DE3508258A1
(de)
|
1985-03-08 |
1986-09-18 |
Bayer Ag, 5090 Leverkusen |
Ss-lactamantibiotika, verfahren zur herstellung und ihre verwendung als und in arzneimitteln
|
FR2643903A1
(fr)
|
1989-03-03 |
1990-09-07 |
Union Pharma Scient Appl |
Nouveaux derives de benzimidazole, leurs procedes de preparation, intermediaires de synthese, compositions pharmaceutiques les contenant, utiles notamment pour le traitement des maladies cardiovasculaires, et des ulceres duodenaux
|
RU1836357C
(ru)
|
1990-07-23 |
1993-08-23 |
Др.Карл Томэ ГмбХ |
Производные бензимидазола, их изомеры, смеси изомеров, гидраты или их физиологически переносимые соли, обладающие антагонистическими в отношении ангиотензина свойствами
|
DE4023369A1
(de)
|
1990-07-23 |
1992-01-30 |
Thomae Gmbh Dr K |
Benzimidazole, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung
|
US5591762A
(en)
|
1991-02-06 |
1997-01-07 |
Dr. Karl Thomae Gmbh |
Benzimidazoles useful as angiotensin-11 antagonists
|
DE4225756A1
(de)
|
1992-01-22 |
1994-03-10 |
Thomae Gmbh Dr K |
Benzimidazole, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
|
DE4224752A1
(de)
|
1992-04-11 |
1994-02-03 |
Thomae Gmbh Dr K |
Benzimidazole, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
|
SI9210098B
(sl)
|
1991-02-06 |
2000-06-30 |
Dr. Karl Thomae |
Benzimidazoli, zdravila, ki te spojine vsebujejo, in postopek za njihovo pripravo
|
US5125961A
(en)
|
1991-08-12 |
1992-06-30 |
Monsanto Company |
Substituted pyridine compounds
|
DE4219534A1
(de)
|
1992-02-19 |
1993-12-16 |
Thomae Gmbh Dr K |
Substituierte Biphenylylderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
|
DE4408497A1
(de)
|
1994-03-14 |
1995-09-21 |
Thomae Gmbh Dr K |
Benzimidazole, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
|
AU699272B2
(en)
|
1994-08-02 |
1998-11-26 |
Merck Sharp & Dohme Limited |
Azetidine, pyrrolidine and piperidine derivatives
|
PL183853B1
(pl)
|
1995-04-21 |
2002-07-31 |
Neurosearch As |
Nowa pochodna benzimidazolu i środek farmaceutyczny
|
JP2000072675A
(ja)
|
1998-08-26 |
2000-03-07 |
Tanabe Seiyaku Co Ltd |
医薬組成物
|
CN1177831C
(zh)
|
1998-12-04 |
2004-12-01 |
神经研究公司 |
作为离子通道调节剂的新的苯并咪唑啉酮一、苯并噁唑酮一或苯并噻唑啉酮衍生物
|
US6380235B1
(en)
|
1999-05-04 |
2002-04-30 |
American Home Products Corporation |
Benzimidazolones and analogues
|
US6664252B2
(en)
|
1999-12-02 |
2003-12-16 |
Osi Pharmaceuticals, Inc. |
4-aminopyrrolo[2,3-d]pyrimidine compounds specific to adenosine A2a receptor and uses thereof
|
GB0002100D0
(en)
|
2000-01-28 |
2000-03-22 |
Novartis Ag |
Organic compounds
|
WO2001057019A1
(en)
|
2000-02-01 |
2001-08-09 |
Cor Therapeutics, Inc. |
INDALONE AND BENZIMIDAZOLONE INHIBITORS OF FACTOR Xa
|
US20120028912A1
(en)
|
2000-02-22 |
2012-02-02 |
J.David Gladstone Institute |
Methods of modulating bromodomains
|
CN1474652A
(zh)
|
2000-10-27 |
2004-02-11 |
�ݶ�ũ������˾ |
取代的4,5-二氢-1,2,4-三嗪-6-酮、1,2,4-三嗪-6-酮以及它们作为杀真菌剂和杀虫剂的应用
|
YU42703A
(sh)
|
2000-12-01 |
2006-03-03 |
Osi Pharmaceuticals Inc. |
Jedinjenja specifična za dobijanje adenozinske a1,a2a i a3 receptore i njihove primene
|
US7148237B2
(en)
|
2001-03-01 |
2006-12-12 |
Shionogi & Co., Ltd. |
Nitrogen-containing heteroaryl compounds having HIV integrase inhibitory activity
|
CA2440211A1
(en)
|
2001-03-09 |
2002-09-19 |
Pfizer Products Inc. |
Benzimidazole anti-inflammatory compounds
|
ATE367814T1
(de)
|
2001-03-15 |
2007-08-15 |
Janssen Pharmaceutica Nv |
Hiv hemmende pyrazinon-derivate
|
MXPA03008658A
(es)
|
2001-03-23 |
2005-04-11 |
Bayer Ag |
Inhibidores de rho-cinasa.
