CN101801383A - 用于治疗骨髓增生性疾病和其他增生性疾病的激酶抑制剂 - Google Patents
用于治疗骨髓增生性疾病和其他增生性疾病的激酶抑制剂 Download PDFInfo
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- CN101801383A CN101801383A CN200880020714A CN200880020714A CN101801383A CN 101801383 A CN101801383 A CN 101801383A CN 200880020714 A CN200880020714 A CN 200880020714A CN 200880020714 A CN200880020714 A CN 200880020714A CN 101801383 A CN101801383 A CN 101801383A
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Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US91321607P | 2007-04-20 | 2007-04-20 | |
| US60/913,216 | 2007-04-20 | ||
| PCT/US2008/060833 WO2008131227A1 (en) | 2007-04-20 | 2008-04-18 | Kinase inhibitors useful for the treatment of myleoproliferative diseases and other proliferative diseases |
Publications (1)
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| CN101801383A true CN101801383A (zh) | 2010-08-11 |
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| CN200880020714A Pending CN101801383A (zh) | 2007-04-20 | 2008-04-18 | 用于治疗骨髓增生性疾病和其他增生性疾病的激酶抑制剂 |
| CN2008800085252A Pending CN101878031A (zh) | 2007-04-20 | 2008-04-18 | 用于治疗骨髓增生性疾病和其他增生性疾病的激酶抑制剂 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
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| CN2008800085252A Pending CN101878031A (zh) | 2007-04-20 | 2008-04-18 | 用于治疗骨髓增生性疾病和其他增生性疾病的激酶抑制剂 |
Country Status (14)
| Country | Link |
|---|---|
| US (4) | US20080269254A1 (enExample) |
| EP (5) | EP2148677A4 (enExample) |
| JP (2) | JP2010524970A (enExample) |
| KR (2) | KR20100017184A (enExample) |
| CN (2) | CN101801383A (enExample) |
| AU (4) | AU2008242697A1 (enExample) |
| BR (2) | BRPI0807717A2 (enExample) |
| CA (4) | CA2684950A1 (enExample) |
| EA (1) | EA200970700A1 (enExample) |
| IL (1) | IL201650A0 (enExample) |
| MX (2) | MX2009009066A (enExample) |
| RU (1) | RU2009142851A (enExample) |
| SG (1) | SG183054A1 (enExample) |
| WO (4) | WO2008140895A1 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| CN102408408A (zh) * | 2010-09-20 | 2012-04-11 | 北大方正集团有限公司 | 具有抗肿瘤作用的芳基脲衍生物 |
| CN102432592A (zh) * | 2010-09-29 | 2012-05-02 | 北大方正集团有限公司 | 具有抗肿瘤作用的芳基脲衍生物及其制备方法 |
| CN102532113A (zh) * | 2010-12-22 | 2012-07-04 | 北大方正集团有限公司 | 芳基脲衍生物 |
| CN102558144A (zh) * | 2010-12-22 | 2012-07-11 | 北大方正集团有限公司 | 一种芳基脲衍生物 |
| CN104974132A (zh) * | 2014-04-08 | 2015-10-14 | 北大方正集团有限公司 | 多取代的吡啶化合物、制备方法、用途及药物组合物 |
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| WO2018137610A1 (zh) * | 2017-01-24 | 2018-08-02 | 四川大学 | 取代的1-(异恶唑-3-基)-3-(3-氟-4-苯基)脲衍生物及其制备方法和用途 |
| CN108341813B (zh) * | 2017-01-24 | 2020-11-17 | 四川大学 | 取代的1-(异恶唑-3-基)-3-(3-氟-4-苯基)脲衍生物及其制备方法和用途 |
| CN111936484A (zh) * | 2017-12-22 | 2020-11-13 | 拉文纳制药公司 | 作为磷脂酰肌醇磷酸激酶抑制剂的色烯并吡啶衍生物 |
| US11584763B2 (en) | 2017-12-22 | 2023-02-21 | Hibercell, Inc. | Chromenopyridine derivatives as phosphatidylinositol phosphate kinase inhibitors |
| CN113507964A (zh) * | 2019-03-06 | 2021-10-15 | 马里兰大学,巴尔的摩 | 作为用于治疗癌症和其他疾病的治疗性肽的纳米载体的四聚体蛋白质支架 |
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