HU191053B - Process for preparing piperidyl-ester- and piperidyl-amide-derivatives of aromatic carboxylic acids and pharmaceutical preparations containing such compounds - Google Patents

Process for preparing piperidyl-ester- and piperidyl-amide-derivatives of aromatic carboxylic acids and pharmaceutical preparations containing such compounds Download PDF

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Publication number
HU191053B
HU191053B HU832335A HU233583A HU191053B HU 191053 B HU191053 B HU 191053B HU 832335 A HU832335 A HU 832335A HU 233583 A HU233583 A HU 233583A HU 191053 B HU191053 B HU 191053B
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HU
Hungary
Prior art keywords
formula
group
compound
hydrogen
alkyl
Prior art date
Application number
HU832335A
Other languages
English (en)
Hungarian (hu)
Inventor
Guenter Engel
Peter Donatsch
Peter B Richardson
Bruno Huegi
Paul Stadler
Original Assignee
Sandoz Ag,Ch
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag,Ch filed Critical Sandoz Ag,Ch
Publication of HU191053B publication Critical patent/HU191053B/hu

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/06—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/12—Oxygen atoms acylated by aromatic or heteroaromatic carboxylic acids, e.g. cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/14—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Indole Compounds (AREA)
HU832335A 1982-06-29 1983-06-28 Process for preparing piperidyl-ester- and piperidyl-amide-derivatives of aromatic carboxylic acids and pharmaceutical preparations containing such compounds HU191053B (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
CH397982 1982-06-29
CH426782 1982-07-13
CH695082 1982-11-30
CH695182 1982-11-30
CH749482 1982-12-22
CH749582 1982-12-22
CH125683 1983-03-09

Publications (1)

Publication Number Publication Date
HU191053B true HU191053B (en) 1986-12-28

Family

ID=27561049

Family Applications (1)

Application Number Title Priority Date Filing Date
HU832335A HU191053B (en) 1982-06-29 1983-06-28 Process for preparing piperidyl-ester- and piperidyl-amide-derivatives of aromatic carboxylic acids and pharmaceutical preparations containing such compounds

Country Status (20)

Country Link
US (3) US4803199A (OSRAM)
AT (1) AT391136B (OSRAM)
AU (2) AU570002B2 (OSRAM)
CH (2) CH669792A5 (OSRAM)
CY (1) CY1500A (OSRAM)
DE (6) DE19475004I2 (OSRAM)
DK (1) DK172475B1 (OSRAM)
FI (1) FI74707C (OSRAM)
FR (1) FR2531083B1 (OSRAM)
GB (4) GB2125398B (OSRAM)
HK (1) HK60690A (OSRAM)
HU (1) HU191053B (OSRAM)
IL (1) IL69081A (OSRAM)
IT (1) IT1173724B (OSRAM)
NL (2) NL191991C (OSRAM)
NZ (1) NZ204714A (OSRAM)
PT (1) PT76937B (OSRAM)
SE (1) SE463210B (OSRAM)
SG (1) SG53789G (OSRAM)
WO (1) WO1984000166A1 (OSRAM)

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FR2531083A1 (fr) 1984-02-03
AT391136B (de) 1990-08-27
AU1628683A (en) 1984-01-05
SE463210B (sv) 1990-10-22
GB2125398B (en) 1986-11-26
DK295183A (da) 1983-12-30
DE3348333C2 (OSRAM) 1992-08-27
DE3348332C2 (OSRAM) 1992-08-06
DE19475004I2 (de) 2003-06-12
AU8243487A (en) 1988-04-28
DE3322574A1 (de) 1983-12-29
FI74707B (fi) 1987-11-30
ATA235883A (de) 1990-02-15
NL8302253A (nl) 1984-01-16
SG53789G (en) 1989-12-08
IT1173724B (it) 1987-06-24
AU570002B2 (en) 1988-03-03
WO1984000166A1 (fr) 1984-01-19
NL191991C (nl) 1996-12-03
US4803199A (en) 1989-02-07
NL191991B (nl) 1996-08-01
DK172475B1 (da) 1998-09-14
GB2166727A (en) 1986-05-14
PT76937B (en) 1986-03-11
GB2125398A (en) 1984-03-07
GB8520187D0 (en) 1985-09-18
GB2166726B (en) 1986-11-26
NL970021I1 (nl) 1997-08-01
NZ204714A (en) 1986-08-08
US4910207A (en) 1990-03-20
GB8317365D0 (en) 1983-07-27
GB8520188D0 (en) 1985-09-18
IT8348580A1 (it) 1984-12-27
GB2166728A (en) 1986-05-14
SE8303651L (sv) 1983-12-30
GB2166726A (en) 1986-05-14
FI832293L (fi) 1983-12-30
SE8303651D0 (sv) 1983-06-27
AU603399B2 (en) 1990-11-15
DK295183D0 (da) 1983-06-27
PT76937A (en) 1983-07-01
CY1500A (en) 1990-08-03
DE3348331C2 (OSRAM) 1992-08-06
US5017582A (en) 1991-05-21
GB8520186D0 (en) 1985-09-18
FI832293A0 (fi) 1983-06-22
HK60690A (en) 1990-08-17
DE3322574C2 (OSRAM) 1992-07-30
DE3348334C2 (OSRAM) 1992-08-06
GB2166727B (en) 1986-11-26
NL970021I2 (nl) 1998-01-05
IL69081A0 (en) 1983-10-31
CH669792A5 (OSRAM) 1989-04-14
CH669954A5 (en) 1989-04-28
IL69081A (en) 1987-02-27
IT8348580A0 (it) 1983-06-27
FI74707C (fi) 1988-03-10
GB2166728B (en) 1986-11-26

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