|
CZ20032615A3
(en)
|
2001-03-28 |
2004-03-17 |
Bristol-Myers Squibb Company |
Novel tyrosine kinase inhibitors
|
US7081454B2
(en)
|
2001-03-28 |
2006-07-25 |
Bristol-Myers Squibb Co. |
Tyrosine kinase inhibitors
|
WO2003068857A1
(fr)
|
2002-02-15 |
2003-08-21 |
Bridgestone Corporation |
Composition de caoutchouc et pneumatique produit a partir de ladite composition
|
TWI276631B
(en)
|
2002-09-12 |
2007-03-21 |
Avanir Pharmaceuticals |
Phenyl-aza-benzimidazole compounds for modulating IgE and inhibiting cellular proliferation
|
US20040166137A1
(en)
|
2002-11-08 |
2004-08-26 |
Lackey John William |
Hetero-substituted benzimidazole compounds and antiviral uses thereof
|
AR043063A1
(es)
|
2002-12-13 |
2005-07-13 |
Altana Pharma Ag |
Bencimidazoles 6-sustituidos y su uso como inhibidores de secreciones gastricas
|
AR042956A1
(es)
|
2003-01-31 |
2005-07-13 |
Vertex Pharma |
Inhibidores de girasa y usos de los mismos
|
CL2004000409A1
(es)
|
2003-03-03 |
2005-01-07 |
Vertex Pharma |
Compuestos derivados de 2-(cilo sustituido)-1-(amino u oxi sustituido)-quinazolina, inhibidores de canales ionicos de sodio y calcio dependientes de voltaje; composicion farmaceutica; y uso del compuesto en el tratamiento de dolor agudo, cronico, neu
|
BRPI0409695B1
(pt)
|
2003-04-25 |
2015-08-04 |
3M Innovative Properties Co |
Método para fabricar um artigo abrasivo
|
AU2003902860A0
(en)
|
2003-06-06 |
2003-06-26 |
Daicel Chemical Industries, Ltd |
Benzimidazole compounds
|
AU2004263190A1
(en)
|
2003-08-08 |
2005-02-17 |
Avanir Pharmaceuticals |
Selective pharmacologic inhibition of protein trafficking and related methods of treating human diseases
|
NL1026826C2
(nl)
|
2003-08-13 |
2007-01-04 |
Pharmacia Corp |
Gesubstitueerde pyridinonen.
