JP2008510828A5 - - Google Patents

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Publication number
JP2008510828A5
JP2008510828A5 JP2007530127A JP2007530127A JP2008510828A5 JP 2008510828 A5 JP2008510828 A5 JP 2008510828A5 JP 2007530127 A JP2007530127 A JP 2007530127A JP 2007530127 A JP2007530127 A JP 2007530127A JP 2008510828 A5 JP2008510828 A5 JP 2008510828A5
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JP
Japan
Prior art keywords
compound according
compound
group
methyl
cyclopropyl
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JP2007530127A
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English (en)
Japanese (ja)
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JP4952943B2 (ja
JP2008510828A (ja
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Priority claimed from PCT/US2005/030259 external-priority patent/WO2006026356A2/en
Publication of JP2008510828A publication Critical patent/JP2008510828A/ja
Publication of JP2008510828A5 publication Critical patent/JP2008510828A5/ja
Application granted granted Critical
Publication of JP4952943B2 publication Critical patent/JP4952943B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2007530127A 2004-08-25 2005-08-25 HIV逆転写酵素のインヒビターとしてのS−トリアゾリルα−メルカプトアセトアニリド Expired - Lifetime JP4952943B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US60422004P 2004-08-25 2004-08-25
US60421904P 2004-08-25 2004-08-25
US60/604,219 2004-08-25
US60/604,220 2004-08-25
US68635105P 2005-05-31 2005-05-31
US60/686,351 2005-05-31
PCT/US2005/030259 WO2006026356A2 (en) 2004-08-25 2005-08-25 S-TRIAZOLYL α-MERCAPTOACETANILDES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2012000790A Division JP5457472B2 (ja) 2004-08-25 2012-01-05 HIV逆転写酵素のインヒビターとしてのS−トリアゾリルα−メルカプトアセトアニリド

Publications (3)

Publication Number Publication Date
JP2008510828A JP2008510828A (ja) 2008-04-10
JP2008510828A5 true JP2008510828A5 (enExample) 2008-07-17
JP4952943B2 JP4952943B2 (ja) 2012-06-13

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ID=36000576

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2007530127A Expired - Lifetime JP4952943B2 (ja) 2004-08-25 2005-08-25 HIV逆転写酵素のインヒビターとしてのS−トリアゾリルα−メルカプトアセトアニリド
JP2012000790A Expired - Lifetime JP5457472B2 (ja) 2004-08-25 2012-01-05 HIV逆転写酵素のインヒビターとしてのS−トリアゾリルα−メルカプトアセトアニリド

Family Applications After (1)

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JP2012000790A Expired - Lifetime JP5457472B2 (ja) 2004-08-25 2012-01-05 HIV逆転写酵素のインヒビターとしてのS−トリアゾリルα−メルカプトアセトアニリド

Country Status (31)

Country Link
US (8) US7947721B2 (enExample)
EP (5) EP2433633A1 (enExample)
JP (2) JP4952943B2 (enExample)
KR (1) KR101241716B1 (enExample)
CN (2) CN101817793B (enExample)
AT (2) ATE528001T1 (enExample)
AU (2) AU2005280130C9 (enExample)
BR (2) BRPI0514630B8 (enExample)
CA (1) CA2578068C (enExample)
CY (2) CY1112221T1 (enExample)
DK (1) DK2135608T3 (enExample)
EA (2) EA014737B1 (enExample)
EC (1) ECSP077322A (enExample)
ES (2) ES2380604T3 (enExample)
FR (1) FR16C0031I2 (enExample)
HR (1) HRP20130075T1 (enExample)
HU (1) HUS1600034I1 (enExample)
IL (3) IL181523A (enExample)
IN (1) IN2014CN03762A (enExample)
LT (1) LTC2135608I2 (enExample)
LU (1) LU93169I2 (enExample)
ME (1) ME01512B (enExample)
MX (1) MX2007002236A (enExample)
NL (1) NL300825I2 (enExample)
NZ (2) NZ553534A (enExample)
PL (1) PL2135608T3 (enExample)
PT (1) PT2135608E (enExample)
RS (1) RS52632B (enExample)
SG (2) SG155246A1 (enExample)
SI (1) SI2135608T1 (enExample)
WO (1) WO2006026356A2 (enExample)

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CN104326993B (zh) * 2014-10-27 2016-08-17 张远强 一种硝基取代三氮唑亚磺酰丙二酸类化合物、其制备方法及用途
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CN105153056A (zh) * 2015-07-01 2015-12-16 安徽万邦医药科技有限公司 一种[5-溴-4-(4-环丙基萘-1-基)-4h-[1,2,4]三唑-3-基硫烷基]-乙酸甲酯的新制备方法
CN105017168A (zh) * 2015-07-01 2015-11-04 安徽万邦医药科技有限公司 一种[5-溴-4-(4-环丙基萘-1-基)-4h-[1,2,4]三唑-3-基硫烷基]-乙酸甲酯的新制备方法
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CN105566237B (zh) * 2016-03-01 2018-05-18 山东大学 一种治疗痛风的三唑巯乙酸类化合物的制备方法
WO2017215589A1 (zh) * 2016-06-17 2017-12-21 南京明德新药研发股份有限公司 一种卤代化合物及其轴手性异构体
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