DOP2001000271A - Compuestos de imidazol condensado con arilo o heteroarilo como agentes antiinflamatorios y analgésicos. - Google Patents

Compuestos de imidazol condensado con arilo o heteroarilo como agentes antiinflamatorios y analgésicos.

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Publication number
DOP2001000271A
DOP2001000271A DO2001000271A DO2001000271A DOP2001000271A DO P2001000271 A DOP2001000271 A DO P2001000271A DO 2001000271 A DO2001000271 A DO 2001000271A DO 2001000271 A DO2001000271 A DO 2001000271A DO P2001000271 A DOP2001000271 A DO P2001000271A
Authority
DO
Dominican Republic
Prior art keywords
alkyl
membered monocyclic
aromatic ring
heteroatoms selected
optionally contains
Prior art date
Application number
DO2001000271A
Other languages
English (en)
Spanish (es)
Inventor
Kazunari Nakao
Yoshiyuki Okumura
Seiji Nukui
Miyako Matsumizu
Naomi UENO
Yoshinobu Hashizumo
Tomoki Kato
Akiyoshi Kawai
Katsuhiro Shinjyo
Kana Taniguchi
Yoriko Miyake
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DOP2001000271A publication Critical patent/DOP2001000271A/es

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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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