|
US8094804B2
(en)
|
2003-09-26 |
2012-01-10 |
Avaya Inc. |
Method and apparatus for assessing the status of work waiting for service
|
WO2005080380A1
(en)
|
2004-02-03 |
2005-09-01 |
Eli Lilly And Company |
Kinase inhibitors
|
WO2005075432A1
(ja)
|
2004-02-06 |
2005-08-18 |
Chugai Seiyaku Kabushiki Kaisha |
1−(2h)−イソキノロン誘導体およびその抗ガン剤としての使用
|
CA2559552A1
(en)
|
2004-03-23 |
2005-09-29 |
F. Hoffmann-La Roche Ag |
Benzyl-pyridazinone derivatives as non-nucleoside reverse transcriptase inhibitors
|
EP1734820A4
(en)
|
2004-04-16 |
2008-01-23 |
Neurogen Corp |
Imidazopyrrazine, imidazopyridine, and imidazo-pyrimidine as CRF1 receptor ligands
|
NZ551775A
(en)
|
2004-06-01 |
2010-12-24 |
Univ Virginia |
Dual small molecule inhibitors of cancer and angiogenesis
|
WO2005121132A1
(ja)
|
2004-06-11 |
2005-12-22 |
Shionogi & Co., Ltd. |
抗hcv作用を有する縮合ヘテロ環化合物
|
CA2578075A1
(en)
|
2004-08-26 |
2006-03-02 |
Pfizer Inc. |
Aminoheteroaryl compounds as protein tyrosine kinase inhibitors
|
GB0420719D0
(en)
|
2004-09-17 |
2004-10-20 |
Addex Pharmaceuticals Sa |
Novel allosteric modulators
|
GB0420722D0
(en)
|
2004-09-17 |
2004-10-20 |
Addex Pharmaceuticals Sa |
Novel allosteric modulators
|
WO2006038734A1
(en)
|
2004-10-08 |
2006-04-13 |
Astellas Pharma Inc. |
Pyridazinone derivatives cytokines inhibitors
|
SG156641A1
(en)
|
2004-10-13 |
2009-11-26 |
Ptc Therapeutics Inc |
Compounds for nonsense suppression, and methods for their use
|
WO2006045010A2
(en)
|
2004-10-20 |
2006-04-27 |
Resverlogix Corp. |
Stilbenes and chalcones for the prevention and treatment of cardiovascular diseases
|
CA2587195A1
(en)
|
2004-11-22 |
2006-07-13 |
Merck & Co., Inc. |
Cycloalkyl keto piperidine tachykinin receptor antagonists
|
AU2006210422B2
(en)
|
2005-02-04 |
2012-09-13 |
Takeda Pharmaceutical Company Limited |
Inhibitors of E1 activating enzymes
|
MX2007011234A
(es)
|
2005-03-14 |
2007-11-12 |
Transtech Pharma Inc |
Derivados de benzazol, composiciones y metodos de uso en la forma de inhibidores de b-secretasa.
|
US7473669B2
(en)
|
2005-05-03 |
2009-01-06 |
Dow Agrosciences Llc |
Substituted 4,5-dihydro-1,2,4-triazin-6-ones, 1,2,4-triazin-6-ones, and their use as fungicides
|
EP2314295B1
(en)
|
2005-07-29 |
2015-01-28 |
Resverlogix, Inc |
Pharmaceutical compositions for the prevention and treatment of complex diseases and their delivery by insertable medical devices
|
WO2007040208A1
(ja)
|
2005-10-03 |
2007-04-12 |
Ono Pharmaceutical Co., Ltd. |
含窒素複素環化合物およびその医薬用途
|
JP2009515997A
(ja)
|
2005-11-18 |
2009-04-16 |
タケダ サン ディエゴ インコーポレイテッド |
グルコキナーゼ活性剤
|
RU2396269C2
(ru)
|
2005-12-01 |
2010-08-10 |
Ф.Хоффманн-Ля Рош Аг |
Производные гетероарилзамещенного пиперидина в качестве ингибиторов печеночной карнитин пальмитоилтрансферазы (l-cpt1)
|
ES2374455T3
(es)
|
2006-02-17 |
2012-02-16 |
Pfizer Limited |
Derivados de 3-deazapurinza como moduladores de tlr7.
|
CN101384593A
(zh)
|
2006-02-17 |
2009-03-11 |
辉瑞有限公司 |
用作tlr7调节剂的3-脱氮嘌呤衍生物
|
MX2008012875A
(es)
|
2006-04-03 |
2008-10-13 |
Glaxo Group Ltd |
Derivados de azabiciclo [3.1.0] hexilo como moduladores de los receptores d3 de la dopamina.
|
WO2008054599A2
(en)
|
2006-09-27 |
2008-05-08 |
Surface Logix, Inc. |
Rho kinase inhibitors
|
MX2009006312A
(es)
|
2006-12-14 |
2009-08-07 |
Astellas Pharma Inc |
Compuestos de acido policiclico utiles como antagonistas crth2 y agentes antialergicos.
