EE03086B1 - N4-(asendatud-oksükarbonüül)-5'-desoksü-5-fluorotsütidiinid, nende saamise meetod ja neid sisaldavad ravimpreparaadid - Google Patents

N4-(asendatud-oksükarbonüül)-5'-desoksü-5-fluorotsütidiinid, nende saamise meetod ja neid sisaldavad ravimpreparaadid

Info

Publication number
EE03086B1
EE03086B1 EE9400154A EE9400154A EE03086B1 EE 03086 B1 EE03086 B1 EE 03086B1 EE 9400154 A EE9400154 A EE 9400154A EE 9400154 A EE9400154 A EE 9400154A EE 03086 B1 EE03086 B1 EE 03086B1
Authority
EE
Estonia
Prior art keywords
radical
formula
deoxy
fluorocytidines
oxycarbonyl
Prior art date
Application number
EE9400154A
Other languages
English (en)
Estonian (et)
Inventor
Arasaki Motohiro
Ishitsuka Hideo
Kuruma Isami
Miwa Masanori
Murasaki Chikako
Shimma Nobuo
Umeda Isao
Original Assignee
F. Hoffmann-La Roche Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8210304&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EE03086(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by F. Hoffmann-La Roche Ag filed Critical F. Hoffmann-La Roche Ag
Publication of EE03086B1 publication Critical patent/EE03086B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
EE9400154A 1992-12-18 1994-11-18 N4-(asendatud-oksükarbonüül)-5'-desoksü-5-fluorotsütidiinid, nende saamise meetod ja neid sisaldavad ravimpreparaadid EE03086B1 (et)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP92121538 1992-12-18

Publications (1)

Publication Number Publication Date
EE03086B1 true EE03086B1 (et) 1998-04-15

Family

ID=8210304

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9400154A EE03086B1 (et) 1992-12-18 1994-11-18 N4-(asendatud-oksükarbonüül)-5'-desoksü-5-fluorotsütidiinid, nende saamise meetod ja neid sisaldavad ravimpreparaadid

Country Status (41)

Country Link
US (1) US5472949A (ar)
EP (1) EP0602454B1 (ar)
JP (1) JP2501297B2 (ar)
KR (1) KR100347218B1 (ar)
CN (1) CN1035617C (ar)
AT (1) ATE137244T1 (ar)
AU (1) AU671491B2 (ar)
BG (1) BG61485B1 (ar)
BR (1) BR9305089A (ar)
CA (1) CA2103324C (ar)
CZ (1) CZ284788B6 (ar)
DE (1) DE69302360T2 (ar)
DK (1) DK0602454T3 (ar)
EE (1) EE03086B1 (ar)
ES (1) ES2086856T3 (ar)
FI (1) FI112365B (ar)
GE (1) GEP20074251B (ar)
GR (1) GR3020286T3 (ar)
HK (1) HK1005875A1 (ar)
HR (1) HRP931430B1 (ar)
HU (2) HU218291B (ar)
IL (1) IL108000A0 (ar)
IS (1) IS4108A (ar)
LT (1) LT3115B (ar)
LV (1) LV10625B (ar)
MY (1) MY109282A (ar)
NO (1) NO300066B1 (ar)
NZ (1) NZ250414A (ar)
PH (1) PH30168A (ar)
PL (1) PL174100B1 (ar)
RO (1) RO112619B1 (ar)
RU (2) RU2493162C1 (ar)
SA (1) SA93140409B1 (ar)
SI (1) SI9300648B (ar)
SK (1) SK281403B6 (ar)
SV (1) SV1993000080A (ar)
TW (1) TW372239B (ar)
UA (1) UA39158C2 (ar)
UY (1) UY23697A1 (ar)
YU (1) YU49411B (ar)
ZA (1) ZA939293B (ar)

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Also Published As

Publication number Publication date
ATE137244T1 (de) 1996-05-15
CN1035617C (zh) 1997-08-13
GEP20074251B (en) 2007-12-10
BG98304A (bg) 1994-01-03
IL108000A0 (en) 1994-04-12
EP0602454A1 (en) 1994-06-22
FI935616A0 (fi) 1993-12-14
HUT65757A (en) 1994-07-28
HU211965A9 (en) 1996-01-29
HU218291B (en) 2000-07-28
HU9303525D0 (en) 1994-04-28
LV10625B (en) 1996-04-20
CN1094056A (zh) 1994-10-26
LV10625A (lv) 1995-04-20
RU2135511C1 (ru) 1999-08-27
PL174100B1 (pl) 1998-06-30
SV1993000080A (es) 1996-01-26
SK144493A3 (en) 1994-10-05
TW372239B (en) 1999-10-21
BR9305089A (pt) 1994-07-05
KR940014428A (ko) 1994-07-18
MY109282A (en) 1996-12-31
SI9300648B (sl) 2000-06-30
FI935616A (fi) 1994-06-19
AU5069093A (en) 1994-06-30
RU2493162C1 (ru) 2013-09-20
ES2086856T3 (es) 1996-07-01
US5472949A (en) 1995-12-05
DE69302360T2 (de) 1996-10-31
YU77993A (sh) 1996-10-18
PH30168A (en) 1997-01-21
RO112619B1 (ro) 1997-11-28
NO934671D0 (no) 1993-12-17
IS4108A (is) 1994-06-19
YU49411B (sh) 2006-01-16
GR3020286T3 (en) 1996-09-30
CZ273193A3 (en) 1994-07-13
JPH06211891A (ja) 1994-08-02
UY23697A1 (es) 1994-06-08
CA2103324C (en) 1997-12-23
SA93140409B1 (ar) 2004-07-24
SK281403B6 (sk) 2001-03-12
FI112365B (fi) 2003-11-28
NO934671L (no) 1994-06-20
UA39158C2 (uk) 2001-06-15
PL301541A1 (en) 1994-06-27
JP2501297B2 (ja) 1996-05-29
AU671491B2 (en) 1996-08-29
HRP931430B1 (en) 1999-08-31
LTIP1627A (en) 1994-07-15
EP0602454B1 (en) 1996-04-24
HRP931430A2 (en) 1998-06-30
ZA939293B (en) 1994-06-18
CA2103324A1 (en) 1994-06-19
LT3115B (en) 1994-12-27
SI9300648A (en) 1994-09-30
DK0602454T3 (da) 1996-07-29
HK1005875A1 (en) 1999-01-29
NO300066B1 (no) 1997-04-01
RU2458932C2 (ru) 2012-08-20
CZ284788B6 (cs) 1999-03-17
DE69302360D1 (de) 1996-05-30
BG61485B1 (bg) 1997-09-30
NZ250414A (en) 1995-12-21
KR100347218B1 (ko) 2003-01-24

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