CY1109911T1 - Πυρρολοβενζοδιαζεπινες - Google Patents

Πυρρολοβενζοδιαζεπινες

Info

Publication number
CY1109911T1
CY1109911T1 CY20101100248T CY101100248T CY1109911T1 CY 1109911 T1 CY1109911 T1 CY 1109911T1 CY 20101100248 T CY20101100248 T CY 20101100248T CY 101100248 T CY101100248 T CY 101100248T CY 1109911 T1 CY1109911 T1 CY 1109911T1
Authority
CY
Cyprus
Prior art keywords
pyrrolovenzodiazepines
compounds
formula
Prior art date
Application number
CY20101100248T
Other languages
English (en)
Inventor
Stephen J Gregson
Zhizhi Chen
Philip Wilson Howard
Original Assignee
Spirogen Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0508084A external-priority patent/GB0508084D0/en
Priority claimed from GB0522746A external-priority patent/GB0522746D0/en
Application filed by Spirogen Limited filed Critical Spirogen Limited
Publication of CY1109911T1 publication Critical patent/CY1109911T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
    • A61K31/5517—1,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/04—Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Ενώσεις του τύπου: (I)
CY20101100248T 2005-04-21 2010-03-18 Πυρρολοβενζοδιαζεπινες CY1109911T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0508084A GB0508084D0 (en) 2005-04-21 2005-04-21 Pyrrolobenzodiazepines
GB0522746A GB0522746D0 (en) 2005-11-07 2005-11-07 Pyrrolobenzodiazepines
EP06726846A EP1879901B1 (en) 2005-04-21 2006-04-21 Pyrrolobenzodiazepines

Publications (1)

Publication Number Publication Date
CY1109911T1 true CY1109911T1 (el) 2014-09-10

Family

ID=36589321

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20101100248T CY1109911T1 (el) 2005-04-21 2010-03-18 Πυρρολοβενζοδιαζεπινες

Country Status (19)

Country Link
US (2) US7612062B2 (el)
EP (1) EP1879901B1 (el)
JP (1) JP5061096B2 (el)
KR (1) KR101396095B1 (el)
AT (1) ATE452898T1 (el)
AU (1) AU2006238686B2 (el)
BR (1) BRPI0610284A8 (el)
CA (1) CA2604805C (el)
CY (1) CY1109911T1 (el)
DE (1) DE602006011300D1 (el)
DK (1) DK1879901T3 (el)
ES (1) ES2338696T3 (el)
GB (1) GB2439881C (el)
MX (1) MX2007013039A (el)
NZ (1) NZ563136A (el)
PL (1) PL1879901T3 (el)
PT (1) PT1879901E (el)
SI (1) SI1879901T1 (el)
WO (1) WO2006111759A1 (el)

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EP1879901A1 (en) 2008-01-23
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KR101396095B1 (ko) 2014-05-15
BRPI0610284A8 (pt) 2017-05-09
US7612062B2 (en) 2009-11-03
GB2439881A (en) 2008-01-09
GB2439881C (en) 2011-08-10
JP5061096B2 (ja) 2012-10-31
ES2338696T3 (es) 2010-05-11
GB2439881B (en) 2009-04-08
WO2006111759A1 (en) 2006-10-26
DE602006011300D1 (de) 2010-02-04
BRPI0610284A2 (pt) 2010-06-08
ATE452898T1 (de) 2010-01-15
PT1879901E (pt) 2010-03-29
DK1879901T3 (da) 2010-05-03
AU2006238686B2 (en) 2011-10-06
CA2604805C (en) 2014-05-27
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MX2007013039A (es) 2008-03-13
GB0720721D0 (en) 2007-12-05
US8633185B2 (en) 2014-01-21
AU2006238686A1 (en) 2006-10-26
PL1879901T3 (pl) 2010-06-30
SI1879901T1 (sl) 2010-04-30
US20100113425A1 (en) 2010-05-06
US20080167293A1 (en) 2008-07-10
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CA2604805A1 (en) 2006-10-26

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