|
SG144809A1
(en)
|
2007-01-11 |
2008-08-28 |
Millipore U K Ltd |
Benzimidazole compounds and their use as chromatographic ligands
|
PL2118074T3
(pl)
|
2007-02-01 |
2014-06-30 |
Resverlogix Corp |
Związki chemiczne do celów profilaktyki i leczenia chorób układu sercowo-naczyniowego
|
WO2008153701A1
(en)
|
2007-05-24 |
2008-12-18 |
Schering Corporation |
Compounds for inhibiting ksp kinesin activity
|
KR20100023907A
(ko)
|
2007-06-26 |
2010-03-04 |
사노피-아벤티스 |
벤즈이미다졸 및 아자벤즈이미다졸의 위치선택적 구리 촉매화 합성
|
DE102007032507A1
(de)
|
2007-07-12 |
2009-04-02 |
Merck Patent Gmbh |
Pyridazinonderivate
|
DE102007038957A1
(de)
|
2007-08-17 |
2009-02-19 |
Merck Patent Gmbh |
6-Thioxo-pyridazinderivate
|
GB0719235D0
(en)
|
2007-10-02 |
2007-11-14 |
Glaxo Group Ltd |
Novel compounds
|
WO2009054790A1
(en)
|
2007-10-26 |
2009-04-30 |
Astrazeneca Ab |
Amide linked heteroaromatic derivatives as modulators of mglur5
|
US8084466B2
(en)
|
2007-12-18 |
2011-12-27 |
Janssen Pharmaceutica Nv |
Bicyclic heteroaryl-substituted imidazoles as modulators of the histamine H4 receptor
|
EP2239264A4
(en)
|
2007-12-28 |
2012-01-11 |
Mitsubishi Tanabe Pharma Corp |
ANTITUMOR AGENT
|
TW200942537A
(en)
|
2008-02-01 |
2009-10-16 |
Irm Llc |
Compounds and compositions as kinase inhibitors
|
WO2009158258A1
(en)
|
2008-06-25 |
2009-12-30 |
E. I. Du Pont De Nemours And Company |
Herbicidal dihydro oxo six-membered azinyl isoxazolines
|
US9540322B2
(en)
|
2008-08-18 |
2017-01-10 |
Yale University |
MIF modulators
|
KR20110042374A
(ko)
|
2008-08-18 |
2011-04-26 |
예일 유니버시티 |
Mif 조정인자
|
US9643922B2
(en)
|
2008-08-18 |
2017-05-09 |
Yale University |
MIF modulators
|
EP3037421A3
(en)
|
2008-11-25 |
2016-11-30 |
University Of Rochester |
Mlk inhibitors and methods of use
|
PT2370413E
(pt)
|
2008-12-08 |
2015-10-23 |
Arena Pharm Inc |
Moduladores do recetor da prostaciclina (pgi2) úteis para o tratamento de distúrbios relacionados com o mesmo
|
EP2196465A1
(en)
|
2008-12-15 |
2010-06-16 |
Almirall, S.A. |
(3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors
|
DE102008062826A1
(de)
|
2008-12-23 |
2010-07-01 |
Merck Patent Gmbh |
Pyridazinonderivate
|
US8389550B2
(en)
|
2009-02-25 |
2013-03-05 |
Hoffmann-La Roche Inc. |
Isoxazoles / O-pyridines with ethyl and ethenyl linker
|
CA2755095A1
(en)
|
2009-03-09 |
2010-09-16 |
Surface Logix, Inc. |
Rho kinase inhibitors
|
JP2012520884A
(ja)
|
2009-03-18 |
2012-09-10 |
ザ ボード オブ トラスティーズ オブ ザ リランド スタンフォード ジュニア ユニバーシティー |
フラビウイルス科ウイルス感染症を治療する方法および組成物
|
AU2010224523B2
(en)
|
2009-03-18 |
2014-05-08 |
Resverlogix Corp. |
Novel anti-inflammatory agents
|
LT2421533T
(lt)
|
2009-04-22 |
2018-12-27 |
Resverlogix Corp. |
Nauji priešuždegiminiai agentai
|
JP5466292B2
(ja)
