ATE453657T1 - Verfahren zur herstellung von 3alpha(beta)- - Google Patents

Verfahren zur herstellung von 3alpha(beta)-

Info

Publication number
ATE453657T1
ATE453657T1 AT06763188T AT06763188T ATE453657T1 AT E453657 T1 ATE453657 T1 AT E453657T1 AT 06763188 T AT06763188 T AT 06763188T AT 06763188 T AT06763188 T AT 06763188T AT E453657 T1 ATE453657 T1 AT E453657T1
Authority
AT
Austria
Prior art keywords
3alpha
beta
producing
alkyl
cholanic
Prior art date
Application number
AT06763188T
Other languages
English (en)
Inventor
Massimo Ferrari
Roberto Pellicciari
Original Assignee
Erregierre Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erregierre Spa filed Critical Erregierre Spa
Application granted granted Critical
Publication of ATE453657T1 publication Critical patent/ATE453657T1/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • C07J9/005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Steroid Compounds (AREA)
  • Seasonings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
AT06763188T 2005-05-19 2006-05-19 Verfahren zur herstellung von 3alpha(beta)- ATE453657T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT000912A ITMI20050912A1 (it) 2005-05-19 2005-05-19 Processo di preparazione di acidi 3-a-ya(b)-diidrossi-6-a(b)-alchil-5b-colanici
PCT/EP2006/062446 WO2006122977A2 (en) 2005-05-19 2006-05-19 PROCESS FOR PREPARING 3α(β)-7α(β)-DIHYDROXY-6α(β)-ALKYL-5β-CHOLANIC ACID

Publications (1)

Publication Number Publication Date
ATE453657T1 true ATE453657T1 (de) 2010-01-15

Family

ID=35841713

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06763188T ATE453657T1 (de) 2005-05-19 2006-05-19 Verfahren zur herstellung von 3alpha(beta)-

Country Status (12)

Country Link
US (1) US7994352B2 (de)
EP (1) EP1888614B1 (de)
JP (1) JP5127700B2 (de)
CN (1) CN101203526B (de)
AT (1) ATE453657T1 (de)
AU (1) AU2006248906B2 (de)
CA (1) CA2608539C (de)
DE (1) DE602006011457D1 (de)
DK (1) DK1888614T3 (de)
ES (1) ES2338698T3 (de)
IT (1) ITMI20050912A1 (de)
WO (1) WO2006122977A2 (de)

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EP1888614B1 (de) 2009-12-30
EP1888614A2 (de) 2008-02-20
DE602006011457D1 (de) 2010-02-11
JP2008540612A (ja) 2008-11-20
ES2338698T3 (es) 2010-05-11
US7994352B2 (en) 2011-08-09
WO2006122977A2 (en) 2006-11-23
DK1888614T3 (da) 2010-05-10
CA2608539C (en) 2013-02-26
WO2006122977A3 (en) 2007-01-18
ITMI20050912A1 (it) 2006-11-20
AU2006248906B2 (en) 2012-04-12
CN101203526B (zh) 2012-09-05
AU2006248906A1 (en) 2006-11-23
CA2608539A1 (en) 2006-11-23
US20080214515A1 (en) 2008-09-04
JP5127700B2 (ja) 2013-01-23
CN101203526A (zh) 2008-06-18

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