JP2004525183A5 - - Google Patents

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Publication number
JP2004525183A5
JP2004525183A5 JP2002581418A JP2002581418A JP2004525183A5 JP 2004525183 A5 JP2004525183 A5 JP 2004525183A5 JP 2002581418 A JP2002581418 A JP 2002581418A JP 2002581418 A JP2002581418 A JP 2002581418A JP 2004525183 A5 JP2004525183 A5 JP 2004525183A5
Authority
JP
Japan
Prior art keywords
formula
alkyl
aryl
compound
compound represented
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002581418A
Other languages
English (en)
Japanese (ja)
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JP2004525183A (ja
Filing date
Publication date
Priority claimed from GBGB0109123.0A external-priority patent/GB0109123D0/en
Priority claimed from GB0205649A external-priority patent/GB0205649D0/en
Application filed filed Critical
Priority claimed from PCT/EP2002/004066 external-priority patent/WO2002083663A1/en
Publication of JP2004525183A publication Critical patent/JP2004525183A/ja
Publication of JP2004525183A5 publication Critical patent/JP2004525183A5/ja
Pending legal-status Critical Current

Links

JP2002581418A 2001-04-11 2002-04-11 Ｎｋ−３およびｎｋ−２受容体アンタゴニストとしてのキノリン−４−カルボキサミド誘導体 Pending JP2004525183A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0109123.0A GB0109123D0 (en) 2001-04-11 2001-04-11 Novel compounds
GB0205649A GB0205649D0 (en) 2002-03-11 2002-03-11 Novel compounds
PCT/EP2002/004066 WO2002083663A1 (en) 2001-04-11 2002-04-11 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists

Publications (2)

Publication Number Publication Date
JP2004525183A JP2004525183A (ja) 2004-08-19
JP2004525183A5 true JP2004525183A5 (enExample) 2005-12-22

Family

ID=26245967

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2002581419A Pending JP2004525184A (ja) 2001-04-11 2002-04-11 Ｎｋ−３およびｎｋ−２受容体アンタゴニストとしての３−置換キノリン−４−カルボキサミド誘導体
JP2002581418A Pending JP2004525183A (ja) 2001-04-11 2002-04-11 Ｎｋ−３およびｎｋ−２受容体アンタゴニストとしてのキノリン−４−カルボキサミド誘導体

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2002581419A Pending JP2004525184A (ja) 2001-04-11 2002-04-11 Ｎｋ−３およびｎｋ−２受容体アンタゴニストとしての３−置換キノリン−４−カルボキサミド誘導体

Country Status (7)

Country Link
US (5) US20040152726A1 (enExample)
EP (3) EP1377567B1 (enExample)
JP (2) JP2004525184A (enExample)
AT (2) ATE318266T1 (enExample)
DE (2) DE60209362T2 (enExample)
ES (2) ES2259096T3 (enExample)
WO (2) WO2002083663A1 (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20031292A1 (it) * 2003-06-25 2004-12-26 Nikem Research Srl Derivati biciclici nk-2 antagonisti selettivi.
US20070060593A1 (en) * 2003-06-25 2007-03-15 Kerns Jeffrey K 4-Carboxamido quinoline derivatives for use as nk-2 and nk-3
AU2005238388B2 (en) 2004-04-28 2011-08-25 Takeda Pharmaceutical Company Limited Fused quinoline derivative and use thereof
GB0417702D0 (en) * 2004-08-09 2004-09-08 Merck Sharp & Dohme New uses
GB0425076D0 (en) * 2004-11-12 2004-12-15 Smithkline Beecham Corp Novel compounds
AU2006253054A1 (en) * 2005-06-03 2006-12-07 Astrazeneca Ab Quinoline derivatives as NK3 anatgonists
MX2007015607A (es) * 2005-06-23 2008-02-25 Astrazeneca Ab Esteres de quinolin 3-sulfonato como moduladores del receptor de nk3.
GB0515580D0 (en) 2005-07-29 2005-09-07 Merck Sharp & Dohme Therapeutic compounds
AR057130A1 (es) 2005-09-21 2007-11-14 Astrazeneca Ab Quinolinas de alquilsulfoxido y una composicion farmaceutica
EP1940795A1 (en) * 2005-09-21 2008-07-09 AstraZeneca AB N-oxo-heterocycle and n-oxo-alkyl quinoline-4-carboxamides as nk-3 receptor ligands
AU2008231384B2 (en) * 2007-03-23 2011-09-15 Amgen Inc. Heterocyclic compounds and their use
WO2008153027A1 (ja) * 2007-06-11 2008-12-18 Takeda Pharmaceutical Company Limited ピロロキノリン誘導体およびその用途
PE20091093A1 (es) 2007-12-03 2009-08-25 Takeda Pharmaceutical Compuesto heterociclico que contiene nitrogeno y su uso
WO2009128262A1 (ja) * 2008-04-15 2009-10-22 武田薬品工業株式会社 キノロン誘導体およびその用途
PL2342182T3 (pl) * 2008-09-15 2013-04-30 H Lundbeck As Pochodne izochinolinonu jako antagoniści NK3
US8242134B2 (en) 2008-09-15 2012-08-14 H. Lundbeck A/S Isoquinolinone derivatives as NK3 antagonists
USRE49686E1 (en) 2008-09-19 2023-10-10 Takeda Pharmaceutical Company Limited Nitrogen-containing heterocyclic compound and use of same
CN102584852B (zh) * 2011-12-30 2014-08-13 厦门大学 真菌代谢产物桥南霉素及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL186665B1 (pl) * 1994-05-27 2004-02-27 Smithkline Beecham Spa Pochodne chinoliny jako antagoniści receptorów NKtachykininy, sposób ich wytwarzania, kompozycja farmaceutyczna zawierająca pochodne chinoliny oraz ich zastosowanie
EP0876347B1 (en) * 1995-11-24 2005-03-02 GlaxoSmithKline S.p.A. Quinoline derivatives
AR004735A1 (es) * 1995-11-24 1999-03-10 Smithkline Beecham Spa Quinoleina 4-amido sustituida, un procedimiento para su preparacion, una composicion farmaceutica que los contiene y el uso de los mismos para lapreparacion de un medicamento.
IL133036A0 (en) * 1997-05-23 2001-03-19 Smithkline Beecham Spa Quinoline-4-carboxamide derivatives as nk-2 and nk-3 receptor antagonists
BR9915475A (pt) * 1998-11-20 2001-12-18 Smithkline Beecham Spa Derivados da quinolina-4-carboxamida comoantagonistas dos receptores de nk-3 e nk-2
GB9825554D0 (en) * 1998-11-20 1999-01-13 Smithkline Beecham Spa Novel Compounds

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