HK1098471A1 - Azaindoles useful as inhibitors of jak and other protein kinases - Google Patents
Azaindoles useful as inhibitors of jak and other protein kinasesInfo
- Publication number
- HK1098471A1 HK1098471A1 HK07104783.6A HK07104783A HK1098471A1 HK 1098471 A1 HK1098471 A1 HK 1098471A1 HK 07104783 A HK07104783 A HK 07104783A HK 1098471 A1 HK1098471 A1 HK 1098471A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- inhibitors
- protein kinases
- jak
- azaindoles useful
- azaindoles
- Prior art date
Links
- 102000001253 Protein Kinase Human genes 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 108060006633 protein kinase Proteins 0.000 title abstract 2
- 125000005334 azaindolyl group Chemical group N1N=C(C2=CC=CC=C12)* 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
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- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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PCT/US2005/010846 WO2005095400A1 (fr) | 2004-03-30 | 2005-03-30 | Azaindoles utiles comme inhibiteurs de janus kinases et d'autres proteines kinases |
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2015
- 2015-02-05 US US14/614,740 patent/US20150152103A1/en not_active Abandoned
- 2015-03-16 JP JP2015051664A patent/JP2015113347A/ja not_active Withdrawn
-
2016
- 2016-05-24 NO NO20160876A patent/NO20160876A1/no not_active Application Discontinuation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20230330 |