|
2009-05-05 |
2014-04-09 |
エフ.ホフマン−ラ ロシュ アーゲー |
イソオキサゾール−ピリジン誘導体
|
GB0919431D0
(en)
|
2009-11-05 |
2009-12-23 |
Glaxosmithkline Llc |
Novel compounds
|
GB0919423D0
(en)
|
2009-11-05 |
2009-12-23 |
Glaxosmithkline Llc |
Novel compounds
|
GB0919434D0
(en)
|
2009-11-05 |
2009-12-23 |
Glaxosmithkline Llc |
Novel compounds
|
GB0919432D0
(en)
|
2009-11-05 |
2009-12-23 |
Glaxosmithkline Llc |
Use
|
CA2779355C
(en)
|
2009-11-05 |
2018-01-16 |
Glaxosmithkline Llc |
Benzodiazepine bromodomain inhibitor
|
SI2496582T1
(sl)
|
2009-11-05 |
2016-04-29 |
Glaxosmithkline Llc Corporation Service Company |
Benzodiazepinski inhibitor bromodomene
|
ES2549502T3
(es)
|
2009-11-20 |
2015-10-28 |
Sk Chemicals Co., Ltd. |
Antagonistas de receptores de gonadoliberina, método de fabricación de los mismos, y composición farmacéutica que los contienen
|
US20130085133A1
(en)
|
2010-02-08 |
2013-04-04 |
Sourthern Research Institute Office of Commercialization and Intellectual Prop. |
Anti-viral treatment and assay to screenfor anti-viral agent
|
KR101165996B1
(ko)
|
2010-04-23 |
2012-07-18 |
주식회사 녹십자 |
프탈라지논 유도체, 이의 제조방법 및 이를 함유하는 약학적 조성물
|
MX362384B
(es)
|
2010-05-14 |
2019-01-15 |
Dana Farber Cancer Inst Inc |
Composiciones y metodos para tratar neoplasias, enfermedades inflamatorias y otros trastornos.
|
US8933096B2
(en)
|
2010-06-09 |
2015-01-13 |
Rugers, The State University of New Jersey |
Antimicrobial agents
|
WO2011159926A1
(en)
|
2010-06-16 |
2011-12-22 |
Rutgers, The State University Of New Jersey |
Antimicrobial agents
|
US20130165426A1
(en)
|
2010-07-06 |
2013-06-27 |
Université de Montréal |
Imidazopyridine, imidazopyrimidine and imidazopyrazine derivatives as melanocortin-4 receptor modulators
|
WO2012009258A2
(en)
|
2010-07-13 |
2012-01-19 |
Edward Roberts |
Peptidomimetic galanin receptor modulators
|
WO2012021382A1
(en)
|
2010-08-12 |
2012-02-16 |
Merck Sharp & Dohme Corp. |
Positive allosteric modulators of mglur2
|
WO2012040499A2
(en)
|
2010-09-22 |
2012-03-29 |
Surface Logix, Inc. |
Metabolic inhibitors
|
KR101242572B1
(ko)
|
2010-10-12 |
2013-03-19 |
한국화학연구원 |
5-환 헤테로 아릴로 치환된 프탈라지논 유도체 또는 이의 약학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 포함하는 약학적 조성물
|
AR084070A1
(es)
|
2010-12-02 |
2013-04-17 |
Constellation Pharmaceuticals Inc |
Inhibidores del bromodominio y usos de los mismos
|
US9249161B2
(en)
|
2010-12-02 |
2016-02-02 |
Constellation Pharmaceuticals, Inc. |
Bromodomain inhibitors and uses thereof
|
CN102731409A
(zh)
|
2011-04-08 |
2012-10-17 |
中国科学院上海药物研究所 |
一类哒嗪酮类化合物,其药物组合物、制备方法及用途
|
GB201106743D0
(en)
|
2011-04-21 |
2011-06-01 |
Glaxosmithkline Llc |
Novel compounds
|
GB201106750D0
(en)
|
2011-04-21 |
2011-06-01 |
Glaxosmithkline Llc |
