DK0513200T3 - Fremgangsmåde og sammensætninger til syntese af BCH-189 og beslægtede forbindelser - Google Patents
Fremgangsmåde og sammensætninger til syntese af BCH-189 og beslægtede forbindelserInfo
- Publication number
- DK0513200T3 DK0513200T3 DK91904454T DK91904454T DK0513200T3 DK 0513200 T3 DK0513200 T3 DK 0513200T3 DK 91904454 T DK91904454 T DK 91904454T DK 91904454 T DK91904454 T DK 91904454T DK 0513200 T3 DK0513200 T3 DK 0513200T3
- Authority
- DK
- Denmark
- Prior art keywords
- bch
- related compounds
- synthesis
- compositions
- methods
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D327/00—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
- C07D327/02—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
- C07D327/04—Five-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
- C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D411/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/06—Pyrimidine radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/06—Pyrimidine radicals
- C07H19/10—Pyrimidine radicals with the saccharide radical esterified by phosphoric or polyphosphoric acids
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/473,318 US5204466A (en) | 1990-02-01 | 1990-02-01 | Method and compositions for the synthesis of bch-189 and related compounds |
PCT/US1991/000685 WO1991011186A1 (en) | 1990-02-01 | 1991-01-31 | Method and compositions for the synthesis of bch-189 and related compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
DK0513200T3 true DK0513200T3 (da) | 1999-05-25 |
DK0513200T4 DK0513200T4 (da) | 2004-07-05 |
Family
ID=23879071
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK91904454T DK0513200T4 (da) | 1990-02-01 | 1991-01-31 | Fremgangsmåde og sammensætninger til syntese af BCH-189 og beslægtede forbindelser |
DK98201737T DK0872237T3 (da) | 1990-02-01 | 1991-01-31 | Fremgangsmåde og sammensætninger til syntese af BCH-189 og beslægtede forbindelser |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK98201737T DK0872237T3 (da) | 1990-02-01 | 1991-01-31 | Fremgangsmåde og sammensætninger til syntese af BCH-189 og beslægtede forbindelser |
Country Status (22)
Country | Link |
---|---|
US (8) | US5204466A (da) |
EP (3) | EP1772151A3 (da) |
JP (6) | JPH07618B2 (da) |
KR (2) | KR100381705B1 (da) |
AT (1) | ATE170750T1 (da) |
AU (6) | AU658136C (da) |
BG (1) | BG62236B1 (da) |
CA (3) | CA2678778A1 (da) |
DE (4) | DE69133556T2 (da) |
DK (2) | DK0513200T4 (da) |
ES (2) | ES2076130T5 (da) |
FI (4) | FI114471B (da) |
GR (1) | GR950300024T1 (da) |
HK (1) | HK1014664A1 (da) |
HU (4) | HU9202496D0 (da) |
LU (1) | LU91073I2 (da) |
MC (1) | MC2233A1 (da) |
NL (1) | NL300148I2 (da) |
NO (6) | NO923014L (da) |
RO (1) | RO108564B1 (da) |
RU (1) | RU2125558C1 (da) |
WO (1) | WO1991011186A1 (da) |
Families Citing this family (150)
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US5925643A (en) * | 1990-12-05 | 1999-07-20 | Emory University | Enantiomerically pure β-D-dioxolane-nucleosides |
IL100502A (en) * | 1991-01-03 | 1995-12-08 | Iaf Biochem Int | PHARMACEUTICAL PREPARATIONS CONTAINING CIS-4-AMINO-1-) 2-HYDROXIMETHIL-1,3-OXETYOLEN-5-IL (- |
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GB9104740D0 (en) * | 1991-03-06 | 1991-04-17 | Wellcome Found | Antiviral nucleoside combination |
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