JP2002535314A - Ｖｌａ−４により媒介される白血球接着を阻害する化合物 - Google Patents

Ｖｌａ−４により媒介される白血球接着を阻害する化合物

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Publication number
JP2002535314A
JP2002535314A JP2000594785A JP2000594785A JP2002535314A JP 2002535314 A JP2002535314 A JP 2002535314A JP 2000594785 A JP2000594785 A JP 2000594785A JP 2000594785 A JP2000594785 A JP 2000594785A JP 2002535314 A JP2002535314 A JP 2002535314A
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JP
Japan
Prior art keywords
substituted
alkyl
aryl
heteroaryl
heterocyclic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2000594785A
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English (en)
Japanese (ja)
Inventor
アンドレイ ダブリュー． コンラディ，
マイケル エイ． プレイス，
ユージーン ディー． ソーセット，
スーザン アシュウェル，
ディミトリオス サランタキス，
グレゴリー エス． ウェルメイカー，
アンソニー クレフト，
クリストファー センコ，
ロバート ウォーレン サリバン，
クリストファー ジョセフ ソアレス，
キーブ スイ リー，
クリスティン エム． タービー，
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth LLC
Original Assignee
Wyeth LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth LLC filed Critical Wyeth LLC
Priority claimed from PCT/US2000/001540 external-priority patent/WO2000043369A1/en
Publication of JP2002535314A publication Critical patent/JP2002535314A/ja
Pending legal-status Critical Current

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JP2002535317A (ja) * 1999-01-22 2002-10-22 エラン ファーマシューティカルズ，インコーポレイテッド Ｖｌａ−４関連障害を処置するアシル誘導体
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JP2002535317A (ja) * 1999-01-22 2002-10-22 エラン ファーマシューティカルズ，インコーポレイテッド Ｖｌａ−４関連障害を処置するアシル誘導体
JP4754693B2 (ja) * 1999-01-22 2011-08-24 エラン ファーマシューティカルズ，インコーポレイテッド Ｖｌａ−４関連障害を処置するアシル誘導体
JP2007526230A (ja) * 2003-06-25 2007-09-13 エラン ファーマシューティカルズ，インコーポレイテッド 関節リウマチを治療する方法および組成物
JP2008540686A (ja) * 2005-05-20 2008-11-20 イーラン ファーマスーティカルズ、インコーポレイテッド Ｖｌａ−４アンタゴニストとしてのイミダゾロンフェニルアラニン誘導体
JP2014237639A (ja) * 2010-06-16 2014-12-18 アルデア バイオサイエンシーズ インク． チオ酢酸化合物、組成物、および、その使用方法
JP2013544285A (ja) * 2010-11-29 2013-12-12 ガリオン ファーマシューティカルズ インコーポレイテッド 呼吸制御障害または呼吸制御疾患の処置用の呼吸刺激薬としての化合物

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US20040147512A1 (en) 2004-07-29
EP1144388B1 (en) 2010-01-13
US20100160341A1 (en) 2010-06-24
KR100711840B1 (ko) 2007-05-02
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US7538215B2 (en) 2009-05-26
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US20050203093A1 (en) 2005-09-15
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