CN102548999A - 含有取代的含氮稠杂环的头孢菌素衍生物 - Google Patents
含有取代的含氮稠杂环的头孢菌素衍生物 Download PDFInfo
- Publication number
- CN102548999A CN102548999A CN2010800049569A CN201080004956A CN102548999A CN 102548999 A CN102548999 A CN 102548999A CN 2010800049569 A CN2010800049569 A CN 2010800049569A CN 201080004956 A CN201080004956 A CN 201080004956A CN 102548999 A CN102548999 A CN 102548999A
- Authority
- CN
- China
- Prior art keywords
- bases
- yue
- ene
- oct
- thia
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/57—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with a further substituent in position 7, e.g. cephamycines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Abstract
Description
PCT国内申请,说明书已公开。
Claims (1)
- PCT国内申请,权利要求书已公开。
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN2010800049569A CN102548999A (zh) | 2009-01-20 | 2010-01-20 | 含有取代的含氮稠杂环的头孢菌素衍生物 |
Applications Claiming Priority (10)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN200910014009.7 | 2009-01-20 | ||
CN200910014009 | 2009-01-20 | ||
CN200910140527.3 | 2009-05-01 | ||
CN200910140527 | 2009-05-01 | ||
CN200910145670 | 2009-05-17 | ||
CN200910145670.1 | 2009-05-17 | ||
CN200910146131.X | 2009-06-09 | ||
CN200910146131 | 2009-06-09 | ||
PCT/CN2010/000086 WO2010083725A1 (zh) | 2009-01-20 | 2010-01-20 | 含有取代的含氮稠杂环的头孢菌素衍生物 |
CN2010800049569A CN102548999A (zh) | 2009-01-20 | 2010-01-20 | 含有取代的含氮稠杂环的头孢菌素衍生物 |
Publications (1)
Publication Number | Publication Date |
---|---|
CN102548999A true CN102548999A (zh) | 2012-07-04 |
Family
ID=42355528
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN2010800049569A Pending CN102548999A (zh) | 2009-01-20 | 2010-01-20 | 含有取代的含氮稠杂环的头孢菌素衍生物 |
Country Status (2)
Country | Link |
---|---|
CN (1) | CN102548999A (zh) |
WO (1) | WO2010083725A1 (zh) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA103195C2 (uk) | 2008-08-11 | 2013-09-25 | Глаксосмитклайн Ллк | Похідні пурину для застосування у лікуванні алергій, запальних та інфекційних захворювань |
DK2734186T3 (en) | 2011-07-22 | 2019-01-07 | Glaxosmithkline Llc | COMPOSITION |
UA114109C2 (xx) | 2012-08-24 | 2017-04-25 | Піразолопіримідинові сполуки | |
RU2640200C2 (ru) | 2012-11-20 | 2017-12-27 | ГЛАКСОСМИТКЛАЙН ЭлЭлСи | Новые соединения |
US9550785B2 (en) | 2012-11-20 | 2017-01-24 | Glaxosmithkline Llc | Pyrrolopyrimidines as therapeutic agents for the treatment of diseases |
LT2922549T (lt) | 2012-11-20 | 2017-09-11 | Glaxosmithkline Llc | Naujieji junginiai |
MA44007A (fr) | 2016-02-05 | 2018-12-19 | Denali Therapeutics Inc | Inhibiteurs du récepteur interagissant avec protéine kinase 1 |
TW201819361A (zh) | 2016-09-03 | 2018-06-01 | 印度商托仁特生技有限公司 | 新穎吲唑化合物 |
PL3552017T3 (pl) | 2016-12-09 | 2022-08-08 | Denali Therapeutics Inc. | Związki użyteczne jako inhibitory RIPK1 |
WO2020206381A1 (en) * | 2019-04-03 | 2020-10-08 | Sutton Larry D | Cephem compounds with latent reactive groups and methods of using and making same |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4590186A (en) * | 1984-01-16 | 1986-05-20 | Fujisawa Pharmaceutical Co., Ltd. | Cephem compounds having 3-bicyclic heterocyclic cation groups |
US5336673A (en) * | 1990-07-05 | 1994-08-09 | Dae Woong Pharmaceutical Co., Ltd. | 3-substituted cephem compounds |
CN101066974A (zh) * | 2007-04-20 | 2007-11-07 | 苏州中联化学制药有限公司 | 一种抗菌素硫酸头孢匹罗的合成方法 |
CN101337971A (zh) * | 2008-08-15 | 2009-01-07 | 苏州万庆药业有限公司 | 一种抗菌素盐酸头孢吡肟的合成方法 |
-
2010
- 2010-01-20 CN CN2010800049569A patent/CN102548999A/zh active Pending
- 2010-01-20 WO PCT/CN2010/000086 patent/WO2010083725A1/zh active Application Filing
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4590186A (en) * | 1984-01-16 | 1986-05-20 | Fujisawa Pharmaceutical Co., Ltd. | Cephem compounds having 3-bicyclic heterocyclic cation groups |
US5336673A (en) * | 1990-07-05 | 1994-08-09 | Dae Woong Pharmaceutical Co., Ltd. | 3-substituted cephem compounds |
CN101066974A (zh) * | 2007-04-20 | 2007-11-07 | 苏州中联化学制药有限公司 | 一种抗菌素硫酸头孢匹罗的合成方法 |
CN101337971A (zh) * | 2008-08-15 | 2009-01-07 | 苏州万庆药业有限公司 | 一种抗菌素盐酸头孢吡肟的合成方法 |
Also Published As
Publication number | Publication date |
---|---|
WO2010083725A1 (zh) | 2010-07-29 |
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C06 | Publication | ||
PB01 | Publication | ||
C10 | Entry into substantive examination | ||
SE01 | Entry into force of request for substantive examination | ||
C12 | Rejection of a patent application after its publication | ||
RJ01 | Rejection of invention patent application after publication |
Application publication date: 20120704 |