CN103432133B - 核受体结合剂的用途 - Google Patents

核受体结合剂的用途 Download PDF

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Publication number
CN103432133B
CN103432133B CN201310311031.4A CN201310311031A CN103432133B CN 103432133 B CN103432133 B CN 103432133B CN 201310311031 A CN201310311031 A CN 201310311031A CN 103432133 B CN103432133 B CN 103432133B
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another embodiment
heterocycle
compound
alkyl
present
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CN103432133A (zh
Inventor
J·T·多尔顿
D·D·米勒
M·L·莫勒
Z·吴
S-S·洪
D·斯里瓦斯塔瓦
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Oncternal Therapeutics Inc
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GTx Inc
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
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    • C07D217/24—Oxygen atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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CN201310311031.4A 2007-01-22 2008-01-22 核受体结合剂的用途 Expired - Fee Related CN103432133B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US88147607P 2007-01-22 2007-01-22
US60/881,476 2007-01-22
US90775407P 2007-04-16 2007-04-16
US60/907,754 2007-04-16
CN200880009379.5A CN101641013B (zh) 2007-01-22 2008-01-22 核受体结合剂

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CN103432133A CN103432133A (zh) 2013-12-11
CN103432133B true CN103432133B (zh) 2016-08-10

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CN201310311031.4A Expired - Fee Related CN103432133B (zh) 2007-01-22 2008-01-22 核受体结合剂的用途

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US (1) US9078888B2 (no)
EP (2) EP2106212B1 (no)
JP (4) JP5484914B2 (no)
KR (3) KR20160020584A (no)
CN (2) CN101641013B (no)
AU (1) AU2008209581B2 (no)
BR (1) BRPI0806371A2 (no)
CA (1) CA2676066C (no)
EA (3) EA201692214A1 (no)
ES (1) ES2475193T3 (no)
IL (2) IL199996A (no)
IS (1) IS8842A (no)
MX (1) MX2009007831A (no)
NO (1) NO20092822L (no)
WO (1) WO2008091555A2 (no)

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