HUP0000323A3 - N-substituted 2-cyanopyrrolidine derivatives, process for producing them and pharmaceutical compositions containing them - Google Patents

N-substituted 2-cyanopyrrolidine derivatives, process for producing them and pharmaceutical compositions containing them

Info

Publication number
HUP0000323A3
HUP0000323A3 HU0000323A HUP0000323A HUP0000323A3 HU P0000323 A3 HUP0000323 A3 HU P0000323A3 HU 0000323 A HU0000323 A HU 0000323A HU P0000323 A HUP0000323 A HU P0000323A HU P0000323 A3 HUP0000323 A3 HU P0000323A3
Authority
HU
Hungary
Prior art keywords
substituted
producing
pharmaceutical compositions
compositions containing
cyanopyrrolidine derivatives
Prior art date
Application number
HU0000323A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25000236&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUP0000323(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of HUP0000323A2 publication Critical patent/HUP0000323A2/hu
Publication of HUP0000323A3 publication Critical patent/HUP0000323A3/hu
Publication of HU227125B1 publication Critical patent/HU227125B1/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU0000323A 1996-11-07 1997-11-05 N-substituted 2-cyanopyrrolidine derivatives, process for producing them and pharmaceutical compositions containing them HU227125B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74629596A 1996-11-07 1996-11-07
PCT/EP1997/006125 WO1998019998A2 (en) 1996-11-07 1997-11-05 N-substituted 2-cyanopyrrolidines

Publications (3)

Publication Number Publication Date
HUP0000323A2 HUP0000323A2 (hu) 2000-08-28
HUP0000323A3 true HUP0000323A3 (en) 2002-02-28
HU227125B1 HU227125B1 (en) 2010-07-28

Family

ID=25000236

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0000323A HU227125B1 (en) 1996-11-07 1997-11-05 N-substituted 2-cyanopyrrolidine derivatives, process for producing them and pharmaceutical compositions containing them

Country Status (28)

Country Link
EP (1) EP0937040B1 (hu)
JP (1) JP3217380B2 (hu)
KR (1) KR20000053081A (hu)
CN (1) CN1134412C (hu)
AR (1) AR009605A1 (hu)
AT (1) ATE271543T1 (hu)
AU (1) AU726186B2 (hu)
BR (1) BR9714130B1 (hu)
CA (1) CA2269810C (hu)
CO (1) CO4910126A1 (hu)
CZ (1) CZ296303B6 (hu)
DE (1) DE69729947T2 (hu)
ES (1) ES2226004T3 (hu)
HK (1) HK1022149A1 (hu)
HU (1) HU227125B1 (hu)
ID (2) ID21350A (hu)
IL (3) IL129561A0 (hu)
NO (1) NO312667B1 (hu)
NZ (1) NZ335146A (hu)
PE (1) PE10699A1 (hu)
PL (1) PL190498B1 (hu)
PT (1) PT937040E (hu)
RU (1) RU2180901C2 (hu)
SK (1) SK282904B6 (hu)
TR (1) TR199901004T2 (hu)
TW (1) TW492957B (hu)
WO (1) WO1998019998A2 (hu)
ZA (1) ZA979985B (hu)

Families Citing this family (249)

* Cited by examiner, † Cited by third party
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CN115322129A (zh) * 2022-08-29 2022-11-11 湖北科技学院 双氰基吡咯烷类衍生物及其制备方法和应用

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DE69729947D1 (de) 2004-08-26
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TW492957B (en) 2002-07-01
AU5318498A (en) 1998-05-29
WO1998019998A2 (en) 1998-05-14
DE69729947T2 (de) 2005-04-21
NO992028D0 (no) 1999-04-28
ID18331A (id) 1998-03-26
BR9714130B1 (pt) 2010-03-23
ATE271543T1 (de) 2004-08-15
CZ161599A3 (cs) 1999-08-11
CN1236361A (zh) 1999-11-24
PE10699A1 (es) 1999-03-02
CZ296303B6 (cs) 2006-02-15
BR9714130A (pt) 2000-02-29
CO4910126A1 (es) 2000-04-24
AU726186B2 (en) 2000-11-02
EP0937040B1 (en) 2004-07-21
ZA979985B (en) 1998-05-07
KR20000053081A (ko) 2000-08-25
PL190498B1 (pl) 2005-12-30
JP2000511559A (ja) 2000-09-05
NO312667B1 (no) 2002-06-17
HK1022149A1 (en) 2000-07-28
SK282904B6 (sk) 2003-01-09
AR009605A1 (es) 2000-04-26
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IL129561A (en) 2006-10-31
NO992028L (no) 1999-04-28
SK60899A3 (en) 2000-04-10
PT937040E (pt) 2004-11-30
HUP0000323A2 (hu) 2000-08-28
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