CN110291087B - 作为雌激素受体降解剂的四氢萘和四氢异喹啉衍生物 - Google Patents

作为雌激素受体降解剂的四氢萘和四氢异喹啉衍生物 Download PDF

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CN110291087B
CN110291087B CN201780085150.9A CN201780085150A CN110291087B CN 110291087 B CN110291087 B CN 110291087B CN 201780085150 A CN201780085150 A CN 201780085150A CN 110291087 B CN110291087 B CN 110291087B
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CN110291087A (zh
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安德鲁·P·克鲁
Y·钱
H·董
J·王
基思·R·霍恩伯格
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Arvinas Inc
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Priority to CN202210386845.3A priority patent/CN114656452B/zh
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CN201780085150.9A 2016-12-01 2017-12-01 作为雌激素受体降解剂的四氢萘和四氢异喹啉衍生物 Active CN110291087B (zh)

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Application Number Priority Date Filing Date Title
CN202010214256.8A CN111454248A (zh) 2016-12-01 2017-12-01 作为雌激素受体降解剂的四氢萘和四氢异喹啉衍生物
CN202410799699.6A CN118834201A (zh) 2016-12-01 2017-12-01 作为雌激素受体降解剂的四氢萘和四氢异喹啉衍生物
CN202210386845.3A CN114656452B (zh) 2016-12-01 2017-12-01 作为雌激素受体降解剂的四氢萘和四氢异喹啉衍生物

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US201662429041P 2016-12-01 2016-12-01
US62/429,041 2016-12-01
US201762540049P 2017-08-01 2017-08-01
US62/540,049 2017-08-01
PCT/US2017/064283 WO2018102725A1 (en) 2016-12-01 2017-12-01 Tetrahydronaphthalene and tetrahydroisoquinoline derivatives as estrogen receptor degraders

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