AR073964A1 - Composiciones que comprenden acido 4-(2-(5-bromo-4-(1-ciclopropilnaftalen -4-il) -4h- 1,2,4-triazol-3-il tio ) acetamido)-3-clorobenzoico y sus sales farmaceuticamente aceptables y metodos de preparacion y uso delos mismos - Google Patents
Composiciones que comprenden acido 4-(2-(5-bromo-4-(1-ciclopropilnaftalen -4-il) -4h- 1,2,4-triazol-3-il tio ) acetamido)-3-clorobenzoico y sus sales farmaceuticamente aceptables y metodos de preparacion y uso delos mismosInfo
- Publication number
- AR073964A1 AR073964A1 ARP090104095A ARP090104095A AR073964A1 AR 073964 A1 AR073964 A1 AR 073964A1 AR P090104095 A ARP090104095 A AR P090104095A AR P090104095 A ARP090104095 A AR P090104095A AR 073964 A1 AR073964 A1 AR 073964A1
- Authority
- AR
- Argentina
- Prior art keywords
- subject
- ciclopropilnaftalen
- chlorobenzoic
- triazol
- acetamide
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4196—1,2,4-Triazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Virology (AREA)
- AIDS & HIV (AREA)
- Molecular Biology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Reivindicacion 1: Una composicion farmacéutica caracterizada porque comprende un compuesto o mezcla de compuestos de estructura (1) donde M es hidrogeno, sodio, potasio, calcio, o arginina; y uno o más diluyentes; uno o más aglutinantes; uno o más agentes recubridores; uno o más agentes dispersantes; y uno o más plastificantes. Reivindicacion 16: Un método para prevenir una infeccion de un virus de inmunodeficiencia en un sujeto, para tratar una infeccion de un virus de inmunodeficiencia en un sujeto, para prevenir el síndrome de inmunodeficiencia adquirida (SIDA) en un sujeto, para tratar el síndrome de inmunodeficiencia adquirida (SIDA) en un sujeto, para prevenir el complejo relacionado con el SIDA (ARC) en un sujeto o para tratar el complejo relacionado con el SIDA (ARC) en un sujeto, caracterizado porque comprende administrarle a un sujeto que lo necesita una cantidad eficaz de una composicion de acuerdo con cualquiera de las reivindicaciones precedentes.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10843708P | 2008-10-24 | 2008-10-24 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR073964A1 true AR073964A1 (es) | 2010-12-15 |
Family
ID=41491449
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP090104095A AR073964A1 (es) | 2008-10-24 | 2009-10-23 | Composiciones que comprenden acido 4-(2-(5-bromo-4-(1-ciclopropilnaftalen -4-il) -4h- 1,2,4-triazol-3-il tio ) acetamido)-3-clorobenzoico y sus sales farmaceuticamente aceptables y metodos de preparacion y uso delos mismos |
Country Status (7)
Country | Link |
---|---|
US (1) | US20110244049A1 (es) |
EP (1) | EP2349258A1 (es) |
AR (1) | AR073964A1 (es) |
CA (1) | CA2741368A1 (es) |
IL (1) | IL212463A0 (es) |
TW (1) | TW201022215A (es) |
WO (1) | WO2010048593A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2433633A1 (en) | 2004-08-25 | 2012-03-28 | Ardea Biosciences, Inc. | Triazolyl alpha -mercaptoacetanildes as inhibitors of HIV reverse transcriptase |
WO2007050087A1 (en) | 2004-08-25 | 2007-05-03 | Ardea Biosciences, Inc. | N[S(4-aryl-triazol-3-yl)α -mercaptoacetyl]-p-amino benozoic acids AS HIV REVERSE TRANSCRIPTASE INHIBITORS |
WO2012114352A2 (en) * | 2011-02-21 | 2012-08-30 | Hetero Research Foundation | Pharmaceutical compositions of maraviroc and process for the preparation thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2433633A1 (en) * | 2004-08-25 | 2012-03-28 | Ardea Biosciences, Inc. | Triazolyl alpha -mercaptoacetanildes as inhibitors of HIV reverse transcriptase |
WO2007050087A1 (en) * | 2004-08-25 | 2007-05-03 | Ardea Biosciences, Inc. | N[S(4-aryl-triazol-3-yl)α -mercaptoacetyl]-p-amino benozoic acids AS HIV REVERSE TRANSCRIPTASE INHIBITORS |
CN103058944B (zh) * | 2007-11-27 | 2015-08-05 | 亚德生化公司 | 调节血液尿酸水平的化合物 |
-
2009
- 2009-10-23 EP EP09749251A patent/EP2349258A1/en not_active Withdrawn
- 2009-10-23 US US13/125,697 patent/US20110244049A1/en not_active Abandoned
- 2009-10-23 WO PCT/US2009/061970 patent/WO2010048593A1/en active Application Filing
- 2009-10-23 AR ARP090104095A patent/AR073964A1/es not_active Application Discontinuation
- 2009-10-23 CA CA2741368A patent/CA2741368A1/en not_active Abandoned
- 2009-10-26 TW TW098136212A patent/TW201022215A/zh unknown
-
2011
- 2011-04-26 IL IL212463A patent/IL212463A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
IL212463A0 (en) | 2011-06-30 |
TW201022215A (en) | 2010-06-16 |
WO2010048593A1 (en) | 2010-04-29 |
US20110244049A1 (en) | 2011-10-06 |
EP2349258A1 (en) | 2011-08-03 |
CA2741368A1 (en) | 2010-04-29 |
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Legal Events
Date | Code | Title | Description |
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FA | Abandonment or withdrawal |