PL365781A1 - Ep4 receptor inhibitors to treat rheumatoid arthritis - Google Patents

Ep4 receptor inhibitors to treat rheumatoid arthritis

Info

Publication number
PL365781A1
PL365781A1 PL01365781A PL36578101A PL365781A1 PL 365781 A1 PL365781 A1 PL 365781A1 PL 01365781 A PL01365781 A PL 01365781A PL 36578101 A PL36578101 A PL 36578101A PL 365781 A1 PL365781 A1 PL 365781A1
Authority
PL
Poland
Prior art keywords
rheumatoid arthritis
receptor inhibitors
treat rheumatoid
treat
inhibitors
Prior art date
Application number
PL01365781A
Other languages
English (en)
Polish (pl)
Inventor
Laurent Pascal Audoly
Takako Okumura
Masato Shimojo
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of PL365781A1 publication Critical patent/PL365781A1/xx

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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