DK1888614T3 - Fremgangsmåde til fremstilling af 3alpha(beta)-7alpha(beta)-dihydroxy-6alpha(beta)-alkyl-5beta-cholansyre - Google Patents

Fremgangsmåde til fremstilling af 3alpha(beta)-7alpha(beta)-dihydroxy-6alpha(beta)-alkyl-5beta-cholansyre

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Publication number
DK1888614T3
DK1888614T3 DK06763188.7T DK06763188T DK1888614T3 DK 1888614 T3 DK1888614 T3 DK 1888614T3 DK 06763188 T DK06763188 T DK 06763188T DK 1888614 T3 DK1888614 T3 DK 1888614T3
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Prior art keywords
beta
alkyl
dihydroxy
5beta
6alpha
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DK06763188.7T
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English (en)
Inventor
Massimo Ferrari
Roberto Pellicciari
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Erregierre Spa
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Publication of DK1888614T3 publication Critical patent/DK1888614T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • C07J9/005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Seasonings (AREA)
DK06763188.7T 2005-05-19 2006-05-19 Fremgangsmåde til fremstilling af 3alpha(beta)-7alpha(beta)-dihydroxy-6alpha(beta)-alkyl-5beta-cholansyre DK1888614T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT000912A ITMI20050912A1 (it) 2005-05-19 2005-05-19 Processo di preparazione di acidi 3-a-ya(b)-diidrossi-6-a(b)-alchil-5b-colanici
PCT/EP2006/062446 WO2006122977A2 (en) 2005-05-19 2006-05-19 PROCESS FOR PREPARING 3α(β)-7α(β)-DIHYDROXY-6α(β)-ALKYL-5β-CHOLANIC ACID

Publications (1)

Publication Number Publication Date
DK1888614T3 true DK1888614T3 (da) 2010-05-10

Family

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DK06763188.7T DK1888614T3 (da) 2005-05-19 2006-05-19 Fremgangsmåde til fremstilling af 3alpha(beta)-7alpha(beta)-dihydroxy-6alpha(beta)-alkyl-5beta-cholansyre

Country Status (12)

Country Link
US (1) US7994352B2 (da)
EP (1) EP1888614B1 (da)
JP (1) JP5127700B2 (da)
CN (1) CN101203526B (da)
AT (1) ATE453657T1 (da)
AU (1) AU2006248906B2 (da)
CA (1) CA2608539C (da)
DE (1) DE602006011457D1 (da)
DK (1) DK1888614T3 (da)
ES (1) ES2338698T3 (da)
IT (1) ITMI20050912A1 (da)
WO (1) WO2006122977A2 (da)

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CA2608539C (en) 2013-02-26
EP1888614A2 (en) 2008-02-20
AU2006248906A1 (en) 2006-11-23
ITMI20050912A1 (it) 2006-11-20
ES2338698T3 (es) 2010-05-11
CA2608539A1 (en) 2006-11-23
EP1888614B1 (en) 2009-12-30
CN101203526A (zh) 2008-06-18
US7994352B2 (en) 2011-08-09
DE602006011457D1 (de) 2010-02-11
WO2006122977A3 (en) 2007-01-18
ATE453657T1 (de) 2010-01-15
JP5127700B2 (ja) 2013-01-23
CN101203526B (zh) 2012-09-05
WO2006122977A2 (en) 2006-11-23
JP2008540612A (ja) 2008-11-20
AU2006248906B2 (en) 2012-04-12

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