JP2019513778A5 - - Google Patents
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- JP2019513778A5 JP2019513778A5 JP2018553876A JP2018553876A JP2019513778A5 JP 2019513778 A5 JP2019513778 A5 JP 2019513778A5 JP 2018553876 A JP2018553876 A JP 2018553876A JP 2018553876 A JP2018553876 A JP 2018553876A JP 2019513778 A5 JP2019513778 A5 JP 2019513778A5
- Authority
- JP
- Japan
- Prior art keywords
- membered
- alkyl
- optionally substituted
- halo
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022036728A JP7420847B2 (ja) | 2016-04-15 | 2022-03-10 | Ehmt1およびehmt2阻害剤としてのアミン置換アリールまたはヘテロアリール化合物 |
| JP2024002232A JP2024045202A (ja) | 2016-04-15 | 2024-01-11 | Ehmt1およびehmt2阻害剤としてのアミン置換アリールまたはヘテロアリール化合物 |
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662323602P | 2016-04-15 | 2016-04-15 | |
| US62/323,602 | 2016-04-15 | ||
| US201662348837P | 2016-06-10 | 2016-06-10 | |
| US62/348,837 | 2016-06-10 | ||
| US201662402997P | 2016-09-30 | 2016-09-30 | |
| US62/402,997 | 2016-09-30 | ||
| PCT/US2017/027918 WO2017181177A1 (en) | 2016-04-15 | 2017-04-17 | Amine-substituted aryl or heteroaryl compounds as ehmt1 and ehmt2 inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022036728A Division JP7420847B2 (ja) | 2016-04-15 | 2022-03-10 | Ehmt1およびehmt2阻害剤としてのアミン置換アリールまたはヘテロアリール化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2019513778A JP2019513778A (ja) | 2019-05-30 |
| JP2019513778A5 true JP2019513778A5 (enExample) | 2020-05-28 |
| JP7041070B2 JP7041070B2 (ja) | 2022-03-23 |
Family
ID=58664786
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018553876A Expired - Fee Related JP7041070B2 (ja) | 2016-04-15 | 2017-04-17 | Ehmt1およびehmt2阻害剤としてのアミン置換アリールまたはヘテロアリール化合物 |
| JP2022036728A Active JP7420847B2 (ja) | 2016-04-15 | 2022-03-10 | Ehmt1およびehmt2阻害剤としてのアミン置換アリールまたはヘテロアリール化合物 |
| JP2024002232A Pending JP2024045202A (ja) | 2016-04-15 | 2024-01-11 | Ehmt1およびehmt2阻害剤としてのアミン置換アリールまたはヘテロアリール化合物 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022036728A Active JP7420847B2 (ja) | 2016-04-15 | 2022-03-10 | Ehmt1およびehmt2阻害剤としてのアミン置換アリールまたはヘテロアリール化合物 |
| JP2024002232A Pending JP2024045202A (ja) | 2016-04-15 | 2024-01-11 | Ehmt1およびehmt2阻害剤としてのアミン置換アリールまたはヘテロアリール化合物 |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US20170355712A1 (enExample) |
| EP (1) | EP3442947B1 (enExample) |
| JP (3) | JP7041070B2 (enExample) |
| KR (2) | KR20230130747A (enExample) |
| CN (1) | CN109153650A (enExample) |
| AU (3) | AU2017250369A1 (enExample) |
| BR (1) | BR112018071093A2 (enExample) |
| CA (1) | CA3021062A1 (enExample) |
| CL (2) | CL2018002928A1 (enExample) |
| CO (1) | CO2018012181A2 (enExample) |
| DK (1) | DK3442947T3 (enExample) |
| ES (1) | ES2953512T3 (enExample) |
| FI (1) | FI3442947T3 (enExample) |
| HU (1) | HUE064145T2 (enExample) |
| IL (3) | IL307931A (enExample) |
| LT (1) | LT3442947T (enExample) |
| MA (1) | MA44666A (enExample) |
| MX (2) | MX395342B (enExample) |
| PL (1) | PL3442947T3 (enExample) |
| PT (1) | PT3442947T (enExample) |
| SG (2) | SG10201913471VA (enExample) |
| SI (1) | SI3442947T1 (enExample) |
| TW (1) | TWI751155B (enExample) |
| WO (1) | WO2017181177A1 (enExample) |
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| JP7425724B2 (ja) * | 2017-10-17 | 2024-01-31 | エピザイム,インコーポレイティド | Ehmt2阻害剤としてのアミン置換複素環化合物及びその誘導体 |