Novel compounds
|
GB201106799D0
(en)
|
2011-04-21 |
2011-06-01 |
Glaxosmithkline Llc |
Novel compounds
|
EP2721031B1
(en)
|
2011-06-17 |
2016-01-20 |
Constellation Pharmaceuticals, Inc. |
Bromodomain inhibitors and uses thereof
|
GB201114103D0
(en)
|
2011-08-17 |
2011-09-28 |
Glaxosmithkline Llc |
Novel compounds
|
WO2013027168A1
(en)
|
2011-08-22 |
2013-02-28 |
Pfizer Inc. |
Novel heterocyclic compounds as bromodomain inhibitors
|
US9610251B2
(en)
|
2011-11-01 |
2017-04-04 |
Resverlogix Corp. |
Pharmaceutical compositions for substituted quinazolinones
|
US8317624B1
(en)
|
2011-11-07 |
2012-11-27 |
TwoChop Inc. |
System and method for creating and/or serving online games embedded in websites
|
EP2785710B1
(en)
|
2011-12-01 |
2017-09-20 |
ChemoCentryx, Inc. |
Substituted benzimidazoles and benzopyrazoles as ccr(4) antagonists
|
US20130281397A1
(en)
|
2012-04-19 |
2013-10-24 |
Rvx Therapeutics Inc. |
Treatment of diseases by epigenetic regulation
|
US20130281399A1
(en)
|
2012-04-19 |
2013-10-24 |
Rvx Therapeutics Inc. |
Treatment of diseases by epigenetic regulation
|
US20130281396A1
(en)
|
2012-04-19 |
2013-10-24 |
Rvx Therapeutics Inc. |
Treatment of diseases by epigenetic regulation
|
US20130281398A1
(en)
|
2012-04-19 |
2013-10-24 |
Rvx Therapeutics Inc. |
Treatment of diseases by epigenetic regulation
|
CA2870931A1
(en)
|
2012-04-20 |
2013-10-24 |
Abbvie Inc. |
Isoindolone derivatives
|
EP2864336B1
(en)
|
2012-06-06 |
2016-11-23 |
Constellation Pharmaceuticals, Inc. |
Benzo[b]isoxazoloazepine bromodomain inhibitors and uses thereof
|
EP2858983B1
(en)
|
2012-06-11 |
2018-04-18 |
UCB Biopharma SPRL |
Tnf-alpha modulating benzimidazoles
|
US20140073634A1
(en)
|
2012-08-24 |
2014-03-13 |
Institute For Applied Cancer Science/The University of Texas MD Anderson Cancer Center |
Heterocyclic modulators of hif activity for treatment of disease
|
AU2013311826A1
(en)
|
2012-09-05 |
2015-03-26 |
Bayer Cropscience Ag |
Use of substituted 2-amidobenzimidazoles, 2-amidobenzoxazoles and 2-amidobenzothiazoles or salts thereof as active substances against abiotic plant stress
|
US20150246888A1
(en)
|
2012-09-11 |
2015-09-03 |
Michael Johnson |
Enoyl reductase inhibitors with antibacterial activity
|
US9663533B2
(en)
|
2012-11-14 |
2017-05-30 |
Glaxosmithkline Llc |
Thieno[3,2-C]pyridin-4(5H)-ones as BET inhibitors
|
WO2014080291A2
(en)
|
2012-11-21 |
2014-05-30 |
Rvx Therapeutics Inc. |
Biaryl derivatives as bromodomain inhibitors
|
WO2014080290A2
(en)
|
2012-11-21 |
2014-05-30 |
Rvx Therapeutics Inc. |
Cyclic amines as bromodomain inhibitors
|
WO2014095775A1
(de)
|
2012-12-20 |
2014-06-26 |
Bayer Pharma Aktiengesellschaft |
Bet-proteininhibitorische dihydrochinoxalinone
|
