JP2010532774A5 - - Google Patents
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- JP2010532774A5 JP2010532774A5 JP2010515398A JP2010515398A JP2010532774A5 JP 2010532774 A5 JP2010532774 A5 JP 2010532774A5 JP 2010515398 A JP2010515398 A JP 2010515398A JP 2010515398 A JP2010515398 A JP 2010515398A JP 2010532774 A5 JP2010532774 A5 JP 2010532774A5
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- JP
- Japan
- Prior art keywords
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- head
- lymphocytic leukemia
- leukemia
- Prior art date
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- 206010028980 Neoplasm Diseases 0.000 claims description 5
- 208000024893 Acute lymphoblastic leukemia Diseases 0.000 claims description 2
- 208000014697 Acute lymphocytic leukaemia Diseases 0.000 claims description 2
- 208000031261 Acute myeloid leukaemia Diseases 0.000 claims description 2
- 208000010839 B-cell chronic lymphocytic leukemia Diseases 0.000 claims description 2
- 208000032791 BCR-ABL1 positive chronic myelogenous leukemia Diseases 0.000 claims description 2
- 208000010833 Chronic myeloid leukaemia Diseases 0.000 claims description 2
- 208000031422 Lymphocytic Chronic B-Cell Leukemia Diseases 0.000 claims description 2
- 208000033761 Myelogenous Chronic BCR-ABL Positive Leukemia Diseases 0.000 claims description 2
- 208000033776 Myeloid Acute Leukemia Diseases 0.000 claims description 2
- 208000006664 Precursor Cell Lymphoblastic Leukemia-Lymphoma Diseases 0.000 claims description 2
- 208000032852 chronic lymphocytic leukemia Diseases 0.000 claims description 2
- 210000003128 head Anatomy 0.000 claims 2
- 210000004556 brain Anatomy 0.000 claims 1
- 210000003679 cervix uteri Anatomy 0.000 claims 1
- 210000000981 epithelium Anatomy 0.000 claims 1
- 210000003238 esophagus Anatomy 0.000 claims 1
- 210000000936 intestine Anatomy 0.000 claims 1
- 210000003734 kidney Anatomy 0.000 claims 1
- 210000004185 liver Anatomy 0.000 claims 1
- 210000004072 lung Anatomy 0.000 claims 1
- 210000004324 lymphatic system Anatomy 0.000 claims 1
- 210000003739 neck Anatomy 0.000 claims 1
- 210000002307 prostate Anatomy 0.000 claims 1
- 210000002784 stomach Anatomy 0.000 claims 1
- 210000001685 thyroid gland Anatomy 0.000 claims 1
- 210000003932 urinary bladder Anatomy 0.000 claims 1
- 210000004369 blood Anatomy 0.000 description 1
- 239000008280 blood Substances 0.000 description 1
- 210000000987 immune system Anatomy 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102007032507.1 | 2007-07-12 | ||
| DE102007032507A DE102007032507A1 (de) | 2007-07-12 | 2007-07-12 | Pyridazinonderivate |
| EPPCT/EP2008/003473 | 2008-04-29 | ||
| PCT/EP2008/003473 WO2009006959A1 (de) | 2007-07-12 | 2008-04-29 | Pyridazinonderivate |
| PCT/EP2008/005508 WO2009007074A1 (de) | 2007-07-12 | 2008-07-04 | Pyrimidinyl-pyridazinonderivate |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010532774A JP2010532774A (ja) | 2010-10-14 |
| JP2010532774A5 true JP2010532774A5 (enExample) | 2011-08-18 |
| JP5426544B2 JP5426544B2 (ja) | 2014-02-26 |
Family
ID=39638671
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010515355A Active JP5426543B2 (ja) | 2007-07-12 | 2008-04-29 | ピリダジノン誘導体 |
| JP2010515398A Active JP5426544B2 (ja) | 2007-07-12 | 2008-07-04 | ピリミジニル−ピリダジノン誘導体 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010515355A Active JP5426543B2 (ja) | 2007-07-12 | 2008-04-29 | ピリダジノン誘導体 |
Country Status (36)
Families Citing this family (79)
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| DE102007026341A1 (de) | 2007-06-06 | 2008-12-11 | Merck Patent Gmbh | Benzoxazolonderivate |
| DE102007032507A1 (de) | 2007-07-12 | 2009-04-02 | Merck Patent Gmbh | Pyridazinonderivate |
| DE102007038957A1 (de) * | 2007-08-17 | 2009-02-19 | Merck Patent Gmbh | 6-Thioxo-pyridazinderivate |
| DE102007041115A1 (de) * | 2007-08-30 | 2009-03-05 | Merck Patent Gmbh | Thiadiazinonderivate |
| DE102007061963A1 (de) | 2007-12-21 | 2009-06-25 | Merck Patent Gmbh | Pyridazinonderivate |
| DE102008019907A1 (de) * | 2008-04-21 | 2009-10-22 | Merck Patent Gmbh | Pyridazinonderivate |
| DE102008028905A1 (de) * | 2008-06-18 | 2009-12-24 | Merck Patent Gmbh | 3-(3-Pyrimidin-2-yl-benzyl)-[1,2,4]triazolo[4,3-b]pyridazinderivate |
| DE102008037790A1 (de) * | 2008-08-14 | 2010-02-18 | Merck Patent Gmbh | Bicyclische Triazolderivate |
| US8586599B2 (en) * | 2008-12-22 | 2013-11-19 | Merck Patent Gmbh | Polymorphic forms of 6-(1-methyl-1H-pyrazol-4-yl)-2-{3-[5-(2-morpholin-4-yl-ethoxy)-pyrimidin-2-yl]-benzyl}-2H-pyridazin-3-one dihydrogenphosphate and processes of manufacturing thereof |
| DE102008062826A1 (de) * | 2008-12-23 | 2010-07-01 | Merck Patent Gmbh | Pyridazinonderivate |
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| SI2373640T1 (sl) * | 2009-01-08 | 2014-11-28 | Merck Patent Gmbh | Nove polimorfne oblike hidrokloridne soli 3-(1-(3-(5-(1-metil-piperidin-4ilmetoksi)-pirimidin-2-il)-benzil)-6- okso-1,6-dihidro-piridazin-3-il)-benzonitrila in postopki proizvodnje le-teh |
| EP2221053A1 (de) * | 2009-02-20 | 2010-08-25 | Albert-Ludwigs-Universität Freiburg | Pharmazeutische Zusammensetzung enthaltend Hemmstoffe der Proteinmethyltransferase I und deren Verwendung zur Behandlung von Tumorerkrankungen |
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