JP2016501827A5 - - Google Patents

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JP2016501827A5
JP2016501827A5 JP2015516335A JP2015516335A JP2016501827A5 JP 2016501827 A5 JP2016501827 A5 JP 2016501827A5 JP 2015516335 A JP2015516335 A JP 2015516335A JP 2015516335 A JP2015516335 A JP 2015516335A JP 2016501827 A5 JP2016501827 A5 JP 2016501827A5
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substituted
unsubstituted
pharmaceutically acceptable
acceptable salt
alkyl
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JP2015516335A
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JP2016501827A (ja
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Priority to JP2015516335A priority Critical patent/JP2016501827A/ja
Priority claimed from PCT/JP2013/079472 external-priority patent/WO2014065434A1/en
Publication of JP2016501827A publication Critical patent/JP2016501827A/ja
Publication of JP2016501827A5 publication Critical patent/JP2016501827A5/ja
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JP2015516335A 2012-10-24 2013-10-23 Ｂａｃｅ１阻害作用を有するジヒドロオキサジンまたはオキサゼピン誘導体 Pending JP2016501827A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2015516335A JP2016501827A (ja) 2012-10-24 2013-10-23 Ｂａｃｅ１阻害作用を有するジヒドロオキサジンまたはオキサゼピン誘導体

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
JP2012234461 2012-10-24
JP2012234461 2012-10-24
JP2013154451 2013-07-25
JP2013154451 2013-07-25
PCT/JP2013/079472 WO2014065434A1 (en) 2012-10-24 2013-10-23 Dihydrooxazine or oxazepine derivatives having bace1 inhibitory activity
JP2015516335A JP2016501827A (ja) 2012-10-24 2013-10-23 Ｂａｃｅ１阻害作用を有するジヒドロオキサジンまたはオキサゼピン誘導体

Publications (2)

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JP2016501827A JP2016501827A (ja) 2016-01-21
JP2016501827A5 true JP2016501827A5 (https=) 2016-10-13

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JP2015516335A Pending JP2016501827A (ja) 2012-10-24 2013-10-23 Ｂａｃｅ１阻害作用を有するジヒドロオキサジンまたはオキサゼピン誘導体

Country Status (4)

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US (2) US9540359B2 (https=)
EP (1) EP2912035A4 (https=)
JP (1) JP2016501827A (https=)
WO (1) WO2014065434A1 (https=)

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JP7149271B2 (ja) 2016-12-15 2022-10-06 アムジエン・インコーポレーテツド β－セクレターゼ阻害剤としての１，４－チアジンジオキシドおよび１，２，４－チアジアジンジオキシド誘導体ならびに使用方法
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TW202014191A (zh) 2018-04-27 2020-04-16 日商鹽野義製藥股份有限公司 具有選擇性ｂａｃｅ１抑制活性的四氫哌喃并衍生物
CN111592557A (zh) * 2020-05-09 2020-08-28 河北合佳医药科技集团股份有限公司 一种7-氨基-3-乙烯基头孢烷酸的一步法环保制备方法

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