentrados de sustancias activas pesticidas y su preparacion. |
| US4970078A (en) * | 1989-05-25 | 1990-11-13 | Aqualon Company | Crosslinked carboxymethyguar tablet disintegrant |
| US5260304A (en) * | 1989-09-07 | 1993-11-09 | Gerhard Gergely | Pharmaceutical preparation binding with gastric acid |
| US5037658A (en) * | 1989-09-14 | 1991-08-06 | Hoechst-Roussel Pharmaceuticals, Inc. | Direct dry compressible acetaminophen composition |
| US5064656A (en) * | 1989-11-14 | 1991-11-12 | Dr. Gergely & Co. | Uncoated pharmaceutical reaction tablet |
| US5136080A (en) * | 1989-12-04 | 1992-08-04 | Burroughs Wellcome Co. | Nitrile compounds |
| JP3069665B2 (ja) * | 1990-03-15 | 2000-07-24 | 住友化学工業株式会社 | 農業用粒状水和剤組成物 |
| GB9012316D0 (en) * | 1990-06-01 | 1990-07-18 | Wellcome Found | Pharmacologically active cns compounds |
| GB9012311D0 (en) * | 1990-06-01 | 1990-07-18 | Wellcome Found | Pharmacologically active cns compounds |
| US5087454A (en) * | 1990-07-30 | 1992-02-11 | American Home Products Corporation | Ibuprofen tablet |
| GB9025372D0 (en) * | 1990-11-22 | 1991-01-09 | Nat Res Dev | Pharmaceutical dosage forms |
-
1992
- 1992-01-29 GB GB9218097A patent/GB2257363B/en not_active Revoked
- 1992-01-29 IE IE920284A patent/IE77165B1/en not_active IP Right Cessation
- 1992-01-29 NL NL9220009A patent/NL9220009A/nl active Search and Examination
- 1992-01-29 JP JP04503284A patent/JP3118255B2/ja not_active Expired - Lifetime
- 1992-01-29 IL IL10079692A patent/IL100796A/en not_active IP Right Cessation
- 1992-01-29 EP EP92903508A patent/EP0522128B1/de not_active Expired - Lifetime
- 1992-01-29 US US08/090,111 patent/US5556639A/en not_active Expired - Lifetime
- 1992-01-29 CZ CZ19931082A patent/CZ286723B6/cs not_active IP Right Cessation
- 1992-01-29 UA UA93002090A patent/UA37214C2/uk unknown
- 1992-01-29 DE DE69207656T patent/DE69207656T2/de not_active Expired - Lifetime
- 1992-01-29 KR KR1019930702233A patent/KR100190254B1/ko not_active IP Right Cessation
- 1992-01-29 MY MYPI92000143A patent/MY110880A/en unknown
- 1992-01-29 HU HU9302212A patent/HU221677B1/hu unknown
- 1992-01-29 WO PCT/GB1992/000163 patent/WO1992013527A1/en not_active IP Right Cessation
- 1992-01-29 BE BE9200088A patent/BE1004461A5/fr not_active IP Right Cessation
- 1992-01-29 DE DE4290300T patent/DE4290300T1/de not_active Withdrawn
- 1992-01-29 FR FR9200938A patent/FR2671970B1/fr not_active Expired - Fee Related
- 1992-01-29 RU RU93051524A patent/RU2106861C1/ru active
- 1992-01-29 SK SK817-93A patent/SK282071B6/sk unknown
- 1992-01-29 DK DK92903508.7T patent/DK0522128T3/da active
- 1992-01-29 CA CA002098108A patent/CA2098108C/en not_active Expired - Lifetime
- 1992-01-29 AU AU11863/92A patent/AU653203B2/en not_active Expired
- 1992-01-29 ES ES92903508T patent/ES2089498T3/es not_active Expired - Lifetime
- 1992-01-29 AT AT92903508T patent/ATE133068T1/de not_active IP Right Cessation
- 1992-01-29 PL PL92300134A patent/PL169106B1/pl unknown
- 1992-01-29 SK SK1655-2000A patent/SK282072B6/sk unknown
- 1992-01-29 CH CH309292A patent/CH685978A5/fr not_active IP Right Cessation
- 1992-01-29 ES ES09250043A patent/ES2080641B1/es not_active Expired - Fee Related
- 1992-01-30 MX MX9200412A patent/MX9200412A/es unknown
- 1992-01-30 IT ITRM920069A patent/IT1257473B/it active IP Right Grant
- 1992-02-02 SA SA92120365A patent/SA92120365B1/ar unknown
-
1993
- 1993-06-22 LU LU88323A patent/LU88323A1/fr unknown
- 1993-07-02 NO NO932422A patent/NO306697B1/no not_active IP Right Cessation
- 1993-07-08 SE SE9302363A patent/SE9302363L/xx not_active Application Discontinuation
- 1993-07-27 DK DK93878A patent/DK87893D0/da not_active Application Discontinuation
- 1993-07-29 FI FI933401A patent/FI111605B/fi active
- 1993-08-26 BG BG098071A patent/BG61665B2/bg unknown
-
1994
- 1994-07-13 AU AU67454/94A patent/AU659581B2/en not_active Expired
- 1994-10-03 US US08/317,300 patent/US5660860A/en not_active Expired - Lifetime
-
1995
- 1995-06-28 HU HU95P/P00506P patent/HU211161A9/hu unknown
- 1995-08-24 PA PA19957695401A patent/PA7695401A1/es unknown
-
1996
- 1996-04-03 GR GR960400936T patent/GR3019545T3/el unknown
-
1997
- 1997-06-12 HK HK78597A patent/HK78597A/xx not_active IP Right Cessation
-
1998
- 1998-02-20 CY CY200798A patent/CY2007A/xx unknown
- 1998-02-27 MY MYPI98000866A patent/MY120025A/en unknown
-
2000
- 2000-03-14 JP JP2000070675A patent/JP3483515B2/ja not_active Expired - Lifetime
-
2002
- 2002-09-24 FI FI20021701A patent/FI20021701A/fi unknown
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