JP2012523425A5 - - Google Patents

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Publication number
JP2012523425A5
JP2012523425A5 JP2012504832A JP2012504832A JP2012523425A5 JP 2012523425 A5 JP2012523425 A5 JP 2012523425A5 JP 2012504832 A JP2012504832 A JP 2012504832A JP 2012504832 A JP2012504832 A JP 2012504832A JP 2012523425 A5 JP2012523425 A5 JP 2012523425A5
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JP
Japan
Prior art keywords
compound
pain
alkyl
aryl
membered heteroaryl
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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JP2012504832A
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English (en)
Japanese (ja)
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JP2012523425A (ja
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Priority claimed from PCT/US2010/030276 external-priority patent/WO2010118159A1/en
Publication of JP2012523425A publication Critical patent/JP2012523425A/ja
Publication of JP2012523425A5 publication Critical patent/JP2012523425A5/ja
Pending legal-status Critical Current

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JP2012504832A 2009-04-07 2010-04-07 脂肪酸アミドヒドロラーゼの阻害薬 Pending JP2012523425A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US16746409P 2009-04-07 2009-04-07
US61/167,464 2009-04-07
PCT/US2010/030276 WO2010118159A1 (en) 2009-04-07 2010-04-07 Inhibitors of fatty acid amide hydrolase

Publications (2)

Publication Number Publication Date
JP2012523425A JP2012523425A (ja) 2012-10-04
JP2012523425A5 true JP2012523425A5 (enExample) 2013-05-30

Family

ID=42936566

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012504832A Pending JP2012523425A (ja) 2009-04-07 2010-04-07 脂肪酸アミドヒドロラーゼの阻害薬

Country Status (6)

Country Link
US (2) US8541581B2 (enExample)
EP (1) EP2417115A4 (enExample)
JP (1) JP2012523425A (enExample)
AU (1) AU2010234449A1 (enExample)
CA (1) CA2757622A1 (enExample)
WO (1) WO2010118159A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
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JO3598B1 (ar) 2006-10-10 2020-07-05 Infinity Discovery Inc الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني
WO2011085216A2 (en) 2010-01-08 2011-07-14 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating parkinson's disease and restless legs syndrome
CA2788587C (en) 2010-02-03 2020-03-10 Infinity Pharmaceuticals, Inc. Fatty acid amide hydrolase inhibitors
WO2011123719A2 (en) 2010-03-31 2011-10-06 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating abdominal, visceral and pelvic pain
CN105566368B (zh) * 2016-01-11 2017-09-15 沧州普瑞东方科技有限公司 一种合成n‑取代哌啶‑4‑硼酸酯的方法
EP3762034B1 (en) 2018-03-05 2025-08-27 Wylder Nation Foundation A fatty acid amide hydrolase (faahi) inhibitor for use in inhibiting the cellular accumulation of a sphingolipid in a subject that has lysosomal storage disease or disorder
CN111171063B (zh) * 2020-01-08 2022-06-14 大连双硼医药化工有限公司 一种合成n-取代哌啶-4-硼酸的工艺方法

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