CN105073744B
(zh)
|
2012-12-21 |
2019-11-08 |
齐尼思表观遗传学有限公司 |
作为溴结构域抑制剂的新型杂环化合物
|
EP2958923A1
(de)
|
2013-02-22 |
2015-12-30 |
Bayer Pharma Aktiengesellschaft |
4-substituierte pyrrolo- und pyrazolo-diazepine
|
EP2958922A1
(de)
|
2013-02-22 |
2015-12-30 |
Bayer Pharma Aktiengesellschaft |
Pyrrolo- und pyrazolo-triazolodiazepine als bet-proteininhibitoren zur behandlung von hyper-proliferativen erkrankungen
|
WO2014128655A1
(en)
|
2013-02-25 |
2014-08-28 |
Aurigene Discovery Technologies Limited |
Substituted imidazo[4,5-c]quinoline derivatives as bromodomain inhibitors
|
US9492460B2
(en)
|
2013-02-27 |
2016-11-15 |
Bristol-Myers Squibb Company |
Carbazole compounds useful as bromodomain inhibitors
|
CN105189488B
(zh)
|
2013-02-27 |
2018-07-24 |
百时美施贵宝公司 |
用作溴区结构域抑制剂的咔唑化合物
|
US9675697B2
(en)
|
2013-03-11 |
2017-06-13 |
The Regents Of The University Of Michigan |
BET bromodomain inhibitors and therapeutic methods using the same
|
US8980879B2
(en)
|
2013-03-11 |
2015-03-17 |
Abbvie Inc. |
Bromodomain inhibitors
|
MX2015012005A
(es)
|
2013-03-11 |
2016-04-04 |
Abbvie Inc |
Inhibidores de bromodominio.
|
EP2970276A1
(en)
|
2013-03-12 |
2016-01-20 |
AbbVie Inc. |
Dihydro-pyrrolopyridinone bromodomain inhibitors
|
BR112015022551A2
(pt)
|
2013-03-12 |
2017-07-18 |
Abbvie Inc |
inibidores de amido pirrol
|
KR101780784B1
(ko)
|
2013-03-14 |
2017-09-21 |
글락소스미스클라인 인털렉츄얼 프로퍼티 (넘버 2) 리미티드 |
2,3-이치환된 1-아실-4-아미노-1,2,3,4-테트라하이드로퀴놀린 유도체 및 이의 브로모도메인 억제제로서의 용도
|
KR20150135359A
(ko)
|
2013-03-14 |
2015-12-02 |
컨버진 엘엘씨 |
브로모도메인-함유 단백질의 억제를 위한 방법 및 조성물
|
ES2654362T3
(es)
|
2013-03-14 |
2018-02-13 |
Glaxosmithkline Intellectual Property (No. 2) Limited |
Furopiridinas como inhibidores de bromodominio
|
EP2968311A4
(en)
|
2013-03-15 |
2016-07-20 |
Epigenetix Inc |
OXAZOLO [5,4-C] CHINOLIN-2-ON COMPOUNDS AS BROMODOMENA INHIBITORS
|
RS57733B1
(sr)
|
2013-03-15 |
2018-12-31 |
Plexxikon Inc |
Heterociklična jedinjenja i njihove upotrebe
|
EP3581576B1
(en)
|
2013-03-15 |
2022-01-26 |
Incyte Holdings Corporation |
Tricyclic heterocycles as bet protein inhibitors for use in the treatment of a proliferative disease in combination with a janus kinase inhibitor
|
US20140303121A1
(en)
|
2013-03-15 |
2014-10-09 |
Plexxikon Inc. |
Heterocyclic compounds and uses thereof
|
US9102684B2
(en)
|
2013-03-27 |
2015-08-11 |
Boehringer Ingelheim International Gmbh |
Indolinone analogues
|
US9199988B2
(en)
|
2013-03-27 |
2015-12-01 |
Boehringer Ingelheim International Gmbh |
Dihydroquinazolinone analogues
|
TWI530499B
(zh)
|
2013-03-28 |
2016-04-21 |
吉李德科學股份有限公司 |
作為溴結構域(bromodomain)抑制劑之苯並咪唑酮衍生物類
|
EP2792355A1
(en)
|
2013-04-17 |
2014-10-22 |
Albert-Ludwigs-Universität Freiburg |
