IN2015DN01119A - - Google Patents

Info

Publication number
IN2015DN01119A
IN2015DN01119A IN1119DEN2015A IN2015DN01119A IN 2015DN01119 A IN2015DN01119 A IN 2015DN01119A IN 1119DEN2015 A IN1119DEN2015 A IN 1119DEN2015A IN 2015DN01119 A IN2015DN01119 A IN 2015DN01119A
Authority
IN
India
Prior art keywords
compounds
disclosed
methods
intermediates
synthesis
Prior art date
Application number
Other languages
English (en)
Inventor
Ende Christopher William Am
Michael Eric Green
Douglas Scott Johnson
Gregory Wayne Kauffman
Christopher John Odonnell
Nandini Chaturbhai Patel
Martin Youngjin Pettersson
Antonia Friederike Stepan
Cory Michael Stiff
Chakrapani Subramanyam
Tuan Phong Tran
Patrick Robert Verhoest
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IN2015DN01119A publication Critical patent/IN2015DN01119A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Epidemiology (AREA)
IN1119DEN2015 2012-09-21 2013-09-06 IN2015DN01119A (OSRAM)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261703969P 2012-09-21 2012-09-21
PCT/IB2013/058347 WO2014045156A1 (en) 2012-09-21 2013-09-06 Novel bicyclic pyridinones

Publications (1)

Publication Number Publication Date
IN2015DN01119A true IN2015DN01119A (OSRAM) 2015-06-26

Family

ID=49585452

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1119DEN2015 IN2015DN01119A (OSRAM) 2012-09-21 2013-09-06

Country Status (46)

Country Link
US (3) US8916564B2 (OSRAM)
EP (1) EP2897956B1 (OSRAM)
JP (1) JP5844018B2 (OSRAM)
KR (1) KR101725696B1 (OSRAM)
CN (1) CN104662021B (OSRAM)
AP (1) AP2015008277A0 (OSRAM)
AR (1) AR092628A1 (OSRAM)
AU (1) AU2013319845B2 (OSRAM)
BR (1) BR112015006436A2 (OSRAM)
CA (1) CA2882386C (OSRAM)
CL (1) CL2015000717A1 (OSRAM)
CR (1) CR20150053A (OSRAM)
CU (1) CU20150021A7 (OSRAM)
CY (1) CY1118662T1 (OSRAM)
DK (1) DK2897956T3 (OSRAM)
DO (1) DOP2015000069A (OSRAM)
EA (1) EA026668B1 (OSRAM)
EC (1) ECSP15015594A (OSRAM)
ES (1) ES2609987T3 (OSRAM)
GE (1) GEP201706659B (OSRAM)
GT (1) GT201500069A (OSRAM)
HR (1) HRP20161558T1 (OSRAM)
HU (1) HUE031248T2 (OSRAM)
IL (1) IL237163A (OSRAM)
IN (1) IN2015DN01119A (OSRAM)
LT (1) LT2897956T (OSRAM)
MA (1) MA37886B1 (OSRAM)
MD (1) MD4583B1 (OSRAM)
ME (1) ME02571B (OSRAM)
MX (1) MX360599B (OSRAM)
MY (1) MY181891A (OSRAM)
NI (1) NI201500038A (OSRAM)
NZ (1) NZ704863A (OSRAM)
PE (1) PE20150686A1 (OSRAM)
PH (1) PH12015500376B1 (OSRAM)
PL (1) PL2897956T3 (OSRAM)
PT (1) PT2897956T (OSRAM)
RS (1) RS55426B1 (OSRAM)
SG (1) SG11201501074WA (OSRAM)
SI (1) SI2897956T1 (OSRAM)
TN (1) TN2015000084A1 (OSRAM)
TW (1) TWI500616B (OSRAM)
UA (1) UA110688C2 (OSRAM)
UY (1) UY35039A (OSRAM)
WO (1) WO2014045156A1 (OSRAM)
ZA (1) ZA201501195B (OSRAM)

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US10562897B2 (en) 2014-01-16 2020-02-18 Janssen Pharmaceutica Nv Substituted 3,4-dihydro-2H-pyrido[1,2-a]pyrazine-1,6-diones as gamma secretase modulators
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US20220192984A1 (en) 2018-10-02 2022-06-23 Frequency Therapeutics, Inc. Pharmaceutical compositions comprising otic therapeutic agents and related methods
SG11202111191YA (en) 2019-04-08 2021-11-29 Frequency Therapeutics Inc Combination of chir99021 and valproic acid for treating hearing loss
PH12022551379A1 (en) 2019-12-06 2023-05-03 Vertex Pharma Substituted tetrahydrofurans as modulators of sodium channels
CN113402490B (zh) * 2021-03-29 2023-01-03 白银京宇新药业有限公司 一种1,2,6,7-四氢-8H-茚并[5,4-b]呋喃-8-酮的制备方法
KR20240031300A (ko) 2021-06-04 2024-03-07 버텍스 파마슈티칼스 인코포레이티드 나트륨 채널 조절제로서의 n-(하이드록시알킬 (헤테로)아릴) 테트라하이드로푸란 카르복스아미드
CN114034792B (zh) * 2021-11-09 2024-06-25 山东新华制药股份有限公司 检测氯酮含量的液相色谱分析方法

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