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| WO2021007488A1 (en) | 2019-07-11 | 2021-01-14 | Enanta Pharmaceuticals, Inc. | Substituted heterocycles as antiviral agents |
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| US20240368139A1 (en) * | 2021-10-15 | 2024-11-07 | Tango Therapeutics, Inc. | Novel modulators of ehmt1 and ehmt2 and therapeutic use thereof |
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| CN115947692B (zh) * | 2022-12-28 | 2024-12-27 | 上海再启生物技术有限公司 | 一种制备2-氯-4-(甲氧基甲基)嘧啶的方法 |
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-
2017
- 2017-04-17 IL IL307931A patent/IL307931A/en unknown
- 2017-04-17 IL IL281319A patent/IL281319B2/en unknown
- 2017-04-17 LT LTEPPCT/US2017/027918T patent/LT3442947T/lt unknown
- 2017-04-17 SG SG10201913471VA patent/SG10201913471VA/en unknown
- 2017-04-17 WO PCT/US2017/027918 patent/WO2017181177A1/en not_active Ceased
- 2017-04-17 MX MX2018012622A patent/MX395342B/es unknown
- 2017-04-17 PT PT177209210T patent/PT3442947T/pt unknown
- 2017-04-17 KR KR1020237028695A patent/KR20230130747A/ko not_active Ceased
- 2017-04-17 CN CN201780030129.9A patent/CN109153650A/zh active Pending
- 2017-04-17 PL PL17720921.0T patent/PL3442947T3/pl unknown
- 2017-04-17 AU AU2017250369A patent/AU2017250369A1/en not_active Abandoned
- 2017-04-17 TW TW106112816A patent/TWI751155B/zh not_active IP Right Cessation
- 2017-04-17 ES ES17720921T patent/ES2953512T3/es active Active
- 2017-04-17 EP EP17720921.0A patent/EP3442947B1/en active Active
- 2017-04-17 BR BR112018071093A patent/BR112018071093A2/pt active Search and Examination
- 2017-04-17 MA MA044666A patent/MA44666A/fr unknown
- 2017-04-17 JP JP2018553876A patent/JP7041070B2/ja not_active Expired - Fee Related
- 2017-04-17 SG SG11201808799SA patent/SG11201808799SA/en unknown
- 2017-04-17 DK DK17720921.0T patent/DK3442947T3/da active
- 2017-04-17 FI FIEP17720921.0T patent/FI3442947T3/fi active
- 2017-04-17 SI SI201731402T patent/SI3442947T1/sl unknown
- 2017-04-17 KR KR1020187032892A patent/KR102571679B1/ko active Active
- 2017-04-17 CA CA3021062A patent/CA3021062A1/en active Pending
- 2017-04-17 HU HUE17720921A patent/HUE064145T2/hu unknown
- 2017-05-22 US US15/601,888 patent/US20170355712A1/en not_active Abandoned
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2018
- 2018-10-04 IL IL262140A patent/IL262140A/en unknown
- 2018-10-12 CL CL2018002928A patent/CL2018002928A1/es unknown
- 2018-10-15 MX MX2022010947A patent/MX2022010947A/es unknown
- 2018-11-13 CO CONC2018/0012181A patent/CO2018012181A2/es unknown
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2019
- 2019-03-28 CL CL2019000815A patent/CL2019000815A1/es unknown
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2020
- 2020-11-20 US US17/100,489 patent/US20210198277A1/en not_active Abandoned
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2021
- 2021-10-07 AU AU2021245168A patent/AU2021245168B2/en not_active Ceased
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2022
- 2022-03-10 JP JP2022036728A patent/JP7420847B2/ja active Active
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2024
- 2024-01-11 JP JP2024002232A patent/JP2024045202A/ja active Pending
- 2024-01-25 AU AU2024200464A patent/AU2024200464A1/en not_active Abandoned