Compounds for use as bromodomain inhibitors
|
EP2996689A1
(en)
|
2013-04-17 |
2016-03-23 |
Albert-Ludwigs-Universität Freiburg |
Compounds for use as bromodomain inhibitors
|
JP6388915B2
(ja)
|
2013-04-26 |
2018-09-12 |
ベイジーン,リミテッド |
置換5−(3,5−ジメチルイソオキサゾール−4−イル)インドリン−2−オン
|
TWI527811B
(zh)
|
2013-05-09 |
2016-04-01 |
吉李德科學股份有限公司 |
作爲溴結構域抑制劑的苯並咪唑衍生物
|
JP6373978B2
(ja)
|
2013-05-27 |
2018-08-15 |
ノバルティス アーゲー |
イミダゾピロリジノン誘導体および疾患の処置におけるその使用
|
US8975417B2
(en)
|
2013-05-27 |
2015-03-10 |
Novartis Ag |
Pyrazolopyrrolidine derivatives and their use in the treatment of disease
|
WO2014202578A1
(de)
|
2013-06-17 |
2014-12-24 |
Bayer Pharma Aktiengesellschaft |
Substituierte phenyl-2,3-benzodiazepine
|
PT3010503T
(pt)
|
2013-06-21 |
2020-06-16 |
Zenith Epigenetics Corp |
Novos inibidores bicíclicos de bromodomínios
|
WO2015004534A2
(en)
|
2013-06-21 |
2015-01-15 |
Zenith Epigenetics Corp. |
Novel substituted bicyclic compounds as bromodomain inhibitors
|
AR096758A1
(es)
|
2013-06-28 |
2016-02-03 |
Abbvie Inc |
Inhibidores cristalinos de bromodominios
|
JP2016523964A
(ja)
|
2013-07-08 |
2016-08-12 |
インサイト・ホールディングス・コーポレイションIncyte Holdings Corporation |
Betタンパク質阻害剤としての三環式複素環
|
CA2918813A1
(en)
|
2013-07-23 |
2015-01-29 |
Bayer Pharma Aktiengesellschaft |
Substituted dihydropyrido[3,4-b]pyrazinones as dual inhibitors of bet proteins and polo-like kinases
|
CN105611835A
(zh)
|
2013-07-25 |
2016-05-25 |
达纳-法伯癌症研究所股份有限公司 |
转录因子抑制剂及其用途
|
US9855271B2
(en)
|
2013-07-31 |
2018-01-02 |
Zenith Epigenetics Ltd. |
Quinazolinones as bromodomain inhibitors
|
US20150051208A1
(en)
|
2013-08-14 |
2015-02-19 |
Boehringer Ingelheim International Gmbh |
Pyridinones
|
US9422281B2
(en)
|
2013-11-18 |
2016-08-23 |
Forma Therapeutics, Inc. |
Benzopiperazine compositions as BET bromodomain inhibitors
|
LT3071203T
(lt)
|
2013-11-18 |
2021-05-25 |
Forma Therapeutics, Inc. |
Tetrahidrochinolino kompozicijos kaip bet bromodomeno inhibitoriai
|
GB201321739D0
(en)
|
2013-12-09 |
2014-01-22 |
Ucb Pharma Sa |
Therapeutic agents
|
US9458156B2
(en)
|
2014-12-23 |
2016-10-04 |
Bristol-Myers Squibb Company |
Tricyclic compounds as anticancer agents
|
WO2016087936A1
(en)
|
2014-12-01 |
2016-06-09 |
Zenith Epigenetics Corp. |
Substituted pyridinones as bromodomain inhibitors
|
WO2016087942A1
(en)
|
2014-12-01 |
2016-06-09 |
Zenith Epigenetics Corp. |
Substituted pyridines as bromodomain inhibitors
|
US10292968B2
(en)
|
2014-12-11 |
2019-05-21 |
Zenith Epigenetics Ltd. |
Substituted heterocycles as bromodomain inhibitors
|
CN107406438B
(zh)
|
2014-12-17 |
2021-05-14 |
恒翼生物医药科技(上海)有限公司 |
溴结构域的抑制剂
|
CA2966452A1
(en)
|
2014-12-17 |
2016-06-23 |
Samuel David Brown |
Substituted bicyclic compounds as bromodomain inhibitors
|