EA006317B1 - Производные хиназолина, содержащие эти соединения лекарственные средства, их применение и способ их получения - Google Patents

Производные хиназолина, содержащие эти соединения лекарственные средства, их применение и способ их получения Download PDF

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Publication number
EA006317B1
EA006317B1 EA200300671A EA200300671A EA006317B1 EA 006317 B1 EA006317 B1 EA 006317B1 EA 200300671 A EA200300671 A EA 200300671A EA 200300671 A EA200300671 A EA 200300671A EA 006317 B1 EA006317 B1 EA 006317B1
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EA
Eurasian Patent Office
Prior art keywords
amino
oxo
chloro
fluorophenyl
buten
Prior art date
Application number
EA200300671A
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English (en)
Russian (ru)
Other versions
EA200300671A1 (ru
Inventor
Франк Химмельсбах
Эльке Лангкопф
Штефан Блех
Биргит Юнг
Эльке Баум
Флавио Золька
Original Assignee
Бёрингер Ингельхайм Фарма Гмбх Унд Ко. Кг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7667887&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA006317(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Бёрингер Ингельхайм Фарма Гмбх Унд Ко. Кг filed Critical Бёрингер Ингельхайм Фарма Гмбх Унд Ко. Кг
Publication of EA200300671A1 publication Critical patent/EA200300671A1/ru
Publication of EA006317B1 publication Critical patent/EA006317B1/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
EA200300671A 2000-12-20 2001-12-12 Производные хиназолина, содержащие эти соединения лекарственные средства, их применение и способ их получения EA006317B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10063435A DE10063435A1 (de) 2000-12-20 2000-12-20 Chinazolinderviate,diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
PCT/EP2001/014569 WO2002050043A1 (de) 2000-12-20 2001-12-12 Chinazolinderivate, diese verbindungen enthaltende arzneimittel, deren verwendung und verfahren zu ihrer herstellung

Publications (2)

Publication Number Publication Date
EA200300671A1 EA200300671A1 (ru) 2004-06-24
EA006317B1 true EA006317B1 (ru) 2005-10-27

Family

ID=7667887

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200300671A EA006317B1 (ru) 2000-12-20 2001-12-12 Производные хиназолина, содержащие эти соединения лекарственные средства, их применение и способ их получения

Country Status (39)

Country Link
EP (2) EP2112140A1 (cg-RX-API-DMAC7.html)
JP (1) JP3827641B2 (cg-RX-API-DMAC7.html)
KR (1) KR100852102B1 (cg-RX-API-DMAC7.html)
CN (1) CN1277822C (cg-RX-API-DMAC7.html)
AR (1) AR040524A1 (cg-RX-API-DMAC7.html)
AT (1) ATE430136T1 (cg-RX-API-DMAC7.html)
AU (2) AU1917402A (cg-RX-API-DMAC7.html)
BE (1) BE2014C009I2 (cg-RX-API-DMAC7.html)
BG (1) BG66139B1 (cg-RX-API-DMAC7.html)
BR (1) BRPI0116266B8 (cg-RX-API-DMAC7.html)
CA (1) CA2432428C (cg-RX-API-DMAC7.html)
CY (2) CY1109290T1 (cg-RX-API-DMAC7.html)
CZ (1) CZ302721B6 (cg-RX-API-DMAC7.html)
DE (2) DE10063435A1 (cg-RX-API-DMAC7.html)
DK (1) DK1345910T3 (cg-RX-API-DMAC7.html)
EA (1) EA006317B1 (cg-RX-API-DMAC7.html)
EE (1) EE05244B1 (cg-RX-API-DMAC7.html)
ES (1) ES2326617T3 (cg-RX-API-DMAC7.html)
FR (1) FR14C0009I2 (cg-RX-API-DMAC7.html)
HR (1) HRP20030504B1 (cg-RX-API-DMAC7.html)
HU (2) HU228874B1 (cg-RX-API-DMAC7.html)
IL (2) IL156277A0 (cg-RX-API-DMAC7.html)
LT (1) LTC1345910I2 (cg-RX-API-DMAC7.html)
LU (1) LU92370I2 (cg-RX-API-DMAC7.html)
ME (1) ME02777B (cg-RX-API-DMAC7.html)
MX (1) MXPA03005559A (cg-RX-API-DMAC7.html)
MY (1) MY136086A (cg-RX-API-DMAC7.html)
NO (3) NO325672B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ526918A (cg-RX-API-DMAC7.html)
PL (1) PL214798B1 (cg-RX-API-DMAC7.html)
PT (1) PT1345910E (cg-RX-API-DMAC7.html)
RS (1) RS50860B (cg-RX-API-DMAC7.html)
SI (1) SI1345910T1 (cg-RX-API-DMAC7.html)
SK (1) SK287573B6 (cg-RX-API-DMAC7.html)
TW (1) TWI295992B (cg-RX-API-DMAC7.html)
UA (1) UA74614C2 (cg-RX-API-DMAC7.html)
UY (1) UY27078A1 (cg-RX-API-DMAC7.html)
WO (1) WO2002050043A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA200304141B (cg-RX-API-DMAC7.html)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2720810C2 (ru) * 2015-03-20 2020-05-13 Чиа Тай Тяньцин Фармасьютикал Груп Ко., Лтд. Соли производного хиназолина и способ их получения

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