IL287136B2 - Receptor inhibitors - interacting with protein kinase 1 - Google Patents
Receptor inhibitors - interacting with protein kinase 1Info
- Publication number
- IL287136B2 IL287136B2 IL287136A IL28713621A IL287136B2 IL 287136 B2 IL287136 B2 IL 287136B2 IL 287136 A IL287136 A IL 287136A IL 28713621 A IL28713621 A IL 28713621A IL 287136 B2 IL287136 B2 IL 287136B2
- Authority
- IL
- Israel
- Prior art keywords
- optionally substituted
- alkyl
- halo
- certain embodiments
- ring
- Prior art date
Links
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- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662292202P | 2016-02-05 | 2016-02-05 | |
| US201662341019P | 2016-05-24 | 2016-05-24 | |
| US201662363775P | 2016-07-18 | 2016-07-18 | |
| US201662385217P | 2016-09-08 | 2016-09-08 | |
| US201662417219P | 2016-11-03 | 2016-11-03 | |
| PCT/US2017/016509 WO2017136727A2 (en) | 2016-02-05 | 2017-02-03 | Compounds, compositions and methods |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| IL287136A IL287136A (en) | 2021-12-01 |
| IL287136B1 IL287136B1 (en) | 2023-05-01 |
| IL287136B2 true IL287136B2 (en) | 2023-09-01 |
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- 2018-08-01 DO DO2018000175A patent/DOP2018000175A/es unknown
- 2018-08-02 MX MX2021013228A patent/MX2021013228A/es unknown
- 2018-08-02 SA SA518392146A patent/SA518392146B1/ar unknown
- 2018-08-02 CL CL2018002081A patent/CL2018002081A1/es unknown
- 2018-08-02 MX MX2021013226A patent/MX2021013226A/es unknown
- 2018-08-21 CO CONC2018/0008707A patent/CO2018008707A2/es unknown
- 2018-09-03 EC ECSENADI201866138A patent/ECSP18066138A/es unknown
- 2018-09-13 US US16/130,817 patent/US10604535B2/en active Active
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2020
- 2020-02-05 US US16/782,446 patent/US20200317691A1/en not_active Abandoned
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2021
- 2021-02-25 US US17/185,684 patent/US20230043400A1/en not_active Abandoned
- 2021-11-02 JP JP2021179107A patent/JP7381543B2/ja active Active
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2023
- 2023-08-10 US US18/232,435 patent/US12358928B2/en active Active
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2014125444A1 (en) * | 2013-02-15 | 2014-08-21 | Glaxosmithkline Intellectual Property Development Limited | Heterocyclic amides as kinase inhibitors |
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