FI112864B - Menetelmä fluorialkoksilla substituoitujen bentsamidien valmistamiseksi - Google Patents

Menetelmä fluorialkoksilla substituoitujen bentsamidien valmistamiseksi Download PDF

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Publication number
FI112864B
FI112864B FI956333A FI956333A FI112864B FI 112864 B FI112864 B FI 112864B FI 956333 A FI956333 A FI 956333A FI 956333 A FI956333 A FI 956333A FI 112864 B FI112864 B FI 112864B
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FI
Finland
Prior art keywords
halogen
alkoxy
alkyl
salts
represents hydrogen
Prior art date
Application number
FI956333A
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English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI956333A0 (fi
FI956333A (fi
Inventor
Hermann Amschler
Rolf Beume
Dieter Flockerzi
Ulrich Kilian
Armin Hatzelmann
Christian Schudt
Beate Gutterer
Horst P O Wolf
Original Assignee
Altana Pharma Ag
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Publication date
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Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Publication of FI956333A0 publication Critical patent/FI956333A0/fi
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C235/56—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
FI956333A 1993-07-02 1995-12-29 Menetelmä fluorialkoksilla substituoitujen bentsamidien valmistamiseksi FI112864B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH199693 1993-07-02
CH199693 1993-07-02
EP9402169 1994-07-02
PCT/EP1994/002169 WO1995001338A1 (fr) 1993-07-02 1994-07-02 Nouveaux benzamides a substituants fluoroalcoxy et leur utilisation comme inhibiteurs de la phosphodiesterase nucleotidique cyclique

Publications (3)

Publication Number Publication Date
FI956333A0 FI956333A0 (fi) 1995-12-29
FI956333A FI956333A (fi) 1995-12-29
FI112864B true FI112864B (fi) 2004-01-30

Family

ID=4223466

Family Applications (1)

Application Number Title Priority Date Filing Date
FI956333A FI112864B (fi) 1993-07-02 1995-12-29 Menetelmä fluorialkoksilla substituoitujen bentsamidien valmistamiseksi

Country Status (28)

Country Link
US (1) US5712298A (fr)
EP (1) EP0706513B1 (fr)
JP (1) JP3093271B2 (fr)
KR (1) KR100331255B1 (fr)
CN (1) CN1046939C (fr)
AT (1) ATE217612T1 (fr)
AU (1) AU687087B2 (fr)
CA (1) CA2165192C (fr)
CY (2) CY2389B1 (fr)
CZ (1) CZ290266B6 (fr)
DE (2) DE59410119D1 (fr)
DK (1) DK0706513T3 (fr)
ES (1) ES2176252T3 (fr)
FI (1) FI112864B (fr)
FR (1) FR10C0052I2 (fr)
HK (1) HK1011690A1 (fr)
HU (1) HU220041B (fr)
LU (1) LU91709I2 (fr)
LV (1) LV13074B (fr)
NO (2) NO305598B1 (fr)
NZ (1) NZ271316A (fr)
PL (1) PL178314B1 (fr)
PT (1) PT706513E (fr)
RU (1) RU2137754C1 (fr)
SG (1) SG143011A1 (fr)
SI (1) SI0706513T1 (fr)
SK (1) SK283263B6 (fr)
WO (1) WO1995001338A1 (fr)

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