DK153787C - Analogifremgangsmaade til fremstilling af substituerede 3,5-diamino-6-phenyl-1,2,4-triaziner og alfa-cyanobenzyliden-aminoguanidinforbindelser til anvendelse som mellemprodukter herved - Google Patents

Analogifremgangsmaade til fremstilling af substituerede 3,5-diamino-6-phenyl-1,2,4-triaziner og alfa-cyanobenzyliden-aminoguanidinforbindelser til anvendelse som mellemprodukter herved

Info

Publication number
DK153787C
DK153787C DK233880A DK233880A DK153787C DK 153787 C DK153787 C DK 153787C DK 233880 A DK233880 A DK 233880A DK 233880 A DK233880 A DK 233880A DK 153787 C DK153787 C DK 153787C
Authority
DK
Denmark
Prior art keywords
cyanobenzylideen
aminoguanide
triazines
alfa
diamino
Prior art date
Application number
DK233880A
Other languages
English (en)
Other versions
DK153787B (da
DK233880A (da
Inventor
Martin George Baxter
Albert Reginald Elphick
Alistair Ainslie Miller
David Alan Sawyer
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10505597&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK153787(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of DK233880A publication Critical patent/DK233880A/da
Publication of DK153787B publication Critical patent/DK153787B/da
Application granted granted Critical
Publication of DK153787C publication Critical patent/DK153787C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D253/00—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/06—1,2,4-Triazines
    • C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
    • C07D253/07—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D253/075—Two hetero atoms, in positions 3 and 5
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C281/00—Derivatives of carbonic acid containing functional groups covered by groups C07C269/00 - C07C279/00 in which at least one nitrogen atom of these functional groups is further bound to another nitrogen atom not being part of a nitro or nitroso group
    • C07C281/16—Compounds containing any of the groups, e.g. aminoguanidine
    • C07C281/18—Compounds containing any of the groups, e.g. aminoguanidine the other nitrogen atom being further doubly-bound to a carbon atom, e.g. guanylhydrazones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/15—Preparation of carboxylic acids or their salts, halides or anhydrides by reaction of organic compounds with carbon dioxide, e.g. Kolbe-Schmitt synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
    • C07C51/363—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
DK233880A 1979-06-01 1980-05-30 Analogifremgangsmaade til fremstilling af substituerede 3,5-diamino-6-phenyl-1,2,4-triaziner og alfa-cyanobenzyliden-aminoguanidinforbindelser til anvendelse som mellemprodukter herved DK153787C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7919257 1979-06-01
GB7919257 1979-06-01

Publications (3)

Publication Number Publication Date
DK233880A DK233880A (da) 1980-12-02
DK153787B DK153787B (da) 1988-09-05
DK153787C true DK153787C (da) 1989-01-16

Family

ID=10505597

Family Applications (1)

Application Number Title Priority Date Filing Date
DK233880A DK153787C (da) 1979-06-01 1980-05-30 Analogifremgangsmaade til fremstilling af substituerede 3,5-diamino-6-phenyl-1,2,4-triaziner og alfa-cyanobenzyliden-aminoguanidinforbindelser til anvendelse som mellemprodukter herved

Country Status (30)

Country Link
US (2) US4486354A (da)
EP (2) EP0021121B1 (da)
JP (2) JPS5625169A (da)
AR (1) AR227521A1 (da)
AT (1) AT370097B (da)
AU (2) AU530999B2 (da)
BG (1) BG60427B2 (da)
CA (1) CA1112643A (da)
CS (1) CS234018B2 (da)
CZ (1) CZ384891A3 (da)
DD (1) DD151309A5 (da)
DK (1) DK153787C (da)
ES (1) ES8104993A1 (da)
FI (1) FI67844C (da)
GE (1) GEP19960470B (da)
GR (1) GR68380B (da)
HU (1) HU182086B (da)
IE (1) IE49823B1 (da)
IL (1) IL60201A (da)
IT (1) IT1147087B (da)
MX (1) MX9202962A (da)
MY (1) MY8500062A (da)
NL (1) NL950007I2 (da)
NZ (1) NZ193890A (da)
PL (1) PL124029B1 (da)
SU (1) SU1055331A3 (da)
UA (1) UA5576A1 (da)
YU (1) YU145680A (da)
ZA (1) ZA803250B (da)
ZW (1) ZW12980A1 (da)

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TWI826531B (zh) 2018-09-21 2023-12-21 南韓商愛思開生物製藥股份有限公司 具有㗁二唑之化合物及包含該化合物之醫藥組合物

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Also Published As

Publication number Publication date
BG60427B2 (bg) 1995-03-31
CS234018B2 (en) 1985-03-14
DD151309A5 (de) 1981-10-14
NZ193890A (en) 1984-07-06
EP0059987A1 (en) 1982-09-15
UA5576A1 (uk) 1994-12-28
DK153787B (da) 1988-09-05
DK233880A (da) 1980-12-02
EP0021121A1 (en) 1981-01-07
NL950007I1 (nl) 1995-06-16
JPH0144706B2 (da) 1989-09-29
IE801126L (en) 1980-12-01
JPS5625169A (en) 1981-03-10
EP0059987B1 (en) 1985-08-14
PL224633A1 (da) 1981-02-13
ES491998A0 (es) 1981-05-16
ZW12980A1 (en) 1982-01-06
ZA803250B (en) 1982-01-27
MY8500062A (en) 1985-12-31
IE49823B1 (en) 1985-12-25
US4486354A (en) 1984-12-04
MX9202962A (es) 1992-07-01
AU566870B2 (en) 1987-11-05
AU5890680A (en) 1980-12-04
US4602017A (en) 1986-07-22
IL60201A (en) 1984-05-31
AR227521A1 (es) 1982-11-15
IT1147087B (it) 1986-11-19
GEP19960470B (en) 1996-08-29
PL124029B1 (en) 1982-12-31
CA1112643A (en) 1981-11-17
AT370097B (de) 1983-02-25
IT8048848A0 (it) 1980-05-30
HU182086B (en) 1983-12-28
ES8104993A1 (es) 1981-05-16
AU530999B2 (en) 1983-08-04
SU1055331A3 (ru) 1983-11-15
CZ384891A3 (en) 1993-10-13
NL950007I2 (nl) 1997-02-03
FI67844B (fi) 1985-02-28
IL60201A0 (en) 1980-07-31
FI67844C (fi) 1985-06-10
JPH0144179B2 (da) 1989-09-26
FI801758A (fi) 1980-12-02
JPS6133163A (ja) 1986-02-17
GR68380B (da) 1981-12-28
ATA289680A (de) 1982-07-15
YU145680A (en) 1983-02-28
EP0021121B1 (en) 1983-05-11

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