CN103180326B - 杂环化合物及其用途 - Google Patents

杂环化合物及其用途 Download PDF

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Publication number
CN103180326B
CN103180326B CN201180048970.3A CN201180048970A CN103180326B CN 103180326 B CN103180326 B CN 103180326B CN 201180048970 A CN201180048970 A CN 201180048970A CN 103180326 B CN103180326 B CN 103180326B
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halogen atom
optionally substituted
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CN103180326A (zh
Inventor
郡正城
今枝稔博
中村信二
丰福昌志
本多荣治
浅野恭臣
宇治川治
望月伦代
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Takeda Pharmaceutical Co Ltd
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Epidemiology (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
CN201180048970.3A 2010-08-10 2011-08-09 杂环化合物及其用途 Active CN103180326B (zh)

Priority Applications (1)

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CN201510259936.0A CN104926837A (zh) 2010-08-10 2011-08-09 杂环化合物及其用途

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JP2010179577 2010-08-10
JP2010-179577 2010-08-10
PCT/JP2011/068497 WO2012020848A1 (en) 2010-08-10 2011-08-09 Heterocyclic compound and use thereof

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CN103180326B true CN103180326B (zh) 2015-06-10

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CN107709310B (zh) 2015-06-02 2021-09-24 Fmc公司 取代的环酰胺及其作为除草剂的用途
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RU2019122791A (ru) 2016-12-21 2021-01-25 Фмк Корпорейшн Гербициды на основе нитрона
CN107892697B (zh) 2016-12-26 2020-11-03 郑州泰基鸿诺医药股份有限公司 一种[1,3]噻嗪-2-胺类化合物及应用,药物组合物
MX2019010969A (es) 2017-03-21 2019-12-02 Fmc Corp Pirrolidinonas y proceso para prepararlas.
CN110740646B (zh) 2017-03-21 2022-05-10 Fmc公司 除草剂混合物、组合物和方法
AR111967A1 (es) 2017-05-30 2019-09-04 Fmc Corp Amidas herbicidas
AR111839A1 (es) 2017-05-30 2019-08-21 Fmc Corp Lactamas 3-sustituidas herbicidas
ES2970624T3 (es) 2017-10-06 2024-05-29 Takeda Pharmaceuticals Co Compuesto heterocíclico
EP3693360B1 (en) * 2017-10-06 2023-12-13 Takeda Pharmaceutical Company Limited Heterocyclic compounds
AU2020348675B2 (en) 2019-09-16 2025-11-20 Takeda Pharmaceutical Company Limited Azole-fused pyridazin-3(2H)-one derivatives
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CN113943294A (zh) * 2020-07-15 2022-01-18 成都海博为药业有限公司 一种作为btk抑制剂的化合物及其制备方法与用途
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MA34509B1 (fr) 2013-09-02
US8916551B2 (en) 2014-12-23
CN104926837A (zh) 2015-09-23
CA2807460A1 (en) 2012-02-16
RS60311B1 (sr) 2020-07-31
CR20130066A (es) 2013-05-03
JP2016006080A (ja) 2016-01-14
GEP20156216B (en) 2015-01-12
CN103180326A (zh) 2013-06-26
UY33551A (es) 2012-03-30
MX349470B (es) 2017-07-31
US9150591B2 (en) 2015-10-06
CL2013000380A1 (es) 2013-05-31
US20240360156A1 (en) 2024-10-31
ES2793723T3 (es) 2020-11-16
KR20130138738A (ko) 2013-12-19
NZ607593A (en) 2015-01-30
JP5788496B2 (ja) 2015-09-30
PT2603513T (pt) 2020-06-08
MX2013001614A (es) 2013-07-05
US8778934B2 (en) 2014-07-15
SI2603513T1 (sl) 2020-07-31
UA111594C2 (uk) 2016-05-25
DOP2013000030A (es) 2013-03-15
US20140080817A1 (en) 2014-03-20
TW201217386A (en) 2012-05-01
ZA201301120B (en) 2014-04-30
AR082618A1 (es) 2012-12-19
AU2011290126A1 (en) 2013-03-07
JP6113789B2 (ja) 2017-04-12
AU2011290126B2 (en) 2016-01-07
CA2807460C (en) 2018-09-18
PH12013500247A1 (en) 2013-03-11
HUE049460T2 (hu) 2020-09-28
DK2603513T3 (da) 2020-06-15
WO2012020848A8 (en) 2012-09-27
US20180162875A1 (en) 2018-06-14
US11279713B2 (en) 2022-03-22
US10654874B2 (en) 2020-05-19
ECSP13012478A (es) 2013-04-30
MY165908A (en) 2018-05-18
EA201390222A1 (ru) 2013-08-30
LT2603513T (lt) 2020-05-25
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EP2603513B1 (en) 2020-03-11
JP2013535408A (ja) 2013-09-12
CO6680700A2 (es) 2013-05-31
US8575154B2 (en) 2013-11-05
US20130190291A1 (en) 2013-07-25
US20190263832A1 (en) 2019-08-29
PL2603513T3 (pl) 2020-07-27
US20150073137A1 (en) 2015-03-12
US20120077799A1 (en) 2012-03-29
US20200317692A1 (en) 2020-10-08
BR112013002250A2 (pt) 2016-05-24
US20170022222A1 (en) 2017-01-26
US9499568B2 (en) 2016-11-22
US9884875B2 (en) 2018-02-06
CY1123507T1 (el) 2022-03-24
US20130184266A1 (en) 2013-07-18
PE20131116A1 (es) 2013-10-24
EA022078B1 (ru) 2015-10-30
WO2012020848A1 (en) 2012-02-16
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IL224452A (en) 2017-11-30
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