DK575887A - Pyridinderivater med anti-ulcer aktivitet - Google Patents

Pyridinderivater med anti-ulcer aktivitet

Info

Publication number
DK575887A
DK575887A DK575887A DK575887A DK575887A DK 575887 A DK575887 A DK 575887A DK 575887 A DK575887 A DK 575887A DK 575887 A DK575887 A DK 575887A DK 575887 A DK575887 A DK 575887A
Authority
DK
Denmark
Prior art keywords
group
stands
alkoxy
alkyl
integer
Prior art date
Application number
DK575887A
Other languages
English (en)
Other versions
DK575887D0 (da
DK171024B1 (da
Inventor
Shigeru Souda
Norihiro Ueda
Shuhei Miyazawa
Katsuya Tagami
Seiichiro Nomoto
Makoto Okita
Naoyuki Shimomura
Toshihiko Kaneko
Masatoshi Fujimoto
Manabu Murakami
Kiyoshi Oketani
Hideaki Fujisaki
Hisashi Shibata
Tsuneo Wakabayashi
Original Assignee
Eisai Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27283658&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK575887(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd
Publication of DK575887D0 publication Critical patent/DK575887D0/da
Publication of DK575887A publication Critical patent/DK575887A/da
Priority to DK199501442A priority Critical patent/DK174366B1/da
Application granted granted Critical
Publication of DK171024B1 publication Critical patent/DK171024B1/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
DK575887A 1986-11-13 1987-11-03 2-(4-(3-Methoxypropoxy)-3-methylpyridin-2-yl)methylsulfinyl-1H-benzimidazol eller salte deraf, farmaceutisk præparat med et indhold deraf samt anvendelse deraf til fremstilling af et præparat til behandling eller forebyggelse af mavesår DK171024B1 (da)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DK199501442A DK174366B1 (da) 1986-11-13 1995-12-19 2-(substitueret methyl) -3-alkyl-4-(substitueret ethoxy)-pyridinforbindelser, farmaceutisk præparat, som indeholder en sådan, samt anvendelse af en sådan til fremstilling af et farmaceutisk præparat til behandling eller forebyggelse af mavesår

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
JP27053686 1986-11-13
JP27053686 1986-11-13
JP2198987 1987-02-02
JP2198987 1987-02-02
JP7778487 1987-03-31
JP7778487 1987-03-31

Publications (3)

Publication Number Publication Date
DK575887D0 DK575887D0 (da) 1987-11-03
DK575887A true DK575887A (da) 1988-05-14
DK171024B1 DK171024B1 (da) 1996-04-22

Family

ID=27283658

Family Applications (2)

Application Number Title Priority Date Filing Date
DK575887A DK171024B1 (da) 1986-11-13 1987-11-03 2-(4-(3-Methoxypropoxy)-3-methylpyridin-2-yl)methylsulfinyl-1H-benzimidazol eller salte deraf, farmaceutisk præparat med et indhold deraf samt anvendelse deraf til fremstilling af et præparat til behandling eller forebyggelse af mavesår
DK131893A DK131893A (da) 1986-11-13 1993-11-24 2-(Substitueret methyl)-4-(substitueret ethoxy)-5-(lavere alkyl)-pyridinforbindelser, farmaceutisk præparat, som indeholder sådanne samt anvendelse af en sådan forbindelse til fremstilling af et farmaceutisk præparat

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK131893A DK131893A (da) 1986-11-13 1993-11-24 2-(Substitueret methyl)-4-(substitueret ethoxy)-5-(lavere alkyl)-pyridinforbindelser, farmaceutisk præparat, som indeholder sådanne samt anvendelse af en sådan forbindelse til fremstilling af et farmaceutisk præparat

Country Status (18)

Country Link
US (3) US5045552A (da)
EP (3) EP0268956B2 (da)
JP (1) JP2544567B2 (da)
KR (1) KR910003330B1 (da)
CN (1) CN1018923B (da)
AT (2) ATE163011T1 (da)
AU (1) AU594836B2 (da)
CA (1) CA1265138A (da)
DE (4) DE3789536T3 (da)
DK (2) DK171024B1 (da)
ES (3) ES2118457T3 (da)
FI (1) FI90544C (da)
HK (1) HK194296A (da)
HU (1) HU198475B (da)
LU (1) LU90396I2 (da)
NL (1) NL990015I2 (da)
NO (2) NO170932C (da)
NZ (1) NZ222488A (da)

Families Citing this family (152)

* Cited by examiner, † Cited by third party
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EP0268956A2 (en) 1988-06-01
CN1018923B (zh) 1992-11-04
KR910003330B1 (ko) 1991-05-27
NL990015I1 (nl) 1999-08-02
ATE168111T1 (de) 1998-07-15
NL990015I2 (nl) 1999-09-01
EP0268956A3 (en) 1990-07-25
JPH05247035A (ja) 1993-09-24
JP2544567B2 (ja) 1996-10-16
DK131893D0 (da) 1993-11-24
EP0268956B2 (en) 1998-04-15
FI874709A0 (fi) 1987-10-26
EP0654471A1 (en) 1995-05-24
DE3789536T3 (de) 1998-08-20
ES2112260T3 (es) 1998-04-01
ES2061471T5 (es) 1998-07-16
ES2061471T3 (es) 1994-12-16
CA1265138A (en) 1990-01-30
DE3752201T2 (de) 1998-12-17
DK575887D0 (da) 1987-11-03
ATE163011T1 (de) 1998-02-15
KR880006229A (ko) 1988-07-22
CN87107777A (zh) 1988-06-01
HUT45524A (en) 1988-07-28
NO874477L (no) 1988-05-16
DE3789536D1 (de) 1994-05-11
US5998445A (en) 1999-12-07
NO170932B (no) 1992-09-21
EP0268956B1 (en) 1994-04-06
HU198475B (en) 1989-10-30
NO874477D0 (no) 1987-10-27
EP0475456B1 (en) 1998-02-04
EP0654471B1 (en) 1998-07-08
NO170932C (no) 1992-12-30
DE19975035I2 (de) 2004-01-29
ES2118457T3 (es) 1998-09-16
FI874709A (fi) 1988-05-14
DE3752167T2 (de) 1998-06-25
US5840910A (en) 1998-11-24
AU8113887A (en) 1988-05-19
AU594836B2 (en) 1990-03-15
NZ222488A (en) 1993-05-26
EP0475456A1 (en) 1992-03-18
US5045552A (en) 1991-09-03
DE3752167D1 (de) 1998-03-12
DK131893A (da) 1993-11-24
FI90544B (fi) 1993-11-15
HK194296A (en) 1996-11-01
DK171024B1 (da) 1996-04-22
DE3789536T2 (de) 1994-08-18
DE3752201D1 (de) 1998-08-13
FI90544C (fi) 1994-02-25
NO2000006I1 (no) 2000-09-18
LU90396I2 (fr) 1999-07-07

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